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Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (Tiagabine) as an anticonvulsant drug candidate
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Published in Journal of medicinal chemistry (01.06.1993)
Published in Journal of medicinal chemistry (01.06.1993)
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Synthesis of Novel GABA Uptake Inhibitors. 4. Bioisosteric Transformation and Successive Optimization of Known GABA Uptake Inhibitors Leading to a Series of Potent Anticonvulsant Drug Candidates
Andersen, Knud Erik, Sørensen, Jan L, Huusfeldt, Per O, Knutsen, Lars J. S, Lau, Jesper, Lundt, Behrend F, Petersen, Hans, Suzdak, Peter D, Swedberg, Michael D. B
Published in Journal of medicinal chemistry (21.10.1999)
Published in Journal of medicinal chemistry (21.10.1999)
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Neurotrophic Immunophilin Ligands Stimulate Structural and Functional Recovery in Neurodegenerative Animal Models
Steiner, Joseph P., Hamilton, Gregory S., Ross, Douglas T., Valentine, Heather L., Guo, Hongzhi, Connolly, Maureen A., Liang, Shi, Ramsey, Cynthia, Li, Jia-He J., Huang, Wei, Howorth, Pamela, Soni, Rajat, Fuller, Michael, Sauer, Hans, Nowotnik, Alison C., Suzdak, Peter D.
Published in Proceedings of the National Academy of Sciences - PNAS (04.03.1997)
Published in Proceedings of the National Academy of Sciences - PNAS (04.03.1997)
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Synthesis of Novel γ-Aminobutyric Acid (GABA) Uptake Inhibitors. 5. Preparation and Structure−Activity Studies of Tricyclic Analogues of Known GABA Uptake Inhibitors
Andersen, Knud Erik, Sørensen, Jan L, Lau, Jesper, Lundt, Behrend F, Petersen, Hans, Huusfeldt, Per O, Suzdak, Peter D, Swedberg, Michael D. B
Published in Journal of medicinal chemistry (21.06.2001)
Published in Journal of medicinal chemistry (21.06.2001)
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Synthesis of novel GABA uptake inhibitors. Part 6 : Preparation and evaluation of N-Ω asymmetrically substituted nipecotic acid derivatives
ANDERSEN, Knud Erik, LAU, Jesper, LUNDT, Behrend F, PETERSEN, Hans, HUUSFELDT, Per O, SUZDAK, Peter D, SWEDBERG, Michael D. B
Published in Bioorganic & medicinal chemistry (01.11.2001)
Published in Bioorganic & medicinal chemistry (01.11.2001)
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Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor
Nielsen, E B, Suzdak, P D, Andersen, K E, Knutsen, L J, Sonnewald, U, Braestrup, C
Published in European journal of pharmacology (24.04.1991)
Published in European journal of pharmacology (24.04.1991)
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Butylthio[2.2.2] (NNC 11â1053/LY297802): An Orally Active Muscarinic Agonist Analgesic
Swedberg, M D, Sheardown, M J, Sauerberg, P, Olesen, P H, Suzdak, P D, Hansen, K T, Bymaster, F P, Ward, J S, Mitch, C H, Calligaro, D O, Delapp, N W, Shannon, H E
Published in The Journal of pharmacology and experimental therapeutics (01.05.1997)
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Published in The Journal of pharmacology and experimental therapeutics (01.05.1997)
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Pharmacology of Butylthio[2.2.2] (LY297802/NNC11-1053): A Novel Analgesic with Mixed Muscarinic Receptor Agonist and Antagonist Activity
Shannon, H E, Sheardown, M J, Bymaster, F P, Calligaro, D O, Delapp, N W, Gidda, J, Mitch, C H, Sawyer, B D, Stengel, P W, Ward, J S, Wong, D T, Olesen, P H, Suzdak, P D, Sauerberg, P, Swedberg, M D
Published in The Journal of pharmacology and experimental therapeutics (01.05.1997)
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Published in The Journal of pharmacology and experimental therapeutics (01.05.1997)
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Effects of bromohomoibotenate on metabotropic glutamate receptors
Thomsen, C, Bau, A, Faarup, P, Foged, C, Kanstrup, A, Suzdak, P D
Published in Neuroreport (20.12.1994)
Published in Neuroreport (20.12.1994)
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Is ethanol antagonist Ro15-4513 selective for ethanol?
Britton, K T, Ehlers, C L, Koob, G F
Published in Science (American Association for the Advancement of Science) (05.02.1988)
Published in Science (American Association for the Advancement of Science) (05.02.1988)
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Effects of t-ACPD on neural survival and second messengers in cultured cerebral cortical neurones
Thomsen, C, Frandsen, A, Suzdak, P D, Andersen, C F, Schousboe, A
Published in Neuroreport (10.09.1993)
Published in Neuroreport (10.09.1993)
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Actions of phenylglycine analogs at subtypes of the metabotropic glutamate receptor family
Thomsen, Christian, Boel, Esper, Suzdak, Peter D.
Published in European journal of pharmacology (15.03.1994)
Published in European journal of pharmacology (15.03.1994)
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L-2-amino-4-phosphonobutyrate (L-AP4) is an agonist at the type IV metabotropic glutamate receptor which is negatively coupled to adenylate cyclase
Thomsen, C, Kristensen, P, Mulvihill, E, Haldeman, B, Suzdak, P D
Published in European journal of pharmacology (02.11.1992)
Published in European journal of pharmacology (02.11.1992)
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