Absorption, distribution, metabolism and excretion of novel phosphodiesterase type 4 inhibitor ASP3258 in rats
Ohtsu, Yoshiaki, Sonoda, Takuya, Susaki, Yoko, Tohda, Toshifumi, Fukunaga, Yasuhisa, Iwatsubo, Takafumi, Noguchi, Kiyoshi
Published in Biopharmaceutics & drug disposition (01.01.2015)
Published in Biopharmaceutics & drug disposition (01.01.2015)
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Inhibitory effect of a novel non-steroidal aromatase inhibitor, YM511 on the proliferation of MCF-7 human breast cancer cell
Kudoh, Masafumi, Susaki, Yoko, Ideyama, Yukitaka, Nanya, Taiki, Mori, Masamichi, Shikama, Hisataka, Fujikura, Takashi
Published in The Journal of steroid biochemistry and molecular biology (01.05.1996)
Published in The Journal of steroid biochemistry and molecular biology (01.05.1996)
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STRUCTURE AND MUTAGENICITY OF A DIRECT-ACTING MUTAGEN DERIVED FROM THE REACTION OF N-NITROSO-N-METHYLBUTYLAMINE WITH HYDROXYL RADICAL
Inami, Keiko, Miura, Motofumi, Tsutsumi, Nozomi, Okochi, Eriko, Susaki, Yoko, Ishikawa, Satoko, Motohashi, Shigeyasu, Shiino, Junko, Takeda, Kei, Mochizuki, Masataka
Published in Heterocycles (01.01.2012)
Published in Heterocycles (01.01.2012)
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YM116, 2-(1H-Imidazol-4-ylmethyl)-9H-carbazole, Decreases Adrenal Androgen Synthesis by Inhibiting C17-20 Lyase Activity in NCI-H295 Human Adrenocortical Carcinoma Cells
Ideyama, Yukitaka, Kudoh, Masafumi, Tanimoto, Kyoko, Susaki, Yoko, Nanya, Taiki, Nakahara, Takahito, Ishikawa, Hiroko, Fujikura, Takashi, Akaza, Hideyuki, Shikama, Hisataka
Published in Japanese Journal of Pharmacology (1999)
Published in Japanese Journal of Pharmacology (1999)
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Inhibitory effects of a novel aromatase inhibitor, YM511, on growth of endometrial explants and insulin-like growth factor-I gene expression in rats with experimental endometriosis
Kudoh, Masafumi, Susaki, Yoko, Ideyama, Yukitaka, Nanya, Taiki, Mori, Masamichi, Shikama, Hisataka
Published in The Journal of steroid biochemistry and molecular biology (01.09.1997)
Published in The Journal of steroid biochemistry and molecular biology (01.09.1997)
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The potent and selective inhibition of estrogen production by non-steroidal aromatase inhibitor, YM511
Kudoh, Masafumi, Susaki, Yoko, Ideyama, Yukitaka, Nanya, Taiki, Okada, Minoru, Shikama, Hisataka, Fujikura, Takashi
Published in The Journal of steroid biochemistry and molecular biology (01.09.1995)
Published in The Journal of steroid biochemistry and molecular biology (01.09.1995)
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Novel nonsteroidal inhibitor of cytochrome P45017α (17α-hydroxylase/C17-20 lyase), YM116, decreased prostatic weights by reducing serum concentrations of testosterone and adrenal androgens in rats
Ideyama, Yukitaka, Kudoh, Masafumi, Tanimoto, Kyoko, Susaki, Yoko, Nanya, Taiki, Nakahara, Takahito, Ishikawa, Hiroko, Yoden, Toru, Okada, Minoru, Fujikura, Takashi, Akaza, Hideyuki, Shikama, Hisataka
Published in The Prostate (15.09.1998)
Published in The Prostate (15.09.1998)
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A novel aromatase inhibitor, YM511
Ideyama, Yukitaka, Nan'ya, Taiki, Susaki, Yoko, Kudo, Masafumi, Abe, Tetsushi, Okada, Minoru, Kawaminami, Eiji, Isomura, Yasuo, Fujikura, Takashi, Takenaka, Toichi
Published in Japanese journal of pharmacology (1993)
Published in Japanese journal of pharmacology (1993)
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