Structure-Based Discovery of SD-36 as a Potent, Selective, and Efficacious PROTAC Degrader of STAT3 Protein
Zhou, Haibin, Bai, Longchuan, Xu, Renqi, Zhao, Yujun, Chen, Jianyong, McEachern, Donna, Chinnaswamy, Krishnapriya, Wen, Bo, Dai, Lipeng, Kumar, Praveen, Yang, Chao-Yie, Liu, Zhaomin, Wang, Mi, Liu, Liu, Meagher, Jennifer L, Yi, Han, Sun, Duxin, Stuckey, Jeanne A, Wang, Shaomeng
Published in Journal of medicinal chemistry (26.12.2019)
Published in Journal of medicinal chemistry (26.12.2019)
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Mutational signature in colorectal cancer caused by genotoxic pks + E. coli
Pleguezuelos-Manzano, Cayetano, Puschhof, Jens, Rosendahl Huber, Axel, van Hoeck, Arne, Wood, Henry M, Nomburg, Jason, Gurjao, Carino, Manders, Freek, Dalmasso, Guillaume, Stege, Paul B, Paganelli, Fernanda L, Geurts, Maarten H, Beumer, Joep, Mizutani, Tomohiro, Miao, Yi, van der Linden, Reinier, van der Elst, Stefan, Garcia, K Christopher, Top, Janetta, Willems, Rob J L, Giannakis, Marios, Bonnet, Richard, Quirke, Phil, Meyerson, Matthew, Cuppen, Edwin, van Boxtel, Ruben, Clevers, Hans
Published in Nature (London) (01.04.2020)
Published in Nature (London) (01.04.2020)
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Hydrolytic catalysis and structural stabilization in a designed metalloprotein
Zastrow, Melissa L, Peacock, Anna F A, Stuckey, Jeanne A, Pecoraro, Vincent L
Published in Nature chemistry (27.11.2011)
Published in Nature chemistry (27.11.2011)
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Selective inhibition of cullin 3 neddylation through covalent targeting DCN1 protects mice from acetaminophen-induced liver toxicity
Zhou, Haibin, Lu, Jianfeng, Chinnaswamy, Krishnapriya, Stuckey, Jeanne A, Liu, Liu, McEachern, Donna, Yang, Chao-Yie, Bernard, Denzil, Shen, Hong, Rui, Liangyou, Sun, Yi, Wang, Shaomeng
Published in Nature communications (11.05.2021)
Published in Nature communications (11.05.2021)
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D3R grand challenge 2015: Evaluation of protein–ligand pose and affinity predictions
Gathiaka, Symon, Liu, Shuai, Chiu, Michael, Yang, Huanwang, Stuckey, Jeanne A., Kang, You Na, Delproposto, Jim, Kubish, Ginger, Dunbar, James B., Carlson, Heather A., Burley, Stephen K., Walters, W. Patrick, Amaro, Rommie E., Feher, Victoria A., Gilson, Michael K.
