Discovery of PF-06873600, a CDK2/4/6 Inhibitor for the Treatment of Cancer
Freeman-Cook, Kevin D, Hoffman, Robert L, Behenna, Douglas C, Boras, Britton, Carelli, Jordan, Diehl, Wade, Ferre, Rose Ann, He, You-Ai, Hui, Andrea, Huang, Buwen, Huser, Nanni, Jones, Rhys, Kephart, Susan E, Lapek, John, McTigue, Michele, Miller, Nichol, Murray, Brion W, Nagata, Asako, Nguyen, Lisa, Niessen, Sherry, Ninkovic, Sacha, O’Doherty, Inish, Ornelas, Martha A, Solowiej, James, Sutton, Scott C, Tran, Khanh, Tseng, Elaine, Visswanathan, Ravi, Xu, Meirong, Zehnder, Luke, Zhang, Qin, Zhang, Cathy, Dann, Stephen
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
Get full text
Journal Article
Multifaceted Substrate–Ligand Interactions Promote the Copper-Catalyzed Hydroboration of Benzylidenecyclobutanes and Related Compounds
Kang, Taeho, Erbay, Tuğçe G, Xu, Kane L, Gallego, Gary M, Burtea, Alexander, Nair, Sajiv K, Patman, Ryan L, Zhou, Ru, Sutton, Scott C, McAlpine, Indrawan J, Liu, Peng, Engle, Keary M
Published in ACS catalysis (06.11.2020)
Published in ACS catalysis (06.11.2020)
Get full text
Journal Article
Synthesis of Aryl Ethers via a Sulfonyl Transfer Reaction
Sach, Neal W, Richter, Daniel T, Cripps, Stephan, Tran-Dubé, Michelle, Zhu, Huichun, Huang, Buwen, Cui, Jean, Sutton, Scott C
Published in Organic letters (03.08.2012)
Published in Organic letters (03.08.2012)
Get full text
Journal Article
Practical Singly and Doubly Electrophilic Aminating Agents: A New, More Sustainable Platform for Carbon–Nitrogen Bond Formation
Kattamuri, Padmanabha V, Yin, Jun, Siriwongsup, Surached, Kwon, Doo-Hyun, Ess, Daniel H, Li, Qun, Li, Guigen, Yousufuddin, Muhammed, Richardson, Paul F, Sutton, Scott C, Kürti, László
Published in Journal of the American Chemical Society (16.08.2017)
Published in Journal of the American Chemical Society (16.08.2017)
Get full text
Journal Article
Design and Characterization of a Pyridone-Containing EZH2 Inhibitor Phosphate Prodrug
Kung, Pei-Pei, Fan, Connie, Gukasyan, Hovhannes J, Huang, Buwen, Kephart, Susan, Kraus, Manfred, Lee, Joseph H, Sutton, Scott C, Yamazaki, Shinji, Zehnder, Luke
Published in Journal of medicinal chemistry (11.02.2021)
Published in Journal of medicinal chemistry (11.02.2021)
Get full text
Journal Article
Twinning behavior and lattice rotation in a Mg–Gd–Y–Zr alloy under ballistic impact
Shi, Xiaoying, Luo, Alan A., Sutton, Scott C., Zeng, Long, Wang, Shiyi, Zeng, Xiaoqin, Li, Dejiang, Ding, Wenjiang
Published in Journal of alloys and compounds (25.11.2015)
Published in Journal of alloys and compounds (25.11.2015)
Get full text
Journal Article
Application of Biocatalytic Reductive Amination for the Synthesis of a Key Intermediate to a CDK 2/4/6 Inhibitor
Duan, Shengquan, Widlicka, Daniel W, Burns, Michael P, Kumar, Rajesh, Hotham, Ian, Desrosiers, Jean-Nicolas, Bowles, Paul, Jones, Kris N, Nicholson, Lindsay D, Buetti-Weekly, Michele T, Han, Lu, Steflik, Jeremy, Hansen, Eric, Hayward, Cheryl M, Strohmeyer, Holly, Monfette, Sébastien, Sutton, Scott C, Morris, Christopher
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
Get full text
Journal Article
Correction to “Practical Singly and Doubly Electrophilic Aminating Agents: A New, More Sustainable Platform for Carbon–Nitrogen Bond Formation”
Kattamuri, Padmanabha V, Yin, Jun, Siriwongsup, Surached, Kwon, Doo-Hyun, Ess, Daniel H, Li, Qun, Li, Guigen, Yousufuddin, Muhammed, Richardson, Paul F, Sutton, Scott C, Kürti, László
Published in Journal of the American Chemical Society (20.02.2019)
Published in Journal of the American Chemical Society (20.02.2019)
Get full text
Journal Article
Synthesis of oxetane-3-carboxaldehyde and methyl oxetane-3-carboxylate via homologation of oxetane-3-one
Kephart, Susan E., Zehnder, Luke R., Huang, Buwen, Sutton, Scott C.
