Characterization of new, efficient Mycobacterium tuberculosis topoisomerase-I inhibitors and their interaction with human ABC multidrug transporters
Temesszentandrási-Ambrus, Csilla, Tóth, Szilárd, Verma, Rinkee, Bánhegyi, Péter, Szabadkai, István, Baska, Ferenc, Szántai-Kis, Csaba, Hartkoorn, Ruben C, Lingerfelt, Mary A, Sarkadi, Balázs, Szakács, Gergely, Őrfi, László, Nagaraja, Valakunja, Ekins, Sean, Telbisz, Ágnes
Published in PloS one (05.09.2018)
Published in PloS one (05.09.2018)
Get full text
Journal Article
Targeting vascular endothelial growth factor receptor 2 and protein kinase D1 related pathways by a multiple kinase inhibitor in angiogenesis and inflammation related processes in vitro
Varga, Attila, Gyulavári, Pál, Greff, Zoltán, Futosi, Krisztina, Németh, Tamás, Simon-Szabó, Laura, Kerekes, Krisztina, Szántai-Kis, Csaba, Brauswetter, Diána, Kokas, Márton, Borbély, Gábor, Erdei, Anna, Mócsai, Attila, Kéri, György, Vántus, Tibor
Published in PloS one (14.04.2015)
Published in PloS one (14.04.2015)
Get full text
Journal Article
Discovery and Biological Evaluation of Novel Dual EGFR/c-Met Inhibitors
Szokol, Bálint, Gyulavári, Pál, Kurkó, Ibolya, Baska, Ferenc, Szántai-Kis, Csaba, Greff, Zoltán, Őrfi, Zoltán, Peták, István, Pénzes, Kinga, Torka, Robert, Ullrich, Axel, Őrfi, László, Vántus, Tibor, Kéri, György
Published in ACS medicinal chemistry letters (10.04.2014)
Published in ACS medicinal chemistry letters (10.04.2014)
Get full text
Journal Article
Protein kinase inhibitor as a potential candidate for epilepsy treatment
Gajda, Zita, Török, Rita, Horváth, Zoltán, Szántai‐Kis, Csaba, Őrfi, László, Kéri, György, Szente, Magdolna
Published in Epilepsia (Copenhagen) (01.03.2011)
Published in Epilepsia (Copenhagen) (01.03.2011)
Get full text
Journal Article
Discovery and development of extreme selective inhibitors of the ITD and D835Y mutant FLT3 kinases
Baska, Ferenc, Sipos, Anna, Őrfi, Zoltán, Nemes, Zoltán, Dobos, Judit, Szántai-Kis, Csaba, Szabó, Eszter, Szénási, Gábor, Dézsi, László, Hamar, Péter, Cserepes, Mihály T., Tóvári, József, Garamvölgyi, Rita, Krekó, Marcell, Őrfi, László
Published in European journal of medicinal chemistry (15.12.2019)
Published in European journal of medicinal chemistry (15.12.2019)
Get full text
Journal Article
Novel compounds with potent CDK9 inhibitory activity for the treatment of myeloma
Czudor, Zsófia, Balogh, Mária, Bánhegyi, Péter, Boros, Sándor, Breza, Nóra, Dobos, Judit, Fábián, Márk, Horváth, Zoltán, Illyés, Eszter, Markó, Péter, Sipos, Anna, Szántai-Kis, Csaba, Szokol, Bálint, Őrfi, László
Published in Bioorganic & medicinal chemistry letters (15.02.2018)
Published in Bioorganic & medicinal chemistry letters (15.02.2018)
Get full text
Journal Article
Design and synthesis of new imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrazine derivatives with antiproliferative activity against melanoma cells
Garamvölgyi, Rita, Dobos, Judit, Sipos, Anna, Boros, Sándor, Illyés, Eszter, Baska, Ferenc, Kékesi, László, Szabadkai, István, Szántai-Kis, Csaba, Kéri, György, Őrfi, László
Published in European journal of medicinal chemistry (27.01.2016)
Published in European journal of medicinal chemistry (27.01.2016)
Get full text
Journal Article
Synthesis and characterization of amino acid substituted sunitinib analogues for the treatment of AML
Nemes, Zoltán, Takács-Novák, Krisztina, Völgyi, Gergely, Valko, Klara, Béni, Szabolcs, Horváth, Zoltán, Szokol, Bálint, Breza, Nóra, Dobos, Judit, Szántai-Kis, Csaba, Illyés, Eszter, Boros, Sándor, Kok, Robbert Jan, Őrfi, László
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
Get full text
Journal Article
Discovery and optimization of novel benzothiophene-3-carboxamides as highly potent inhibitors of Aurora kinases A and B
Gyulavári, Pál, Szokol, Bálint, Szabadkai, István, Brauswetter, Diána, Bánhegyi, Péter, Varga, Attila, Markó, Péter, Boros, Sándor, Illyés, Eszter, Szántai-Kis, Csaba, Krekó, Marcell, Czudor, Zsófia, Őrfi, László
Published in Bioorganic & medicinal chemistry letters (15.10.2018)
Published in Bioorganic & medicinal chemistry letters (15.10.2018)
Get full text
Journal Article
Leads for antitubercular compounds from kinase inhibitor library screens
Magnet, Sophie, Hartkoorn, Ruben C, Székely, Rita, Pató, János, Triccas, James A, Schneider, Patricia, Szántai-Kis, Csaba, Őrfi, László, Chambon, Marc, Banfi, Damiano, Bueno, Manuel, Turcatti, Gerardo, Kéri, György, Cole, Stewart T
Published in Tuberculosis (Edinburgh, Scotland) (01.11.2010)
Published in Tuberculosis (Edinburgh, Scotland) (01.11.2010)
Get full text
Journal Article
Development of a 3D Tissue Culture–Based High-Content Screening Platform That Uses Phenotypic Profiling to Discriminate Selective Inhibitors of Receptor Tyrosine Kinases
Booij, Tijmen H., Klop, Maarten J. D., Yan, Kuan, Szántai-Kis, Csaba, Szokol, Balint, Orfi, Laszlo, van de Water, Bob, Keri, Gyorgy, Price, Leo S.
