Improving the in Vitro Prediction of in Vivo Central Nervous System Penetration: Integrating Permeability, P-glycoprotein Efflux, and Free Fractions in Blood and Brain
Summerfield, Scott G, Stevens, Alexander J, Cutler, Leanne, del Carmen Osuna, Maria, Hammond, Beverley, Tang, Sac-Pham, Hersey, Ann, Spalding, David J, Jeffrey, Phil
Published in The Journal of pharmacology and experimental therapeutics (01.03.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2006)
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Inhibition of colonic motility and defecation by RS‐127445 suggests an involvement of the 5‐HT 2B receptor in rodent large bowel physiology
Bassil, AK, Taylor, CM, Bolton, VJN, Gray, KM, Brown, JD, Cutler, L, Summerfield, SG, Bruton, G, Winchester, WJ, Lee, K, Sanger, GJ
Published in British journal of pharmacology (01.09.2009)
Published in British journal of pharmacology (01.09.2009)
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Journal Article
Influence of Secondary Structure on the Fragmentation of Protonated Peptides
Tsaprailis, George, Nair, Hari, Somogyi, Árpád, Wysocki, Vicki H, Zhong, Wenqing, Futrell, Jean H, Summerfield, Scott G, Gaskell, Simon J
Published in Journal of the American Chemical Society (09.06.1999)
Published in Journal of the American Chemical Society (09.06.1999)
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Journal Article
Characterization of three diaminopyrimidines as potent and selective antagonists of P2X3 and P2X2/3 receptors with in vivo efficacy in a pain model
Ballini, E, Virginio, C, Medhurst, SJ, Summerfield, SG, Aldegheri, L, Buson, A, Carignani, C, Chen, YH, Giacometti, A, Lago, I, Powell, AJ, Jarolimek, W
Published in British journal of pharmacology (01.07.2011)
Published in British journal of pharmacology (01.07.2011)
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Investigation into the role of P2X(3)/P2X(2/3) receptors in neuropathic pain following chronic constriction injury in the rat: an electrophysiological study
Sharp, Caroline J, Reeve, Alison J, Collins, Sue D, Martindale, Jo C, Summerfield, Scott G, Sargent, Becky S, Bate, Simon T, Chessell, Iain P
Published in British journal of pharmacology (01.07.2006)
Published in British journal of pharmacology (01.07.2006)
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Journal Article
Inhibition of colonic motility and defecation by RS‐127445 suggests an involvement of the 5‐HT2B receptor in rodent large bowel physiology
Bassil, AK, Taylor, CM, Bolton, VJN, Gray, KM, Brown, JD, Cutler, L, Summerfield, SG, Bruton, G, Winchester, WJ, Lee, K, Sanger, GJ
Published in British journal of pharmacology (01.09.2009)
Published in British journal of pharmacology (01.09.2009)
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Journal Article
Novel HY peptide antigens presented by HLA-B27
Simmons, WA, Summerfield, SG, Roopenian, DC, Slaughter, CA, Zuberi, AR, Gaskell, SJ, Bordoli, RS, Hoyes, J, Moomaw, CR, Colbert, RA, Leong, LY, Butcher, GW, Hammer, RE, Taurog, JD
Published in The Journal of immunology (1950) (15.09.1997)
Published in The Journal of immunology (1950) (15.09.1997)
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Journal Article
Novel HY peptide antigens presented by HLA-B27
Taurog, J D, Hammer, R E, Moomaw, C R, Slaughter, C A, Roopenian, D C, Zuberi, A R, Gaskell, S J, Bordoli, R S, Colbert, R A, Butcher, G W, Leong, L Y
Published in The Journal of immunology (1950) (15.11.1999)
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Published in The Journal of immunology (1950) (15.11.1999)
Journal Article
A New MHC Locus That Influences Class I Peptide Presentation
Simmons, William A, Roopenian, Derry C, Summerfield, Scott G, Jones, Richard C, Galocha, Begoña, Christianson, Gregory J, Maika, Shanna D, Zhou, Ming, Gaskell, Simon J, Bordoli, Robert S, Ploegh, Hidde L, Slaughter, Clive A, Lindahl, Kirsten Fischer, Hammer, Robert E, Taurog, Joel D
Published in Immunity (Cambridge, Mass.) (01.11.1997)
Published in Immunity (Cambridge, Mass.) (01.11.1997)
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Synthetic and mass spectral fragmentation studies on trisubstituted 2H-pyran-2-ones and comparative EIMS behaviour of biologically active 3,5-disubstituted pyrazoles and isoxazoles
Parmar, VS, Jain, SC, Jha, A, Kumar, N, Kumar, A, Vats, A, Jha, HN, Mukherjee, S, Singh, SK, Jennings, KR, Summerfield, SG, Errington, W, Olsen, CE
Published in Indian journal of chemistry. Sect. B. Organic chemistry, including medicinal chemistry (01.10.1997)
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Published in Indian journal of chemistry. Sect. B. Organic chemistry, including medicinal chemistry (01.10.1997)
Journal Article
Intra-ionic interactions in electrosprayed peptide ions
Summerfield, Scott G., Whiting, Andrew, Gaskell, Simon J.
Published in International journal of mass spectrometry and ion processes (01.03.1997)
Published in International journal of mass spectrometry and ion processes (01.03.1997)
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