Published in Tetrahedron (30.06.2016)
Published in Tetrahedron (30.06.2016)
Get full text
Journal Article
Pfizer Global Virtual Library (PGVL): A Chemistry Design Tool Powered by Experimentally Validated Parallel Synthesis Information
Hu, Qiyue, Peng, Zhengwei, Sutton, Scott C, Na, Jim, Kostrowicki, Jaroslav, Yang, Bo, Thacher, Thomas, Kong, Xianjun, Mattaparti, Sarathy, Zhou, Joe Zhongxiang, Gonzalez, Javier, Ramirez-Weinhouse, Michele, Kuki, Atsuo
Published in ACS combinatorial science (12.11.2012)
Published in ACS combinatorial science (12.11.2012)
Get full text
Journal Article
Synthesis of Novel 2-Cyano-7-deaza-8-azapurine- and 2-Cyano-8-azapurine-Derived Nucleosides
Wainwright, Philip, Maddaford, Adrian, Simms, Michael, Forrest, Neil, Glen, Rebecca, Hart, James, Zhang, Xiurong, Pryde, David C., Stephenson, Peter T., Middleton, Donald S., Guyot, Thierry, Sutton, Scott C.
Published in Synlett (01.08.2011)
Published in Synlett (01.08.2011)
Get more information
Journal Article
Biomimetic Total Syntheses of (+)-Cephalostatin 7, (+)-Cephalostatin 12, and (+)-Ritterazine K
Jeong, Jae Uk, Sutton, Scott C, Kim, Seongkon, Fuchs, P. L
Published in Journal of the American Chemical Society (01.10.1995)
Published in Journal of the American Chemical Society (01.10.1995)
Get full text
Journal Article
Development of a Cost-Efficient Process Toward a Key Synthetic Intermediate of the EZH2 Inhibitor PF-06821497
Ashcroft, Christopher P., Berne, Alexander M., Blasberg, Florian, Catlin, Kelly, Collins, Michael R., Critcher, Doug J., Desrosiers, Jean-Nicolas, Goetz, Adam, Hayward, Cheryl, Jones, Ricky A., Karmilowicz, Michael J., Keene, Nandell, Martinez, Carlos A., Monfette, Sebastien, Pattavina, Sebastian David, Perfect, Hahdi H., Ragan, John A., Rauschenberger, Blake, Sach, Neal W., Scotney, Gemma, Sutton, Scott C., Talicska, Courtney, Twiddle, Steven J.R., Haitsma, Jared Van, Wisdom, Richard
Published in Organic process research & development (21.06.2024)
Published in Organic process research & development (21.06.2024)
Get full text
Journal Article
Synthesis of the North 1 Unit of the Cephalostatin Family from Hecogenin Acetate1
Kim, Seongkon, Sutton, Scott C, Guo, Chuangxing, LaCour, Thomas G, Fuchs, P. L
Published in Journal of the American Chemical Society (17.03.1999)
Published in Journal of the American Chemical Society (17.03.1999)
Get full text
Journal Article