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Bhattacharyya, Anuradha, Trotta, Christopher R, Narasimhan, Jana, Wiedinger, Kari J, Li, Wencheng, Effenberger, Kerstin A, Woll, Matthew G, Jani, Minakshi B, Risher, Nicole, Yeh, Shirley, Cheng, Yaofeng, Sydorenko, Nadiya, Moon, Young-Choon, Karp, Gary M, Weetall, Marla, Dakka, Amal, Gabbeta, Vijayalakshmi, Naryshkin, Nikolai A, Graci, Jason D, Tripodi, Jr, Thomas, Southwell, Amber, Hayden, Michael, Colacino, Joseph M, Peltz, Stuart W
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Published in Nature communications (15.12.2021)
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Self-renewal as a therapeutic target in human colorectal cancer
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Published in Nature medicine (01.01.2014)
Published in Nature medicine (01.01.2014)
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Evaluating the Mechanism and Therapeutic Potential of PTC-028, a Novel Inhibitor of BMI-1 Function in Ovarian Cancer
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Published in Molecular cancer therapeutics (01.01.2018)
Published in Molecular cancer therapeutics (01.01.2018)
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A Formal [3 + 3] Cycloaddition Approach to Natural-Product Synthesis
Hsung, Richard P., Kurdyumov, Aleksey V., Sydorenko, Nadiya
Published in European journal of organic chemistry (01.01.2005)
Published in European journal of organic chemistry (01.01.2005)
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A Formal [3 + 3] Cycloaddition Reaction. 5. An Enantioselective Intramolecular Formal Aza-[3 + 3] Cycloaddition Reaction Promoted by Chiral Amine Salts
Gerasyuto, Aleksey I, Hsung, Richard P, Sydorenko, Nadiya, Slafer, Brian
Published in Journal of organic chemistry (27.05.2005)
Published in Journal of organic chemistry (27.05.2005)
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Abstract 5517: PTC596-induced Bmi1 hyper-phosphorylation via Cdk1/2 activation resulting in tumor stem cell depletion
Kim, Min Jung, Cao, Liangxian, Sheedy, Josephine, Risher, Nicole, Dumble, Melissa, Lee, Chang-Sun, Sydorenko, Nadiya, Baiazitov, Ramil, Du, Wu, Moon, Young-Choon, Weetall, Marla L., Colacino, Joseph, Davis, Thomas W.
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Unexpected Observation of the Dimroth Rearrangement in the Ribosylation of 4‑Aminopyrimidines
Baiazitov, Ramil Y, Sydorenko, Nadiya, Ren, Hongyu, Moon, Young-Choon
Published in Journal of organic chemistry (02.06.2017)
Published in Journal of organic chemistry (02.06.2017)
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I01 Orally bioavailable small molecule splicing modifiers with systemic and even htt-lowering activity in vitro and in vivo
Bhattacharyya, Anuradha, Effenberger, Kerstin, Trotta, Christopher, Narasimhan, Jana, Li, Wencheng, Woll, Matthew, Jani, Minakshi, Risher, Nicole, Yeh, Shirley, Cheng, Yaofeng, Sydorenko, Nadiya, Weetall, Marla, Southwell, Amber L, Hayden, Michael R, Colacino, Joseph, Peltz, Stuart
Published in Journal of neurology, neurosurgery and psychiatry (01.09.2021)
Published in Journal of neurology, neurosurgery and psychiatry (01.09.2021)
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BMI-1 Targeting Interferes with Patient-Derived Tumor-Initiating Cell Survival and Tumor Growth in Prostate Cancer
Bansal, Nitu, Bartucci, Monica, Yusuff, Shamila, Davis, Stephani, Flaherty, Kathleen, Huselid, Eric, Patrizii, Michele, Jones, Daniel, Cao, Liangxian, Sydorenko, Nadiya, Moon, Young-Choon, Zhong, Hua, Medina, Daniel J, Kerrigan, John, Stein, Mark N, Kim, Isaac Y, Davis, Thomas W, DiPaola, Robert S, Bertino, Joseph R, Sabaawy, Hatem E
Published in Clinical cancer research (15.12.2016)
Published in Clinical cancer research (15.12.2016)