Published in Journal of computer-aided molecular design (01.09.2016)
Published in Journal of computer-aided molecular design (01.09.2016)
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A novel small-molecule inhibitor of mcl-1 blocks pancreatic cancer growth in vitro and in vivo
Abulwerdi, Fardokht, Liao, Chenzhong, Liu, Meilan, Azmi, Asfar S, Aboukameel, Amro, Mady, Ahmed S A, Gulappa, Thippeswamy, Cierpicki, Tomasz, Owens, Scott, Zhang, Tao, Sun, Duxin, Stuckey, Jeanne A, Mohammad, Ramzi M, Nikolovska-Coleska, Zaneta
Published in Molecular cancer therapeutics (01.03.2014)
Published in Molecular cancer therapeutics (01.03.2014)
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CSAR Benchmark Exercise 2011–2012: Evaluation of Results from Docking and Relative Ranking of Blinded Congeneric Series
Damm-Ganamet, Kelly L, Smith, Richard D, Dunbar, James B, Stuckey, Jeanne A, Carlson, Heather A
Published in Journal of chemical information and modeling (26.08.2013)
Published in Journal of chemical information and modeling (26.08.2013)
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Discovery of a Highly Potent, Cell-Permeable Macrocyclic Peptidomimetic (MM-589) Targeting the WD Repeat Domain 5 Protein (WDR5)–Mixed Lineage Leukemia (MLL) Protein–Protein Interaction
Karatas, Hacer, Li, Yangbing, Liu, Liu, Ji, Jiao, Lee, Shirley, Chen, Yong, Yang, Jiuling, Huang, Liyue, Bernard, Denzil, Xu, Jing, Townsend, Elizabeth C, Cao, Fang, Ran, Xu, Li, Xiaoqin, Wen, Bo, Sun, Duxin, Stuckey, Jeanne A, Lei, Ming, Dou, Yali, Wang, Shaomeng
Published in Journal of medicinal chemistry (22.06.2017)
Published in Journal of medicinal chemistry (22.06.2017)
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Probing the interaction between the histone methyltransferase/deacetylase subunit RBBP4/7 and the transcription factor BCL11A in epigenetic complexes
Moody, Rebecca Reed, Lo, Miao-Chia, Meagher, Jennifer L., Lin, Chang-Ching, Stevers, Nicholas O., Tinsley, Samantha L., Jung, Inkyung, Matvekas, Aleksas, Stuckey, Jeanne A., Sun, Duxin
Published in The Journal of biological chemistry (09.02.2018)
Published in The Journal of biological chemistry (09.02.2018)
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Mechanistic evaluation and transcriptional signature of a glutathione S-transferase omega 1 inhibitor
Ramkumar, Kavya, Samanta, Soma, Kyani, Anahita, Yang, Suhui, Tamura, Shuzo, Ziemke, Elizabeth, Stuckey, Jeanne A, Li, Si, Chinnaswamy, Krishnapriya, Otake, Hiroyuki, Debnath, Bikash, Yarovenko, Vladimir, Sebolt-Leopold, Judith S, Ljungman, Mats, Neamati, Nouri
Published in Nature communications (05.10.2016)
Published in Nature communications (05.10.2016)
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Discovery of EEDi-5273 as an Exceptionally Potent and Orally Efficacious EED Inhibitor Capable of Achieving Complete and Persistent Tumor Regression
Rej, Rohan Kalyan, Wang, Changwei, Lu, Jianfeng, Wang, Mi, Petrunak, Elyse, Zawacki, Kaitlin P, McEachern, Donna, Yang, Chao-Yie, Wang, Lu, Li, Ruiting, Chinnaswamy, Krishnapriya, Wen, Bo, Sun, Duxin, Stuckey, Jeanne A, Zhou, Yunlong, Chen, Jianyong, Tang, Guozhi, Wang, Shaomeng
Published in Journal of medicinal chemistry (14.10.2021)
Published in Journal of medicinal chemistry (14.10.2021)
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CSAR Benchmark Exercise of 2010: Selection of the Protein–Ligand Complexes
Dunbar, James B, Smith, Richard D, Yang, Chao-Yie, Ung, Peter Man-Un, Lexa, Katrina W, Khazanov, Nickolay A, Stuckey, Jeanne A, Wang, Shaomeng, Carlson, Heather A
Published in Journal of chemical information and modeling (26.09.2011)
