Loading…
Design, Synthesis, and Structure–Activity Relationship of 2‑(Piperazin-1-yl)quinazolin-4(3H)‑one Derivatives as Active Agents against Toxoplasma gondii
Deng, Yu, Yu, Yuan-Di, Song, Chao, Xu, Guo-Yang, Xu, Yue, Ye, Chang-Ju
Published in Journal of agricultural and food chemistry (12.03.2025)
Published in Journal of agricultural and food chemistry (12.03.2025)
Get full text
Journal Article
Loading…
Enzyme inhibitory activities an insight into the structure–Activity relationship of biscoumarin derivatives
Faisal, Muhammad, Saeed, Aamer, Shahzad, Danish, Fattah, Tanzeela Abdul, Lal, Bhajan, Channar, Pervaiz Ali, Mahar, Jamaluddin, Saeed, Shomaila, Mahesar, Parvez Ali, Larik, Fayaz Ali
Published in European journal of medicinal chemistry (01.12.2017)
Published in European journal of medicinal chemistry (01.12.2017)
Get full text
Journal Article
Loading…
Structure–Activity Relationship of Terpenes with Anti‐Inflammatory Profile – A Systematic Review
Santana Souza, Marilia Trindade, Almeida, Jackson Roberto Guedes da Silva, Souza Araujo, Adriano Antunes, Duarte, Marcelo Cavalcante, Gelain, Daniel Pens, Moreira, José Cláudio Fonseca, Santos, Marcio Roberto Viana, Quintans‐Júnior, Lucindo José
Published in Basic & clinical pharmacology & toxicology (01.09.2014)
Published in Basic & clinical pharmacology & toxicology (01.09.2014)
Get full text
Journal Article
Loading…
Immunomodulatory Effects of Enzymatic-Synthesized α‑Galactooligosaccharides and Evaluation of the Structure–Activity Relationship
Dai, Zhuqing, Lyu, Wanyong, Xiang, Xiaoli, Tang, Yuhong, Hu, Bing, Ou, Shiyi, Zeng, Xiaoxiong
Published in Journal of agricultural and food chemistry (29.08.2018)
Published in Journal of agricultural and food chemistry (29.08.2018)
Get full text
Journal Article
Loading…
Loading…
Loading…
Tyrosinase inhibitory peptides: Structure-activity relationship study on peptide chemical properties, terminal preferences and intracellular regulation of melanogenesis signaling pathways
Yap, Pei-Gee, Gan, Chee-Yuen
Published in Biochimica et biophysica acta. General subjects (01.01.2024)
Published in Biochimica et biophysica acta. General subjects (01.01.2024)
Get full text
Journal Article
Loading…
Tapinarof and its structure-activity relationship for redox chemistry and phototoxicity on human skin keratinocytes
Zatloukalova, Martina, Hanyk, Jiri, Papouskova, Barbora, Kabelac, Martin, Vostalova, Jitka, Vacek, Jan
Published in Free radical biology & medicine (01.10.2024)
Published in Free radical biology & medicine (01.10.2024)
Get full text
Journal Article
Loading…
Redox Active vs Redox Neutral in Ru/Pd-Catalyzed Sulfonylation: Theoretical Insights into Structure–Activity Relationship between Metal Centers and Regio-Selectivity
Lin, Qingqing, Lv, Huan, Lu, Yu, Yang, Chengkai, Yu, Yan, Liu, Zheyuan
Published in Journal of organic chemistry (20.12.2024)
Published in Journal of organic chemistry (20.12.2024)
Get full text
Journal Article
Loading…
Structure–Activity Relationship of Propargylamine‐Based HDAC Inhibitors
Wünsch, Matthias, Senger, Johanna, Schultheisz, Philipp, Schwarzbich, Sabrina, Schmidtkunz, Karin, Michalek, Carmela, Klaß, Michaela, Goskowitz, Stefanie, Borchert, Philipp, Praetorius, Lucas, Sippl, Wolfgang, Jung, Manfred, Sewald, Norbert
Published in ChemMedChem (19.12.2017)
Published in ChemMedChem (19.12.2017)
Get full text
Journal Article
Loading…
Flavonols and flavones as BACE-1 inhibitors: Structure–activity relationship in cell-free, cell-based and in silico studies reveal novel pharmacophore features
Shimmyo, Yoshiari, Kihara, Takeshi, Akaike, Akinori, Niidome, Tetsuhiro, Sugimoto, Hachiro
Published in Biochimica et biophysica acta (01.05.2008)
Published in Biochimica et biophysica acta (01.05.2008)
Get full text
Journal Article
Loading…
Evaluation of human intestinal absorption data and subsequent derivation of a quantitative structure–activity relationship (QSAR) with the Abraham descriptors
Zhao, Yuan H., Le, Joelle, Abraham, Michael H., Hersey, Anne, Eddershaw, Peter J., Luscombe, Chris N., Boutina, Darko, Beck, Gordon, Sherborne, Brad, Cooper, Ian, Platts, James A.
