Inhibition of DNA topoisomerase I activity and induction of apoptosis by thiazacridine derivatives
Barros, Francisco W.A., Bezerra, Daniel P., Ferreira, Paulo M.P., Cavalcanti, Bruno C., Silva, Teresinha G., Pitta, Marina G.R., de Lima, Maria do C.A., Galdino, Suely L., Pitta, Ivan da R., Costa-Lotufo, Letícia V., Moraes, Manoel O., Burbano, Rommel R., Guecheva, Temenouga N., Henriques, João A.P., Pessoa, Cláudia
Published in Toxicology and applied pharmacology (01.04.2013)
Published in Toxicology and applied pharmacology (01.04.2013)
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Effect of chronic treatment with Rosiglitazone on Leydig cell steroidogenesis in rats: in vivo and ex vivo studies
Couto, Janaína A, Saraiva, Karina L A, Barros, Cleiton D, Udrisar, Daniel P, Peixoto, Christina A, Vieira, Juliany S B César, Lima, Maria C, Galdino, Suely L, Pitta, Ivan R, Wanderley, Maria I
Published in Reproductive biology and endocrinology (09.02.2010)
Published in Reproductive biology and endocrinology (09.02.2010)
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GQ-16, a Novel Peroxisome Proliferator-activated Receptor γ (PPARγ) Ligand, Promotes Insulin Sensitization without Weight Gain
Amato, Angélica A., Rajagopalan, Senapathy, Lin, Jean Z., Carvalho, Bruno M., Figueira, Ana C.M., Lu, Jenny, Ayers, Stephen D., Mottin, Melina, Silveira, Rodrigo L., Souza, Paulo C.T., Mourão, Rosa H.V., Saad, Mário J.A., Togashi, Marie, Simeoni, Luiz A., Abdalla, Dulcinéia S.P., Skaf, Munir S., Polikparpov, Igor, Lima, Maria C.A., Galdino, Suely L., Brennan, Richard G., Baxter, John D., Pitta, Ivan R., Webb, Paul, Phillips, Kevin J., Neves, Francisco A.R.
Published in The Journal of biological chemistry (10.08.2012)
Published in The Journal of biological chemistry (10.08.2012)
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New imidazolidinic bioisosters: potential candidates for antischistosomal drugs
Pitta, Maira G R, Silva, Andréa C A, Neves, Juliana Kelle A L, Silva, Poliana G, Irmão, João I, Malagueño, Elizabeth, Santana, José V, Lima, Maria C A, Galdino, Suely L, Pitta, Ivan R, Albuquerque, Mônica C P A
Published in Memórias do Instituto Oswaldo Cruz (01.10.2006)
Published in Memórias do Instituto Oswaldo Cruz (01.10.2006)
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Photodynamic antimicrobial chemotherapy (PACT) using phenothiazine derivatives as photosensitizers against Leishmania braziliensis
Barbosa, Artur F., Sangiorgi, Bruno B., Galdino, Suely L., Barral-Netto, Manoel, Pitta, Ivan R., Pinheiro, Antônio L.
Published in Lasers in surgery and medicine (01.12.2012)
Published in Lasers in surgery and medicine (01.12.2012)
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Chemical synthesis, docking studies and biological effects of a pan peroxisome proliferator-activated receptor agonist and cyclooxygenase inhibitor
Santin, José Roberto, Uchôa, Flávia D.T., Lima, Maria do Carmo A., Rabello, Marcelo M., Machado, Isabel Daufenback, Hernandes, Marcelo Z., Amato, Angelica A., Milton, Flora Aparecida, Webb, Paul, Neves, Francisco de Assis Rocha, Galdino, Suely L., Pitta, Ivan Rocha, Farsky, Sandra H.P.
Published in European journal of pharmaceutical sciences (12.03.2013)
Published in European journal of pharmaceutical sciences (12.03.2013)
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A theoretical study of red-shifting and blue-shifting hydrogen bonds occurring between imidazolidine derivatives and PEG/PVP polymers
Oliveira, Boaz G., Lima, Maria C. A., Pitta, Ivan R., Galdino, Suely L., Hernandes, Marcelo Z.
Published in Journal of molecular modeling (2010)
Published in Journal of molecular modeling (2010)
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Effect of thiazolidine LPSF SF29 on the growth and morphology of Trypanosoma cruzi
de B. Moreira, Thiago Luiz, Barbosa, Artur F.S, Veiga-Santos, Phercyles, Henriques, Cristina, Henriques-Pons, Andrea, Galdino, Suely L, de Lima, Maria do Carmo A, Pitta, Ivan da R, de Souza, Wanderley, de Carvalho, Tecia Maria U
Published in International journal of antimicrobial agents (01.02.2013)
Published in International journal of antimicrobial agents (01.02.2013)
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Enhanced Antiproliferative Activity of the New Anticancer Candidate LPSF/AC04 in Cyclodextrin Inclusion Complexes Encapsulated into Liposomes
Mendonça, Elisângela A. M., Lira, Mariane C. B., Rabello, Marcelo M., Cavalcanti, Isabella M. F., Galdino, Suely L., Pitta, Ivan R., do Carmo A. Lima, Maria, Pitta, Maira G. R., Hernandes, Marcelo Z., Santos-Magalhães, Nereide S.
