Unique Anti-Human Immunodeficiency Virus Activities of the Nonnucleoside Reverse Transcriptase Inhibitors Calanolide A, Costatolide, and Dihydrocostatolide
BUCKHEIT, R. W, WHITE, E. L, FLIAKAS-BOLTZ, V, RUSSELL, J, STUP, T. L, KINJERSKI, T. L, OSTERLING, M. C, WEIGAND, A, BADER, J. P
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Published in Antimicrobial Agents and Chemotherapy (01.08.1999)
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Novel Modifications in the Alkenyldiarylmethane (ADAM) Series of Non-Nucleoside Reverse Transcriptase Inhibitors
Casimiro-Garcia, Agustin, Micklatcher, Mark, Turpin, Jim A, Stup, Tracy L, Watson, Karen, Buckheit, Robert W, Cushman, Mark
Published in Journal of medicinal chemistry (18.11.1999)
Published in Journal of medicinal chemistry (18.11.1999)
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Structural Analogues of the Calanolide Anti-HIV Agents. Modification of the trans-10,11-Dimethyldihydropyran-12-ol Ring (Ring C)
Zembower, David E, Liao, Shuyuan, Flavin, Michael T, Xu, Ze-Qi, Stup, Tracy L, Buckheit, Robert W, Khilevich, Albert, Mar, Aye Aye, Sheinkman, Abram K
Published in Journal of medicinal chemistry (14.03.1997)
Published in Journal of medicinal chemistry (14.03.1997)
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Synthesis and Anti-HIV Activity of Cosalane Analogues with Substituted Benzoic Acid Rings Attached to the Pharmacophore through Methylene and Amide Linkers
Ruell, Jeffrey A, De Clercq, Erik, Pannecouque, Christophe, Witvrouw, Myriam, Stup, Tracy L, Turpin, Jim A, Buckheit, Robert W, Cushman, Mark
Published in Journal of organic chemistry (06.08.1999)
Published in Journal of organic chemistry (06.08.1999)
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In vitro anti-human immunodeficiency virus (HIV) activity of the chromanone derivative, 12-oxocalanolide A, a novel NNRTI
Ze-Qi Xu, Buckheit, Robert W., Stup, Tracy L., Flavin, Michael T., Khilevich, Albert, Rizzo, John D., Lin, Lin, Zembower, David E.
Published in Bioorganic & medicinal chemistry letters (18.08.1998)
Published in Bioorganic & medicinal chemistry letters (18.08.1998)
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Comparative anti-HIV evaluation of diverse HIV-1-specific reverse transcriptase inhibitor-resistant virus isolates demonstrates the existence of distinct phenotypic subgroups
Buckheit, Robert W., Fliakas-Boltz, Valerie, Decker, William Don, Roberson, Joseph L., Stup, Tracy L., Pyle, Cathi A., White, E.Lucile, McMahon, James B., Currens, Michael J., Boyd, Michael R., Bader, John P.
Published in Antiviral research (01.03.1995)
Published in Antiviral research (01.03.1995)
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