Fragment-based discovery of potent inhibitors of the anti-apoptotic MCL-1 protein
Petros, Andrew M., Swann, Steven L., Song, Danying, Swinger, Kerren, Park, Chang, Zhang, Haichao, Wendt, Michael D., Kunzer, Aaron R., Souers, Andrew J., Sun, Chaohong
Published in Bioorganic & medicinal chemistry letters (15.03.2014)
Published in Bioorganic & medicinal chemistry letters (15.03.2014)
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Journal Article
Development of Orally Efficacious Allosteric Inhibitors of TNFα via Fragment-Based Drug Design
Dietrich, Justin D, Longenecker, Kenton L, Wilson, Noel S, Goess, Christian, Panchal, Sanjay C, Swann, Steven L, Petros, Andrew M, Hobson, Adrian D, Ihle, David, Song, Danying, Richardson, Paul, Comess, Kenneth M, Cox, Philip B, Dombrowski, Amanda, Sarris, Kathy, Donnelly-Roberts, Diana L, Duignan, David B, Gomtsyan, Arthur, Jung, Paul, Krueger, A Chris, Mathieu, Suzanne, McClure, Andrea, Stoll, Vincent S, Wetter, Jill, Mankovich, John A, Hajduk, Philip J, Vasudevan, Anil, Stoffel, Robert H, Sun, Chaohong
Published in Journal of medicinal chemistry (14.01.2021)
Published in Journal of medicinal chemistry (14.01.2021)
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Journal Article
Design of Aminobenzothiazole Inhibitors of Rho Kinases 1 and 2 by Using Protein Kinase A as a Structure Surrogate
Judge, Russell A., Vasudevan, Anil, Scott, Victoria E., Simler, Gricelda H., Pratt, Steve D., Namovic, Marian T., Putman, C. Brent, Aguirre, Ana, Stoll, Vincent S., Mamo, Mulugeta, Swann, Steven I., Cassar, Steven C., Faltynek, Connie R., Kage, Karen L., Boyce‐Rustay, Janel M., Hobson, Adrian D.
Published in Chembiochem : a European journal of chemical biology (16.03.2018)
Published in Chembiochem : a European journal of chemical biology (16.03.2018)
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Journal Article
Corrigendum: Design of Aminobenzothiazole Inhibitors of Rho Kinases 1 and 2 by Using Protein Kinase A as a Structure Surrogate
Judge, Russell A., Vasudevan, Anil, Scott, Victoria E., Simler, Gricelda H., Pratt, Steve D., Namovic, Marian T., Putman, C. Brent, Aguirre, Ana, Stoll, Vincent S., Mamo, Mulugeta, Swann, Steven I., Cassar, Steven C., Faltynek, Connie R., Kage, Karen L., Boyce‐Rustay, Janel M., Hobson, Adrian D.
