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Towards natural mimetics of metformin and rapamycin
Aliper, Alexander, Jellen, Leslie, Cortese, Franco, Artemov, Artem, Karpinsky-Semper, Darla, Moskalev, Alexey, Swick, Andrew G, Zhavoronkov, Alex
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The effects of oral administration of curcumin-galactomannan complex on brain waves are consistent with brain penetration: a randomized, double-blinded, placebo-controlled pilot study
Khanna, Aman, Das S, Syam, Kannan, R., Swick, Andrew G., Matthewman, Cristina, Maliakel, Balu, Ittiyavirah, Sibi P., Krishnakumar, I. M.
Published in Nutritional neuroscience (03.06.2022)
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In search for geroprotectors: in silico screening and in vitro validation of signalome-level mimetics of young healthy state
Aliper, Alexander, Belikov, Aleksey V, Garazha, Andrew, Jellen, Leslie, Artemov, Artem, Suntsova, Maria, Ivanova, Alena, Venkova, Larisa, Borisov, Nicolas, Buzdin, Anton, Mamoshina, Polina, Putin, Evgeny, Swick, Andrew G, Moskalev, Alexey, Zhavoronkov, Alex
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Published in Aging (Albany, NY.) (24.09.2016)
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Enhanced bioavailability and pharmacokinetics of a novel hybrid-hydrogel formulation of fisetin orally administered in healthy individuals: a randomised double-blinded comparative crossover study
Krishnakumar, Illathu Madhavamenon, Jaja-Chimedza, Asha, Joseph, Ashil, Balakrishnan, Abhilash, Maliakel, Balu, Swick, Andrew
Published in Journal of nutritional science (Cambridge) (2022)
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The effects of an SPM-enriched marine oil and bioavailable curcumin combination on inflammation-associated discomfort in generally healthy individuals: a virtual open-label pilot study
Jaja-Chimedza, Asha, Hirsh, Steven, Bruce, Dainian, Bou-Sliman, Tony, Joyal, Steven, Swick, Andrew G.
Published in Translational medicine communications (14.11.2022)
Published in Translational medicine communications (14.11.2022)
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CP-809,101, a selective 5-HT2C agonist, shows activity in animal models of antipsychotic activity
Siuciak, Judith A, Chapin, Douglas S, McCarthy, Sheryl A, Guanowsky, Victor, Brown, Janice, Chiang, Phoebe, Marala, Ravi, Patterson, Terrell, Seymour, Patricia A, Swick, Andrew, Iredale, Philip A
Published in Neuropharmacology (01.02.2007)
Published in Neuropharmacology (01.02.2007)
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Leptin potentiates the anti-obesity effects of rimonabant
Boustany-Kari, Carine M., Jackson, V. Margaret, Gibbons, Colleen P., Swick, Andrew G.
Published in European journal of pharmacology (11.05.2011)
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Identification and characterization of a leptin-responsive neuroblastoma cell line
Wang, Ruduan, Swick, Andrew G.
Published in Biochemical and biophysical research communications (20.02.2009)
Published in Biochemical and biophysical research communications (20.02.2009)
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Role of leptin in fat regulation
Collins, Sheila, Kuhn, Cysnthia M, Petro, Ann E, Swick, Andrew G, Chrunyk, Boris A, Surwit, Richard S
Published in Nature (London) (25.04.1996)
Published in Nature (London) (25.04.1996)
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Discovery of microsomal triglyceride transfer protein (MTP) inhibitors with potential for decreased active metabolite load compared to dirlotapide
Robinson, Ralph P., Bartlett, Jeremy A., Bertinato, Peter, Bessire, Andrew J., Cosgrove, Judith, Foley, Patrick M., Manion, Tara B., Minich, Martha L., Ramos, Brenda, Reese, Matthew R., Schmahai, Theodore J., Swick, Andrew G., Tess, David A., Vaz, Alfin, Wolford, Angela
Published in Bioorganic & medicinal chemistry letters (15.07.2011)
Published in Bioorganic & medicinal chemistry letters (15.07.2011)
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Discovery of new piperidine amide triazolobenzodiazepinones as intestinal-selective CCK1 receptor agonists
Cameron, Kimberly O., Beretta, Elena E., Chen, Yue, Chu-Moyer, Margaret, Fernando, Dilinie, Gao, Hua, Kohrt, Jeffrey, Lavergne, Sophie, Jardine, Paul Da Silva, Guzman-Perez, Angel, Hoth, Christopher, Perry, David A., Hadcock, John R., Gautreau, Denise, Makowski, Michael, Perez, Sylvie, Polivkova, Jana, Rogers, Lucy, Scott, Dennis O., Swick, Andrew G., Thiede, Lucinda, Trebino, Catherine E., Trilles, Richard V., Wilmowski, Julie, Zhang, Yingxin
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
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Discovery of N-benzyl-2-[(4S)-4-(1H-indol-3-ylmethyl)-5-oxo-1-phenyl-4,5-dihydro-6H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-6-yl]-N-isopropylacetamide, an orally active, gut-selective CCK1 receptor agonist for the potential treatment of obesity
Elliott, Richard L., Cameron, Kimberly O., Chin, Janice E., Bartlett, Jeremy A., Beretta, Elena E., Chen, Yue, Jardine, Paul Da Silva, Dubins, Jeffrey S., Gillaspy, Melissa L., Hargrove, Diane M., Kalgutkar, Amit S., LaFlamme, Janet A., Lame, Mary E., Martin, Kelly A., Maurer, Tristan S., Nardone, Nancy A., Oliver, Robert M., Scott, Dennis O., Sun, Dexue, Swick, Andrew G., Trebino, Catherine E., Zhang, Yingxin
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
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