Targeting Transcriptional Enhanced Associate Domains (TEADs)
Gibault, Floriane, Sturbaut, Manon, Bailly, Fabrice, Melnyk, Patricia, Cotelle, Philippe
Published in Journal of medicinal chemistry (28.06.2018)
Published in Journal of medicinal chemistry (28.06.2018)
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Design of a Cereblon construct for crystallographic and biophysical studies of protein degraders
Kroupova, Alena, Spiteri, Valentina A., Rutter, Zoe J., Furihata, Hirotake, Darren, Darren, Ramachandran, Sarath, Chakraborti, Sohini, Haubrich, Kevin, Pethe, Julie, Gonzales, Denzel, Wijaya, Andre J., Rodriguez-Rios, Maria, Sturbaut, Manon, Lynch, Dylan M., Farnaby, William, Nakasone, Mark A., Zollman, David, Ciulli, Alessio
Published in Nature communications (15.10.2024)
Published in Nature communications (15.10.2024)
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Targeting Transcriptional Enhanced Associate Domains (TEADs): Miniperspective
Gibault, Floriane, Sturbaut, Manon, Bailly, Fabrice, Melnyk, Patricia, Cotelle, Philippe
Published in Journal of medicinal chemistry (28.06.2018)
Published in Journal of medicinal chemistry (28.06.2018)
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Journal Article
Discovery of a cryptic site at the interface 2 of TEAD – Towards a new family of YAP/TAZ-TEAD inhibitors
Sturbaut, Manon, Bailly, Fabrice, Coevoet, Mathilde, Sileo, Pasquale, Pugniere, Martine, Liberelle, Maxime, Magnez, Romain, Thuru, Xavier, Chartier-Harlin, Marie-Christine, Melnyk, Patricia, Gelin, Muriel, Allemand, Frédéric, Guichou, Jean-François, Cotelle, Philippe
Published in European journal of medicinal chemistry (15.12.2021)
Published in European journal of medicinal chemistry (15.12.2021)
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Design, Synthesis and Evaluation of a Series of 1,5‐Diaryl‐1,2,3‐triazole‐4‐carbohydrazones as Inhibitors of the YAP‐TAZ/TEAD Complex
Gibault, Floriane, Sturbaut, Manon, Coevoet, Mathilde, Pugnière, Martine, Burtscher, Ashley, Allemand, Frédéric, Melnyk, Patricia, Hong, Wanjin, Rubin, Brian P., Pobbati, Ajaybabu V., Guichou, Jean‐François, Cotelle, Philippe, Bailly, Fabrice
Published in ChemMedChem (16.09.2021)
Published in ChemMedChem (16.09.2021)
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Toward the Discovery of a Novel Class of YAP⁻TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP⁻TEAD Protein⁻Protein Interface
Gibault, Floriane, Coevoet, Mathilde, Sturbaut, Manon, Farce, Amaury, Renault, Nicolas, Allemand, Frédéric, Guichou, Jean-François, Drucbert, Anne-Sophie, Foulon, Catherine, Magnez, Romain, Thuru, Xavier, Corvaisier, Matthieu, Huet, Guillemette, Chavatte, Philippe, Melnyk, Patricia, Bailly, Fabrice, Cotelle, Philippe
Published in Cancers (08.05.2018)
Published in Cancers (08.05.2018)
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