Published in Chembiochem : a European journal of chemical biology (16.04.2018)
Published in Chembiochem : a European journal of chemical biology (16.04.2018)
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Journal Article
Labeled Ligand Displacement: Extending NMR-Based Screening of Protein Targets
Swann, Steven L, Song, Danying, Sun, Chaohong, Hajduk, Philip J, Petros, Andrew M
Published in ACS medicinal chemistry letters (09.09.2010)
Published in ACS medicinal chemistry letters (09.09.2010)
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Journal Article
Critical Aspartic Acid Residues in Pseudouridine Synthases
Ramamurthy, V, Swann, S L, Paulson, J L, Spedaliere, C J, Mueller, E G
Published in The Journal of biological chemistry (06.08.1999)
Published in The Journal of biological chemistry (06.08.1999)
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Journal Article
Structure-guided optimization of a novel class of ASK1 inhibitors with increased sp(3) character and an exquisite selectivity profile
Bigi-Botterill, Simone V., Ivetac, Anthony, Bradshaw, Erica L., Cole, Derek, Dougan, Douglas R., Ermolieff, Jacques, Halkowycz, Petro, Johnson, Ben, McBride, Christopher, Pickens, Jason, Sabat, Mark, Swann, Steven
Published in Bioorganic & medicinal chemistry letters (01.09.2020)
Published in Bioorganic & medicinal chemistry letters (01.09.2020)
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Journal Article
Role of Cysteine Residues in Pseudouridine Synthases of Different Families
Ramamurthy, Vidhyashankar, Swann, Steven L, Spedaliere, Christopher J, Mueller, Eugene G
Published in Biochemistry (Easton) (05.10.1999)
Published in Biochemistry (Easton) (05.10.1999)
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Journal Article
Structure-based drug design of novel ASK1 inhibitors using an integrated lead optimization strategy
Gibson, Tony S., Johnson, Benjamin, Fanjul, Andrea, Halkowycz, Petro, Dougan, Douglas R., Cole, Derek, Swann, Steven
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
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Journal Article
Structure-guided optimization of a novel class of ASK1 inhibitors with increased sp3 character and an exquisite selectivity profile
Bigi-Botterill, Simone V., Ivetac, Anthony, Bradshaw, Erica L., Cole, Derek, Dougan, Douglas R., Ermolieff, Jacques, Halkowycz, Petro, Johnson, Ben, McBride, Christopher, Pickens, Jason, Sabat, Mark, Swann, Steven
Published in Bioorganic & medicinal chemistry letters (01.09.2020)
Published in Bioorganic & medicinal chemistry letters (01.09.2020)
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Journal Article
Conditional Recommendations for Specific Dietary Ingredients as an Approach to Chronic Musculoskeletal Pain: Evidence-Based Decision Aid for Health Care Providers, Participants, and Policy Makers
Boyd, Courtney, Crawford, Cindy, Berry, Kevin, Deuster, Patricia
Published in Pain medicine (Malden, Mass.) (01.07.2019)
Published in Pain medicine (Malden, Mass.) (01.07.2019)
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Journal Article
Mind–Body Therapies for the Self‐Management of Chronic Pain Symptoms
Lee, Courtney, Crawford, Cindy, Hickey, Anita, Buckenmaier, Chester C., Crawford, Cindy, Crawford, Paul, Delgado, Roxana, Freilich, Daniel, Hickey, Anita, Jonas, Wayne B., Lee, Courtney, May, Todd, Petri, Richard P., Schoomaker, Eric B., Spevak, Christopher, Swann, Steven, York, Alexandra
Published in Pain medicine (Malden, Mass.) (01.04.2014)
Published in Pain medicine (Malden, Mass.) (01.04.2014)
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Journal Article
Abstract LB-A20: True small molecule STING agonist generates systemic and potent anti-tumor immunity required for effective cancer immunotherapy
Kulkarni, Meghana M, Dwight, Timothy, Marino, Kristen, Allen, Bryce K, Taimi, Mohammed, Bastos, Cecilia, Lai, Sujen, Koh, Cheryl, Samant, Ramya, Tesar, Bethany, Huang, Huang, Chamberlain, Brian, Rice, James M, Tan, Dazhi, Lin, Zhixiong, Shechter, Sharon, Li, Stella, Sparks, Sam, Soutter, Holly, Swann, Steven, Sherman, Woody, Winter, Christopher
Published in Molecular cancer therapeutics (01.12.2019)
Published in Molecular cancer therapeutics (01.12.2019)
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Journal Article
Multimodal, Integrative Therapies for the Self‐Management of Chronic Pain Symptoms
Lee, Courtney, Crawford, Cindy, Swann, Steven, Buckenmaier, Chester C., Crawford, Cindy, Crawford, Paul, Delgado, Roxana, Freilich, Daniel, Hickey, Anita, Jonas, Wayne B., Lee, Courtney, May, Todd, Petri, Richard P., Schoomaker, Eric B., Spevak, Christopher, Swann, Steven, York, Alexandra
Published in Pain medicine (Malden, Mass.) (01.04.2014)
Published in Pain medicine (Malden, Mass.) (01.04.2014)
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