Comparative genotypic and phenotypic analysis of human peripheral blood monocytes and surrogate monocyte-like cell lines commonly used in metabolic disease research
Riddy, Darren M, Goy, Emily, Delerive, Philippe, Summers, Roger J, Sexton, Patrick M, Langmead, Christopher J
Published in PloS one (10.05.2018)
Published in PloS one (10.05.2018)
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Journal Article
The actions of relaxin on the human cardiovascular system
Sarwar, Mohsin, Du, Xiao‐Jun, Dschietzig, Thomas B, Summers, Roger J
Published in British journal of pharmacology (01.05.2017)
Published in British journal of pharmacology (01.05.2017)
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Journal Article
International Union of Basic and Clinical Pharmacology. XCV. Recent advances in the understanding of the pharmacology and biological roles of relaxin family peptide receptors 1-4, the receptors for relaxin family peptides
Halls, Michelle L, Bathgate, Ross A D, Sutton, Steve W, Dschietzig, Thomas B, Summers, Roger J
Published in Pharmacological reviews (01.04.2015)
Published in Pharmacological reviews (01.04.2015)
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Journal Article
Allosteric ligands of the glucagon-like peptide 1 receptor (GLP-1R) differentially modulate endogenous and exogenous peptide responses in a pathway-selective manner: implications for drug screening
Koole, Cassandra, Wootten, Denise, Simms, John, Valant, Celine, Sridhar, Rohan, Woodman, Owen L, Miller, Laurence J, Summers, Roger J, Christopoulos, Arthur, Sexton, Patrick M
Published in Molecular pharmacology (01.09.2010)
Published in Molecular pharmacology (01.09.2010)
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Journal Article
Adrenoceptors—New roles for old players
Michel, Martin C., Bond, Richard A., Summers, Roger J.
Published in British journal of pharmacology (01.07.2019)
Published in British journal of pharmacology (01.07.2019)
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Journal Article
Evolution of β-blockers: from anti-anginal drugs to ligand-directed signalling
Baker, Jillian G, Hill, Stephen J, Summers, Roger J
Published in Trends in pharmacological sciences (Regular ed.) (01.04.2011)
Published in Trends in pharmacological sciences (Regular ed.) (01.04.2011)
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Journal Article
Murine GPRC6A Mediates Cellular Responses to L-Amino Acids, but Not Osteocalcin Variants
Rueda, Patricia, Harley, Elizabeth, Lu, Yao, Stewart, Gregory D, Fabb, Stewart, Diepenhorst, Natalie, Cremers, Béatrice, Rouillon, Marie-Hélène, Wehrle, Isabelle, Geant, Anne, Lamarche, Gwladys, Leach, Katie, Charman, William N, Christopoulos, Arthur, Summers, Roger J, Sexton, Patrick M, Langmead, Christopher J
Published in PloS one (19.01.2016)
Published in PloS one (19.01.2016)
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Journal Article
Antifibrotic Actions of Serelaxin – New Roles for an Old Player
Samuel, Chrishan S, Summers, Roger J, Hewitson, Tim D
Published in Trends in pharmacological sciences (Regular ed.) (01.06.2016)
Published in Trends in pharmacological sciences (Regular ed.) (01.06.2016)
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Journal Article
Relaxin requires the angiotensin II type 2 receptor to abrogate renal interstitial fibrosis
Chow, Bryna S. Man, Kocan, Martina, Bosnyak, Sanja, Sarwar, Mohsin, Wigg, Belinda, Jones, Emma S., Widdop, Robert E., Summers, Roger J., Bathgate, Ross A.D., Hewitson, Tim D., Samuel, Chrishan S.