Published in Journal of biomolecular screening (01.10.2016)
Published in Journal of biomolecular screening (01.10.2016)
Get full text
Journal Article
Lead selection and characterization of antitubercular compounds using the Nested Chemical Library
Sipos, Anna, Pató, János, Székely, Rita, Hartkoorn, Ruben C, Kékesi, László, Őrfi, László, Szántai-Kis, Csaba, Mikušová, Katarína, Svetlíková, Zuzana, Korduláková, Jana, Nagaraja, Valakunja, Godbole, Adwait Anand, Bush, Natassja, Collin, Frédéric, Maxwell, Anthony, Cole, Stewart T, Kéri, György
Published in Tuberculosis (Edinburgh, Scotland) (01.06.2015)
Published in Tuberculosis (Edinburgh, Scotland) (01.06.2015)
Get full text
Journal Article
Novel compounds reducing IRS-1 serine phosphorylation for treatment of diabetes
Simon-Szabó, Laura, Kokas, Márton, Greff, Zoltán, Boros, Sándor, Bánhegyi, Péter, Zsákai, Lilián, Szántai-Kis, Csaba, Vantus, Tibor, Mandl, József, Bánhegyi, Gábor, Vályi-Nagy, István, Őrfi, László, Ullrich, Axel, Csala, Miklós, Kéri, György
Published in Bioorganic & medicinal chemistry letters (15.01.2016)
Published in Bioorganic & medicinal chemistry letters (15.01.2016)
Get full text
Journal Article
Correction: Targeting Vascular Endothelial Growth Factor Receptor 2 and Protein Kinase D1 Related Pathways by a Multiple Kinase Inhibitor in Angiogenesis and Inflammation Related Processes In Vitro
Varga, Attila, Gyulavári, Pál, Greff, Zoltán, Futosi, Krisztina, Németh, Tamás, Simon-Szabó, Laura, Kerekes, Krisztina, Szántai-Kis, Csaba, Brauswetter, Diána, Kokas, Márton, Borbély, Gábor, Erdei, Anna, Mócsai, Attila, Kéri, György, Vántus, Tibor
Published in PloS one (16.12.2015)
Published in PloS one (16.12.2015)
Get full text
Journal Article
NADPH Oxidase 4 Is Expressed in Pulmonary Artery Adventitia and Contributes to Hypertensive Vascular Remodeling
Barman, Scott A, Chen, Feng, Su, Yunchao, Dimitropoulou, Christiana, Wang, Yusi, Catravas, John D, Han, Weihong, Orfi, Laszlo, Szantai-Kis, Csaba, Keri, Gyorgy, Szabadkai, Istvan, Barabutis, Nektarios, Rafikova, Olga, Rafikov, Ruslan, Black, Stephen M, Jonigk, Danny, Giannis, Athanassios, Asmis, Reto, Stepp, David W, Ramesh, Ganesan, Fulton, David J.R
Published in Arteriosclerosis, thrombosis, and vascular biology (01.08.2014)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.08.2014)
Get full text
Journal Article
Validation subset selections for extrapolation oriented QSPAR models
Szántai-Kis, Csaba, Kövesdi, István, Kéri, György, Orfi, László
Published in Molecular diversity (2003)
Published in Molecular diversity (2003)
Get full text
Journal Article
Targeted drug combination therapy design based on driver genes
Zsákai, Lilian, Sipos, Anna, Dobos, Judit, Erős, Dániel, Szántai-Kis, Csaba, Bánhegyi, Péter, Pató, János, Őrfi, László, Matula, Zsolt, Mikala, Gábor, Kéri, György, Peták, István, Vályi-Nagy, István
Published in Oncotarget (03.09.2019)
Published in Oncotarget (03.09.2019)
Get full text
Journal Article
Tyrosine kinase inhibitors - small molecular weight compounds inhibiting EGFR
Hegymegi-Barakonyi, Bálint, Eros, Dániel, Szántai-Kis, Csaba, Breza, Nóra, Bánhegyi, Péter, Szabó, Gábor Viktor, Várkondi, Edit, Peták, István, Orfi, László, Kéri, György
Published in Current opinion in molecular therapeutics (01.06.2009)
Get more information
Published in Current opinion in molecular therapeutics (01.06.2009)
Journal Article