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Discovery and SAR Studies of Potent Modulators of BMI-1 Expression
Baiazitov, Ramil Y., Sydorenko, Nadiya, Du, Wu, Ren, Hongyu, Cao, Liang, Davis, Thomas, Cintron-Lue, Katherine, Kim, Min-Jung, Zhuo, Jin, Mody, Shreshtha, Weetall, Marla, Sheedy, Josephine, Risher, Nicole, Almstead, Neil, Moon, Young-Choon
Published in Helvetica chimica acta (01.09.2023)
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Targeted BMI1 inhibition impairs tumor growth in lung adenocarcinomas with low CEBPα expression
Yong, Kol Jia, Basseres, Daniela S, Welner, Robert S, Zhang, Wen Cai, Yang, Henry, Yan, Benedict, Alberich-Jorda, Meritxell, Zhang, Junyan, de Figueiredo-Pontes, Lorena Lobo, Battelli, Chiara, Hetherington, Christopher J, Ye, Min, Zhang, Hong, Maroni, Giorgia, O'Brien, Karen, Magli, Maria Cristina, Borczuk, Alain C, Varticovski, Lyuba, Kocher, Olivier, Zhang, Pu, Moon, Young-Choon, Sydorenko, Nadiya, Cao, Liangxian, Davis, Thomas W, Thakkar, Bhavin M, Soo, Ross A, Iwama, Atsushi, Lim, Bing, Halmos, Balazs, Neuberg, Donna, Tenen, Daniel G, Levantini, Elena
Published in Science translational medicine (03.08.2016)
Published in Science translational medicine (03.08.2016)
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SYDORENKO NADIYA, JANI MINAKSHI, BABU SURESH, BHATTACHARYYA ANURADHA, MOON YOUNG CHOON, HWANG SEONGWOO
Year of Publication 15.07.2022
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Year of Publication 15.07.2022
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HETEROARYL COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE
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Year of Publication 25.04.2024
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Year of Publication 25.04.2024
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Abstract 2529: Optimization of small molecules targeting BMI1 protein expression. Part 1. Amino-thiazoles: the first-in-class highly potent inhibitors of BMI1 protein
Sydorenko, Nadiya, Baiazitov, Ramil, Choi, Soongyu, Lee, Chang-Sun, Cao, Liangxian, Davis, Thomas W., Almstead, Neil G., Moon, Young-Choon
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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헌팅턴병 치료 화합물
SYDORENKO NADIYA, NARASIMHAN JANA, BABU SURESH, PATEL JIGAR S, BHATTACHARYYA ANURADHA, MOON YOUNG CHOON
Year of Publication 14.01.2021
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Year of Publication 14.01.2021
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Year of Publication 20.05.2024
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Year of Publication 20.05.2024
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Abstract 2528: Optimization of small molecules targeting BMI1 protein expression. Part 2. Improved potency, oral bioavailability, and in vivo efficacy of amino-pyrazines and amino-pyridines
Baiazitov, Ramil, Sydorenko, Nadiya, Ren, Hongyu, Du, Wu, Paget, Steve, Wilde, Richard, Liu, Ronggang, Lee, Chang-Sun, Cao, Liangxian, Davis, Thomas W., Almstead, Neil G., Moon, Young-Choon
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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1 SUBSTITUTED REVERSE PYRIMIDINE BMI-1 INHIBITORS
SYDORENKO NADIYA, REN HONGYU, CAO LIANGXIAN, PAGET STEVEN D, BAIAZITOV RAMIL, MOON YOUNG CHOON, LEE CHANG SUN, WILDE RICHARD GERALD, LIU RONGGANG, DAVIS THOMAS W, DU WU
Year of Publication 24.10.2022
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Year of Publication 24.10.2022
Patent
1 SUBSTITUTED REVERSE PYRIMIDINE BMI-1 INHIBITORS
SYDORENKO NADIYA, REN HONGYU, CAO LIANGXIAN, PAGET STEVEN D, BAIAZITOV RAMIL, MOON YOUNG CHOON, LEE CHANG SUN, WILDE RICHARD GERALD, LIU RONGGANG, DAVIS THOMAS W, DU WU
Year of Publication 08.02.2022
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Year of Publication 08.02.2022
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