Ligand design by targeting a binding site water
Matricon, Pierre, Suresh, R. Rama, Gao, Zhan-Guo, Panel, Nicolas, Jacobson, Kenneth A, Carlsson, Jens
Published in Chemical science (Cambridge) (19.11.2020)
Published in Chemical science (Cambridge) (19.11.2020)
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Journal Article
Pathophysiological Role and Medicinal Chemistry of A2A Adenosine Receptor Antagonists in Alzheimer’s Disease
Merighi, Stefania, Borea, Pier Andrea, Varani, Katia, Vincenzi, Fabrizio, Travagli, Alessia, Nigro, Manuela, Pasquini, Silvia, Suresh, R. Rama, Kim, Sung Won, Volkow, Nora D., Jacobson, Kenneth A., Gessi, Stefania
Published in Molecules (Basel, Switzerland) (21.04.2022)
Published in Molecules (Basel, Switzerland) (21.04.2022)
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Journal Article
Exploring allene chemistry using phosphorus-based allenes as scaffolds
Swamy, K. C. Kumara, Anitha, Mandala, Gangadhararao, G., Rama Suresh, R.
Published in Pure and applied chemistry (01.03.2017)
Published in Pure and applied chemistry (01.03.2017)
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Journal Article
Pharmacological characterization of DPTN and other selective A3 adenosine receptor antagonists
Gao, Zhan-Guo, Suresh, R. Rama, Jacobson, Kenneth A.
Published in Purinergic signalling (01.12.2021)
Published in Purinergic signalling (01.12.2021)
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Journal Article
Expanding the repertoire of methanocarba nucleosides from purinergic signaling to diverse targets
Jacobson, Kenneth A, Salmaso, Veronica, Suresh, R. Rama, Tosh, Dilip K
Published in MedChemComm (17.11.2021)
Published in MedChemComm (17.11.2021)
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Journal Article
Design and in vivo activity of A3 adenosine receptor agonist prodrugs
Suresh, R. Rama, Jain, Shanu, Chen, Zhoumou, Tosh, Dilip K., Ma, Yanling, Podszun, Maren C., Rotman, Yaron, Salvemini, Daniela, Jacobson, Kenneth A.
Published in Purinergic signalling (01.09.2020)
Published in Purinergic signalling (01.09.2020)
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Journal Article
Fluorescent A2A and A3 adenosine receptor antagonists as flow cytometry probes
Toti, Kiran S., Campbell, Ryan G., Lee, Hobin, Salmaso, Veronica, Suresh, R. Rama, Gao, Zhan-Guo, Jacobson, Kenneth A.
Published in Purinergic signalling (01.09.2023)
Published in Purinergic signalling (01.09.2023)
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Journal Article
Convergent synthesis of 2-thioether-substituted ()-methanocarba-adenosines as purine receptor agonists
Suresh, R. Rama, Poe, Russell B, Lin, Baorui, Lv, Kexin, Campbell, Ryan G, Gao, Zhan-Guo, Liston, Theodore E, Toti, Kiran S, Jacobson, Kenneth A
Published in RSC advances (09.08.2021)
Published in RSC advances (09.08.2021)
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Journal Article
Nucleotide P2Y1 receptor agonists are in vitro and in vivo prodrugs of A1/A3 adenosine receptor agonists: implications for roles of P2Y1 and A1/A3 receptors in physiology and pathology
Liston, Theodore E., Hinz, Sonja, Müller, Christa E., Holstein, Deborah M., Wendling, Jay, Melton, Roger J., Campbell, Mary, Korinek, William S., Suresh, R. Rama, Sethre-Hofstad, Dane A., Gao, Zhan-Guo, Tosh, Dilip K., Jacobson, Kenneth A., Lechleiter, James D.
Published in Purinergic signalling (01.12.2020)
Published in Purinergic signalling (01.12.2020)
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Journal Article
Activation of adenosine A2A or A2B receptors causes hypothermia in mice
Carlin, Jesse Lea, Jain, Shalini, Duroux, Romain, Suresh, R. Rama, Xiao, Cuiying, Auchampach, John A., Jacobson, Kenneth A., Gavrilova, Oksana, Reitman, Marc L.
Published in Neuropharmacology (01.09.2018)
Published in Neuropharmacology (01.09.2018)
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Journal Article
Allosteric Antagonism of the A2A Adenosine Receptor by a Series of Bitopic Ligands
Gao, Zhan-Guo, Toti, Kiran S., Campbell, Ryan, Suresh, R. Rama, Yang, Huijun, Jacobson, Kenneth A.
Published in Cells (Basel, Switzerland) (12.05.2020)
Published in Cells (Basel, Switzerland) (12.05.2020)
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Journal Article
Molecularly Nonstoichiometric Crystals in Phosphorus Compounds
Chakravarty, Manab, Rama Suresh, R, Kumara Swamy, K. C
Published in Inorganic chemistry (12.11.2007)
Published in Inorganic chemistry (12.11.2007)
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Journal Article
Lipid Trolling to Optimize A3 Adenosine Receptor-Positive Allosteric Modulators (PAMs)
Pradhan, Balaram, Pavan, Matteo, Fisher, Courtney L., Salmaso, Veronica, Wan, Tina C., Keyes, Robert F., Rollison, Noah, Suresh, R. Rama, Kumar, T. Santhosh, Gao, Zhan-Guo, Smith, Brian C., Auchampach, John A., Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Journal Article
Structure–Activity Studies of 1H‑Imidazo[4,5‑c]quinolin-4-amine Derivatives as A3 Adenosine Receptor Positive Allosteric Modulators
Fallot, Lucas B., Suresh, R. Rama, Fisher, Courtney L., Salmaso, Veronica, O’Connor, Robert D., Kaufman, Noy, Gao, Zhan-Guo, Auchampach, John A., Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (24.11.2022)
Published in Journal of medicinal chemistry (24.11.2022)
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Journal Article
Structure-Activity Studies of 1 H -Imidazo[4,5- c ]quinolin-4-amine Derivatives as A 3 Adenosine Receptor Positive Allosteric Modulators
Fallot, Lucas B, Suresh, R Rama, Fisher, Courtney L, Salmaso, Veronica, O'Connor, Robert D, Kaufman, Noy, Gao, Zhan-Guo, Auchampach, John A, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (24.11.2022)
Published in Journal of medicinal chemistry (24.11.2022)
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Journal Article
Activation of adenosine A 2A or A 2B receptors causes hypothermia in mice
Carlin, Jesse Lea, Jain, Shalini, Duroux, Romain, Suresh, R Rama, Xiao, Cuiying, Auchampach, John A, Jacobson, Kenneth A, Gavrilova, Oksana, Reitman, Marc L
Published in Neuropharmacology (01.09.2018)
Published in Neuropharmacology (01.09.2018)
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Journal Article
A2A adenosine receptor agonists, antagonists, inverse agonists and partial agonists
Jacobson, Kenneth A, Suresh, R Rama, Oliva, Paola
Published in International review of neurobiology (01.01.2023)
Published in International review of neurobiology (01.01.2023)
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Journal Article
2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A 1 Adenosine Receptor Positive Allosteric Modulators
Oliva, Paola, Suresh, R Rama, Pasquini, Silvia, Salmaso, Veronica, Will, Edward J, Tosh, Dilip K, Gao, Zhan-Guo, Liu, Naili, Gavrilova, Oksana, Vincenzi, Fabrizio, Varani, Katia, Jacobson, Kenneth A
Published in ACS medicinal chemistry letters (14.12.2023)
Published in ACS medicinal chemistry letters (14.12.2023)
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Journal Article