Fluorescent ligands for adenosine receptors
Kozma, Eszter, Suresh Jayasekara, P., Squarcialupi, Lucia, Paoletta, Silvia, Moro, Stefano, Federico, Stephanie, Spalluto, Giampiero, Jacobson, Kenneth A.
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
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Journal Article
Synthesis, Characterization, and Direct Intracellular Imaging of Ultrasmall and Uniform Glutathione-Coated Gold Nanoparticles
Sousa, Alioscka A., Morgan, Jeffrey T., Brown, Patrick H., Adams, April, Jayasekara, M. P. Suresh, Zhang, Guofeng, Ackerson, Christopher J., Kruhlak, Michael J., Leapman, Richard D.
Published in Small (Weinheim an der Bergstrasse, Germany) (23.07.2012)
Published in Small (Weinheim an der Bergstrasse, Germany) (23.07.2012)
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Journal Article
A selective high-affinity antagonist of the P2Y14 receptor inhibits UDP-glucose-stimulated chemotaxis of human neutrophils
Barrett, Matthew O, Sesma, Juliana I, Ball, Christopher B, Jayasekara, P Suresh, Jacobson, Kenneth A, Lazarowski, Eduardo R, Harden, T Kendall
Published in Molecular pharmacology (01.07.2013)
Published in Molecular pharmacology (01.07.2013)
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Journal Article
John Daly Lecture: Structure-guided Drug Design for Adenosine and P2Y Receptors
Jacobson, Kenneth A, Gao, Zhan-Guo, Paoletta, Silvia, Kiselev, Evgeny, Chakraborty, Saibal, Jayasekara, P Suresh, Balasubramanian, Ramachandran, Tosh, Dilip K
Published in Computational and structural biotechnology journal (01.01.2015)
Published in Computational and structural biotechnology journal (01.01.2015)
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Journal Article
Assessing the impact of expert knowledge on ICH M7 (Q)SAR predictions. Is expert review still needed?
Jayasekara, P. Suresh, Skanchy, Sophie K., Kim, Marlene T., Kumaran, Govindaraj, Mugabe, Benon E., Woodard, Lauren E., Yang, Jian, Zych, Andrew J., Kruhlak, Naomi L.
Published in Regulatory toxicology and pharmacology (01.10.2021)
Published in Regulatory toxicology and pharmacology (01.10.2021)
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Journal Article
AMP-activated protein kinase as regulator of P2Y(6) receptor-induced insulin secretion in mouse pancreatic β-cells
Balasubramanian, Ramachandran, Maruoka, Hiroshi, Jayasekara, P Suresh, Gao, Zhan-Guo, Jacobson, Kenneth A
Published in Biochemical pharmacology (01.04.2013)
Published in Biochemical pharmacology (01.04.2013)
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Journal Article
P2Y2 receptor agonist with enhanced stability protects the heart from ischemic damage in vitro and in vivo
Hochhauser, Edith, Cohen, Ronit, Waldman, Maayan, Maksin, Anna, Isak, Ahuva, Aravot, Dan, Jayasekara, P. Suresh, Müller, Christa E., Jacobson, Kenneth A., Shainberg, Asher
Published in Purinergic signalling (01.12.2013)
Published in Purinergic signalling (01.12.2013)
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Journal Article
4‑Alkyloxyimino Derivatives of Uridine-5′-triphosphate: Distal Modification of Potent Agonists as a Strategy for Molecular Probes of P2Y2, P2Y4, and P2Y6 Receptors
Jayasekara, P. Suresh, Barrett, Matthew O, Ball, Christopher B, Brown, Kyle A, Hammes, Eva, Balasubramanian, Ramachandran, Harden, T. Kendall, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (08.05.2014)
Published in Journal of medicinal chemistry (08.05.2014)
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Journal Article
The role of P2Y14 and other P2Y receptors in degranulation of human LAD2 mast cells
Gao, Zhan-Guo, Wei, Qiang, Jayasekara, M. P. Suresh, Jacobson, Kenneth A.
Published in Purinergic signalling (01.03.2013)
Published in Purinergic signalling (01.03.2013)
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Journal Article
4-Alkyloxyimino-cytosine nucleotides: tethering approaches to molecular probes for the P2Y6 receptor
Jayasekara, P. Suresh, Barrett, Matthew O., Ball, Christopher B., Brown, Kyle A., Kozma, Eszter, Costanzi, Stefano, Squarcialupi, Lucia, Balasubramanian, Ramachandran, Maruoka, Hiroshi, Jacobson, Kenneth A.
Published in MedChemComm (30.05.2013)
Published in MedChemComm (30.05.2013)
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Journal Article
Modulation of G protein-coupled adenosine receptors by strategically functionalized agonists and antagonists immobilized on gold nanoparticles
Jayasekara, P. Suresh, Phan, Khai, Tosh, Dilip K., Kumar, T. Santhosh, Moss, Steven M., Zhang, Guofeng, Barchi, Joseph J., Gao, Zhan-Guo, Jacobson, Kenneth A.
Published in Purinergic signalling (01.06.2013)
Published in Purinergic signalling (01.06.2013)
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Journal Article
The role of P2Y(14) and other P2Y receptors in degranulation of human LAD2 mast cells
Gao, Zhan-Guo, Wei, Qiang, Jayasekara, M P Suresh, Jacobson, Kenneth A
Published in Purinergic signalling (01.03.2013)
Published in Purinergic signalling (01.03.2013)
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Journal Article
Pyrimidine Nucleotides with 4-Alkyloxyimino and Terminal Tetraphosphate delta-Ester Modifications as Selective Agonists of the P2Y(4) Receptor
Maruoka, Hiroshi, Jayasekara, M. P. Suresh, Barrett, Matthew O., Franklin, Derek A., de Castro, Sonia, Kim, Nathaniel, Costanzi, Stefano, Harden, T. Kendall, Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (23.06.2011)
Published in Journal of medicinal chemistry (23.06.2011)
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