Published in Journal of chemical information and modeling (26.09.2011)
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CSAR Data Set Release 2012: Ligands, Affinities, Complexes, and Docking Decoys
Dunbar, James B, Smith, Richard D, Damm-Ganamet, Kelly L, Ahmed, Aqeel, Esposito, Emilio Xavier, Delproposto, James, Chinnaswamy, Krishnapriya, Kang, You-Na, Kubish, Ginger, Gestwicki, Jason E, Stuckey, Jeanne A, Carlson, Heather A
Published in Journal of chemical information and modeling (26.08.2013)
Published in Journal of chemical information and modeling (26.08.2013)
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Comparison of in silico strategies to prioritize rare genomic variants impacting RNA splicing for the diagnosis of genomic disorders
Rowlands, Charlie, Thomas, Huw B, Lord, Jenny, Wai, Htoo A, Arno, Gavin, Beaman, Glenda, Sergouniotis, Panagiotis, Gomes-Silva, Beatriz, Campbell, Christopher, Gossan, Nicole, Hardcastle, Claire, Webb, Kevin, O'Callaghan, Christopher, Hirst, Robert A, Ramsden, Simon, Jones, Elizabeth, Clayton-Smith, Jill, Webster, Andrew R, Douglas, Andrew G L, O'Keefe, Raymond T, Newman, William G, Baralle, Diana, Black, Graeme C M, Ellingford, Jamie M
Published in Scientific reports (18.10.2021)
Published in Scientific reports (18.10.2021)
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Development and optimization of a binding assay for the XIAP BIR3 domain using fluorescence polarization
Nikolovska-Coleska, Zaneta, Wang, Renxiao, Fang, Xueliang, Pan, Hongguang, Tomita, York, Li, Peng, Roller, Peter P., Krajewski, Krzysztof, Saito, Naoyuki G., Stuckey, Jeanne A., Wang, Shaomeng
Published in Analytical biochemistry (15.09.2004)
Published in Analytical biochemistry (15.09.2004)
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Molecular Mechanism for Isoform-Selective Inhibition of Acyl Protein Thioesterases 1 and 2 (APT1 and APT2)
Won, Sang Joon, Davda, Dahvid, Labby, Kristin J, Hwang, Sin Ye, Pricer, Rachel, Majmudar, Jaimeen D, Armacost, Kira A, Rodriguez, Laura A, Rodriguez, Christina L, Chong, Fei San, Torossian, Kristopher A, Palakurthi, Jasmine, Hur, Edward S, Meagher, Jennifer L, Brooks, Charles L, Stuckey, Jeanne A, Martin, Brent R
Published in ACS chemical biology (16.12.2016)
Published in ACS chemical biology (16.12.2016)
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Overall survival in patients with endometrial cancer treated with dostarlimab plus carboplatin–paclitaxel in the randomized ENGOT-EN6/GOG-3031/RUBY trial
Powell, M.A., Bjørge, L., Willmott, L., Novák, Z., Black, D., Gilbert, L., Sharma, S., Valabrega, G., Landrum, L.M., Gropp-Meier, M., Stuckey, A., Boere, I., Gold, M.A., Segev, Y., Gill, S.E., Gennigens, C., Sebastianelli, A., Shahin, M.S., Pothuri, B., Monk, B.J., Buscema, J., Coleman, R.L., Slomovitz, B.M., Ring, K.L., Herzog, T.J., Balas, M.M., Grimshaw, M., Stevens, S., Lai, D.W., McCourt, C., Mirza, M.R.
Published in Annals of oncology (01.08.2024)
Published in Annals of oncology (01.08.2024)
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KRAS Engages AGO2 to Enhance Cellular Transformation
Shankar, Sunita, Pitchiaya, Sethuramasundaram, Malik, Rohit, Kothari, Vishal, Hosono, Yasuyuki, Yocum, Anastasia K., Gundlapalli, Harika, White, Yasmine, Firestone, Ari, Cao, Xuhong, Dhanasekaran, Saravana M., Stuckey, Jeanne A., Bollag, Gideon, Shannon, Kevin, Walter, Nils G., Kumar-Sinha, Chandan, Chinnaiyan, Arul M.
Published in Cell reports (Cambridge) (16.02.2016)
Published in Cell reports (Cambridge) (16.02.2016)
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