Discovery of a Potent and Orally Active Hedgehog Pathway Antagonist (IPI-926)
Tremblay, Martin R, Lescarbeau, André, Grogan, Michael J, Tan, Eddy, Lin, Grace, Austad, Brian C, Yu, Lin-Chen, Behnke, Mark L, Nair, Somarajan J, Hagel, Margit, White, Kerry, Conley, James, Manna, Joseph D, Alvarez-Diez, Teresa M, Hoyt, Jennifer, Woodward, Caroline N, Sydor, Jens R, Pink, Melissa, MacDougall, John, Campbell, Matthew J, Cushing, Jill, Ferguson, Jeanne, Curtis, Michael S, McGovern, Karen, Read, Margaret A, Palombella, Vito J, Adams, Julian, Castro, Alfredo C
Published in Journal of medicinal chemistry (23.07.2009)
Published in Journal of medicinal chemistry (23.07.2009)
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Journal Article
Development of 17-Allylamino-17-Demethoxygeldanamycin Hydroquinone Hydrochloride (IPI-504), an Anti-Cancer Agent Directed against Hsp90
Sydor, Jens R., Normant, Emmanuel, Pien, Christine S., Porter, James R., Ge, Jie, Grenier, Louis, Pak, Roger H., Ali, Janid A., Dembski, Marlene S., Hudak, Jebecka, Patterson, Jon, Penders, Courtney, Pink, Melissa, Read, Margaret A., Sang, Jim, Woodward, Caroline, Zhang, Yilong, Grayzel, David S., Wright, Jim, Barrett, John A., Palombella, Vito J., Adams, Julian, Tong, Jeffrey K.
Published in Proceedings of the National Academy of Sciences - PNAS (14.11.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (14.11.2006)
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Journal Article
Design, Synthesis, and Biological Evaluation of Hydroquinone Derivatives of 17-Amino-17-demethoxygeldanamycin as Potent, Water-Soluble Inhibitors of Hsp90
Ge, Jie, Normant, Emmanuel, Porter, James R, Ali, Janid A, Dembski, Marlene S, Gao, Yun, Georges, Asimina T, Grenier, Louis, Pak, Roger H, Patterson, Jon, Sydor, Jens R, Tibbitts, Thomas T, Tong, Jeffrey K, Adams, Julian, Palombella, Vito J
Published in Journal of medicinal chemistry (27.07.2006)
Published in Journal of medicinal chemistry (27.07.2006)
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Journal Article
Transient Kinetic Studies on the Interaction of Ras and the Ras-Binding Domain of c-Raf-1 Reveal Rapid Equilibration of the Complex
Sydor, Jens R, Engelhard, Martin, Wittinghofer, Alfred, Goody, Roger S, Herrmann, Christian
Published in Biochemistry (Easton) (06.10.1998)
Published in Biochemistry (Easton) (06.10.1998)
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Journal Article
Perspective on high-throughput bioanalysis to support in vitro assays in early drug discovery
Santiago, Brandon G, Eisennagel, Stephen H, Peckham, Gregory E, Liebhardt, Amanda M, Alburn, Chad L, Roethke, Theresa J, Reilly, Michael A, Sydor, Jens R, Karlinsey, Molly Z
Published in Bioanalysis (01.02.2023)
Published in Bioanalysis (01.02.2023)
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Journal Article
Semisynthetic Cyclopamine Analogues as Potent and Orally Bioavailable Hedgehog Pathway Antagonists
Tremblay, Martin R, Nevalainen, Marta, Nair, Somarajan J, Porter, James R, Castro, Alfredo C, Behnke, Mark L, Yu, Lin-Chen, Hagel, Margit, White, Kerry, Faia, Kerrie, Grenier, Louis, Campbell, Matthew J, Cushing, Jill, Woodward, Caroline N, Hoyt, Jennifer, Foley, Michael A, Read, Margaret A, Sydor, Jens R, Tong, Jeffrey K, Palombella, Vito J, McGovern, Karen, Adams, Julian
Published in Journal of medicinal chemistry (13.11.2008)
Published in Journal of medicinal chemistry (13.11.2008)
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Journal Article
Design, Total Chemical Synthesis, and Binding Properties of a [Leu-91-N1-methyl-7-azaTrp]Ras-Binding Domain of c-Raf-1
Sydor, Jens R., Herrmann, Christian, Stephen B. H. Kent, Goody, Roger S., Engelhard, Martin
Published in Proceedings of the National Academy of Sciences - PNAS (06.07.1999)
Published in Proceedings of the National Academy of Sciences - PNAS (06.07.1999)
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Journal Article
The Photophobic Receptor from Natronobacterium pharaonis: Temperature and pH Dependencies of the Photocycle of Sensory Rhodopsin II
Chizhov, Igor, Schmies, Georg, Seidel, Ralf, Sydor, Jens R., Lüttenberg, Beate, Engelhard, Martin
Published in Biophysical journal (01.08.1998)
Published in Biophysical journal (01.08.1998)
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Journal Article
Chip-Based Analysis of Protein−Protein Interactions by Fluorescence Detection and On-Chip Immunoprecipitation Combined with μLC−MS/MS Analysis
Sydor, Jens R, Scalf, Mark, Sideris, Steve, Mao, Guo Dong, Pandey, Yash, Tan, Ming, Mariano, Maria, Moran, Michael F, Nock, Steffen, Wagner, Peter
Published in Analytical chemistry (Washington) (15.11.2003)
Published in Analytical chemistry (Washington) (15.11.2003)
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Journal Article
Cell-free synthesis of the Ras-binding domain of c-Raf-1: binding studies to fluorescently labelled H-Ras
Sydor, Jens R, Seidel, Ralf P, Goody, Roger S, Engelhard, Martin
Published in FEBS letters (11.06.1999)
Published in FEBS letters (11.06.1999)
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Journal Article
Chip-based analysis of protein-protein interactions by fluorescence detection and on-chip immunoprecipitation combined with microLC-MS/MS analysis
Sydor, Jens R, Scalf, Mark, Sideris, Steve, Mao, Guo Dong, Pandey, Yash, Tan, Ming, Mariano, Maria, Moran, Michael F, Nock, Steffen, Wagner, Peter
Published in Analytical chemistry (Washington) (15.11.2003)
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Published in Analytical chemistry (Washington) (15.11.2003)
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