Published in Journal of pharmaceutical sciences (01.06.2001)
Published in Journal of pharmaceutical sciences (01.06.2001)
Get full text
Journal Article
Loading…
Loading…
Anti-HIV-1 activity and structure–activity-relationship study of a fucosylated glycosaminoglycan from an echinoderm by targeting the conserved CD4 induced epitope
Lian, Wu, Wu, Mingyi, Huang, Ning, Gao, Na, Xiao, Chuang, Li, Zi, Zhang, Zhigang, Zheng, Yongtang, Peng, Wenlie, Zhao, Jinhua
Published in Biochimica et biophysica acta (01.10.2013)
Published in Biochimica et biophysica acta (01.10.2013)
Get full text
Journal Article
Loading…
Building Highly Reliable Quantitative Structure–Activity Relationship Classification Models Using the Rivality Index Neighborhood Algorithm with Feature Selection
Ruiz, Irene Luque, Gómez-Nieto, Miguel Ángel
Published in Journal of chemical information and modeling (27.01.2020)
Published in Journal of chemical information and modeling (27.01.2020)
Get full text
Journal Article
Loading…
Exploring the structure-activity relationship of benzylidene-2,3-dihydro-1H-inden-1-one compared to benzofuran-3(2H)-one derivatives as inhibitors of tau amyloid fibers
Boukherrouba, Emeline, Larosa, Camille, Nguyen, Kim-Anh, Caburet, Jérémy, Lunven, Laurent, Bonnet, Hugues, Fortuné, Antoine, Boumendjel, Ahcène, Boucherle, Benjamin, Chierici, Sabine, Peuchmaur, Marine
Published in European journal of medicinal chemistry (05.03.2022)
Published in European journal of medicinal chemistry (05.03.2022)
Get full text
Journal Article
Loading…
Deferiprone: Pan-selective Histone Lysine Demethylase Inhibition Activity and Structure Activity Relationship Study
Khodaverdian, Verjine, Tapadar, Subhasish, MacDonald, Ian A., Xu, Yuan, Ho, Po-Yi, Bridges, Allison, Rajpurohit, Pragya, Sanghani, Bhakti A., Fan, Yuhong, Thangaraju, Muthusamy, Hathaway, Nathaniel A., Oyelere, Adegboyega K.
Published in Scientific reports (18.03.2019)
Published in Scientific reports (18.03.2019)
Get full text
Journal Article
Loading…
Binary Classification of a Large Collection of Environmental Chemicals from Estrogen Receptor Assays by Quantitative Structure–Activity Relationship and Machine Learning Methods
Zang, Qingda, Rotroff, Daniel M, Judson, Richard S
Published in Journal of chemical information and modeling (23.12.2013)
Published in Journal of chemical information and modeling (23.12.2013)
Get full text
Journal Article
Loading…
Unraveling the synthetic strategy, structure activity relationship of azetidinones: Insights into their multidrug and toxin extrusion protein (MATE transporter) inhibition facilitating drug development against MDR
Mal, Suvadeep, Mahapatra, Monalisa, Pakeeraiah, Kakarla, Panda, Preetesh Kumar, Sahoo, Jyotirmaya, Roy, Partha, Paidesetty, Sudhir Kumar
Published in Bioorganic chemistry (01.03.2025)
Published in Bioorganic chemistry (01.03.2025)
Get full text
Journal Article
Loading…
Identification of a New Class of Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors Followed by a Structure–Activity Relationship Study
Hansen, Stinne W, Erichsen, Mette N, Fu, Bingru, Bjørn-Yoshimoto, Walden E, Abrahamsen, Bjarke, Hansen, Jacob C, Jensen, Anders A, Bunch, Lennart
Published in Journal of medicinal chemistry (13.10.2016)
Published in Journal of medicinal chemistry (13.10.2016)
Get full text
Journal Article