Published in Kidney international (01.07.2014)
Published in Kidney international (01.07.2014)
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Journal Article
Multipathway In Vitro Pharmacological Characterization of Specialized Proresolving G Protein-Coupled Receptors
Merlin, Jon, Park, Julia, Vandekolk, Teresa H, Fabb, Stewart A, Allinne, Jeanne, Summers, Roger J, Langmead, Christopher J, Riddy, Darren M
Published in Molecular pharmacology (01.04.2022)
Published in Molecular pharmacology (01.04.2022)
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Journal Article
Improving type 2 diabetes through a distinct adrenergic signaling pathway involving mTORC2 that mediates glucose uptake in skeletal muscle
Sato, Masaaki, Dehvari, Nodi, Oberg, Anette I, Dallner, Olof S, Sandström, Anna L, Olsen, Jessica M, Csikasz, Robert I, Summers, Roger J, Hutchinson, Dana S, Bengtsson, Tore
Published in Diabetes (New York, N.Y.) (01.12.2014)
Published in Diabetes (New York, N.Y.) (01.12.2014)
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Journal Article
Ligand‐directed signalling at β‐adrenoceptors
Evans, Bronwyn A., Sato, Masaaki, Sarwar, Mohsin, Hutchinson, Dana S., Summers, Roger J.
Published in British journal of pharmacology (01.03.2010)
Published in British journal of pharmacology (01.03.2010)
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Journal Article
The PPARγ agonist rosiglitazone promotes the induction of brite adipocytes, increasing β-adrenoceptor-mediated mitochondrial function and glucose uptake
Merlin, Jon, Sato, Masaaki, Nowell, Cameron, Pakzad, Mohsen, Fahey, Richard, Gao, Jie, Dehvari, Nodi, Summers, Roger J., Bengtsson, Tore, Evans, Bronwyn A., Hutchinson, Dana S.
Published in Cellular signalling (01.01.2018)
Published in Cellular signalling (01.01.2018)
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Journal Article
Divergent effects of strontium and calcium‐sensing receptor positive allosteric modulators (calcimimetics) on human osteoclast activity
Diepenhorst, Natalie A, Leach, Katie, Keller, Andrew N, Rueda, Patricia, Cook, Anna E, Pierce, Tracie L, Nowell, Cameron, Pastoureau, Philippe, Sabatini, Massimo, Summers, Roger J, Charman, William N, Sexton, Patrick M, Christopoulos, Arthur, Langmead, Christopher J
Published in British journal of pharmacology (01.11.2018)
Published in British journal of pharmacology (01.11.2018)
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Journal Article
ML290 is a biased allosteric agonist at the relaxin receptor RXFP1
Kocan, Martina, Sarwar, Mohsin, Ang, Sheng Y, Xiao, Jingbo, Marugan, Juan J, Hossain, Mohammed A, Wang, Chao, Hutchinson, Dana S, Samuel, Chrishan S, Agoulnik, Alexander I, Bathgate, Ross A D, Summers, Roger J
Published in Scientific reports (07.06.2017)
Published in Scientific reports (07.06.2017)
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Journal Article
Factors influencing biased agonism in recombinant cells expressing the human α1A‐adrenoceptor
Silva Junior, Edilson Dantas, Sato, Masaaki, Merlin, Jon, Broxton, Natalie, Hutchinson, Dana S, Ventura, Sabatino, Evans, Bronwyn A, Summers, Roger J
Published in British journal of pharmacology (01.07.2017)
Published in British journal of pharmacology (01.07.2017)
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Journal Article
AT1R-AT2R-RXFP1 Functional Crosstalk in Myofibroblasts: Impact on the Therapeutic Targeting of Renal and Cardiac Fibrosis
Chow, Bryna S M, Kocan, Martina, Shen, Matthew, Wang, Yan, Han, Lei, Chew, Jacqueline Y, Wang, Chao, Bosnyak, Sanja, Mirabito-Colafella, Katrina M, Barsha, Giannie, Wigg, Belinda, Johnstone, Elizabeth K M, Hossain, Mohammed A, Pfleger, Kevin D G, Denton, Kate M, Widdop, Robert E, Summers, Roger J, Bathgate, Ross A D, Hewitson, Tim D, Samuel, Chrishan S
Published in Journal of the American Society of Nephrology (01.11.2019)
Published in Journal of the American Society of Nephrology (01.11.2019)
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Journal Article