Published in AAPS PharmSciTech (01.12.2012)
Published in AAPS PharmSciTech (01.12.2012)
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Preliminary antifungal and cytotoxic evaluation of synthetic cycloalkyl[b]thiophene derivatives with PLS-DA analysis
Souza, Beatriz, De Oliveira, Tiago, Aquino, Thiago, de Lima, Maria, Pitta, Ivan, Galdino, Suely, Lima, Edeltrudes, Gonçalves-Silva, Teresinha, Militão, Gardênia, Scotti, Luciana, Scotti, Marcus, Mendonça, Francisco
Published in Acta pharmaceutica (Zagreb, Croatia) (01.06.2012)
Published in Acta pharmaceutica (Zagreb, Croatia) (01.06.2012)
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Reduction of carrageenan-induced acute pulmonary inflammation in mice by novel thiazolidinedione derivative LPSF/RA-4
Barbosa, Karla P.S., Santos, Laise A.M., Ribeiro, Edlene L., Fragoso, Ingrid T., Rocha, Sura W.S., Nunes, Ana K.S., França, Maria E.R., Silva, Bruna S., Silva, Amanda K.S.e., Donato, Mariana A.M., Gomes, Fabiana O.S., Silva, Teresinha G., Pitta, Ivan R., Pitta, Marina R., Lima, Maria C.A., Uchôa, Flávia D.T., Galdino, Suely L., Peixoto, Christina A.
Published in European journal of pharmacology (15.10.2013)
Published in European journal of pharmacology (15.10.2013)
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Solid Dispersions of Imidazolidinedione by PEG and PVP Polymers with Potential Antischistosomal Activities
Guedes, Francimary L., de Oliveira, Boaz G., Hernandes, Marcelo Z., De Simone, Carlos A., Veiga, Francisco J. B., de Lima, Maria do Carmo A., Pitta, Ivan R., Galdino, Suely L., Neto, Pedro José Rolim
Published in AAPS PharmSciTech (01.03.2011)
Published in AAPS PharmSciTech (01.03.2011)
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Anti-atherogenic and anti-inflammatory effects of novel thiazolidine-2,4-diones in RAW 264.7 macrophages and in low-density lipoprotein receptor-deficient mice
César, Fernanda A, Rudnicki, Martina, Saito, Cristiane A.I, Galdino, Suely L, Pitta, Ivan R, Lima, Maria C.A, Abdalla, Dulcineia S.P
Published in Vascular pharmacology (01.05.2012)
Published in Vascular pharmacology (01.05.2012)
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Anti-inflammatory and proangiogenic properties of new thiazolidinedione in endothelial cells
Rudnicki, Martina, Fuchigami, Fernando S, Saito, Cristiane A.I, César, Fernanda A, Lima, Maria C.A, Galdino, Suely L, Pitta, Ivan R, Abdalla, Dulcineia S.P
Published in Vascular pharmacology (01.05.2012)
Published in Vascular pharmacology (01.05.2012)
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Development and validation of an LC-UV method for quantification of a new thiazolidinedione (LPSF/AC-23) with antitumor activity in rat plasma
Valério, Raphael D., Silva, Ricardo M., Cunha, Hellencléia P., Lima, Maria C. A., Galdino, Suely L., Pitta, Ivan R., Maia, Maria Bernadete S.
Published in Journal of the Brazilian Chemical Society (01.11.2012)
Published in Journal of the Brazilian Chemical Society (01.11.2012)
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Development and validation of an HPLC/MS/MS method for determining the thiazolidinone PG15 in rat plasma
Uchôa, Flávia D T, Palma, Eduardo C, Souza, Natalia F, Lima, Maria C A, Galdino, Suely L, Pitta, Ivan R, Dalla Costa, Teresa
Published in Journal of AOAC International (01.07.2010)
Published in Journal of AOAC International (01.07.2010)
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2-(2-Nitroanilino)-4,5,6,7-tetrahydrobenzo[ b ]thiophene-3-carbonitrile
Mendonça Junior, Francisco J.B., Lima, Maria do Carmo A. de, Galdino, Suely L., Pitta, Ivan R., Simone, Carlos A. de
Published in Acta crystallographica. Section E, Structure reports online (01.10.2010)
Published in Acta crystallographica. Section E, Structure reports online (01.10.2010)
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Synthesis of 4-octyl-2H-1,4-benzo-thiazin-3-ones
Guarda, VLD, Perrissin, M, Thomasson, F, Ximenes, EA, Galdino, SL, Pitta, IR, Luu-Duc, C, Barbe, J
Published in European journal of medicinal chemistry (01.07.2003)
Published in European journal of medicinal chemistry (01.07.2003)
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