Microbial efflux pump inhibition: tactics and strategies
Tegos, George P, Haynes, Mark, Strouse, J Jacob, Khan, Mohiuddin Md T, Bologa, Cristian G, Oprea, Tudor I, Sklar, Larry A
Published in Current pharmaceutical design (01.05.2011)
Published in Current pharmaceutical design (01.05.2011)
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Fluorescent substrates for flow cytometric evaluation of efflux inhibition in ABCB1, ABCC1, and ABCG2 transporters
Strouse, J. Jacob, Ivnitski-Steele, Irena, Waller, Anna, Young, Susan M., Perez, Dominique, Evangelisti, Annette M., Ursu, Oleg, Bologa, Cristian G., Carter, Mark B., Salas, Virginia M., Tegos, George, Larson, Richard S., Oprea, Tudor I., Edwards, Bruce S., Sklar, Larry A.
Published in Analytical biochemistry (01.06.2013)
Published in Analytical biochemistry (01.06.2013)
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A novel flow cytometric HTS assay reveals functional modulators of ATP binding cassette transporter ABCB6
Polireddy, Kishore, Khan, Mohiuddin Md Taimur, Chavan, Hemantkumar, Young, Susan, Ma, Xiaochao, Waller, Anna, Garcia, Matthew, Perez, Dominique, Chavez, Stephanie, Strouse, Jacob J, Haynes, Mark K, Bologa, Cristian G, Oprea, Tudor I, Tegos, George P, Sklar, Larry A, Krishnamurthy, Partha
Published in PloS one (10.07.2012)
Published in PloS one (10.07.2012)
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Discovery of Small-Molecule Nonfluorescent Inhibitors of Fluorogen-Fluorogen Activating Protein Binding Pair
Wu, Yang, Stauffer, Shaun R, Stanfield, Robyn L, Tapia, Phillip H, Ursu, Oleg, Fisher, Gregory W, Szent-Gyorgyi, Christopher, Evangelisti, Annette, Waller, Anna, Strouse, J Jacob, Carter, Mark B, Bologa, Cristian, Gouveia, Kristine, Poslusney, Mike, Waggoner, Alan S, Lindsley, Craig W, Jarvik, Jonathan W, Sklar, Larry A
Published in Journal of biomolecular screening (01.01.2016)
Published in Journal of biomolecular screening (01.01.2016)
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A selective ATP-binding cassette subfamily G member 2 efflux inhibitor revealed via high-throughput flow cytometry
Strouse, J Jacob, Ivnitski-Steele, Irena, Khawaja, Hadya M, Perez, Dominique, Ricci, Jerec, Yao, Tuanli, Weiner, Warren S, Schroeder, Chad E, Simpson, Denise S, Maki, Brooks E, Li, Kelin, Golden, Jennifer E, Foutz, Terry D, Waller, Anna, Evangelisti, Annette M, Young, Susan M, Chavez, Stephanie E, Garcia, Matthew J, Ursu, Oleg, Bologa, Cristian G, Carter, Mark B, Salas, Virginia M, Gouveia, Kristine, Tegos, George P, Oprea, Tudor I, Edwards, Bruce S, Aubé, Jeffrey, Larson, Richard S, Sklar, Larry A
Published in Journal of biomolecular screening (01.01.2013)
Published in Journal of biomolecular screening (01.01.2013)
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Targeting efflux pumps to overcome antifungal drug resistance
Holmes, Ann R, Cardno, Tony S, Strouse, J Jacob, Ivnitski-Steele, Irena, Keniya, Mikhail V, Lackovic, Kurt, Monk, Brian C, Sklar, Larry A, Cannon, Richard D
Published in Future medicinal chemistry (01.08.2016)
Published in Future medicinal chemistry (01.08.2016)
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Characterization of a Cdc42 Protein Inhibitor and Its Use as a Molecular Probe
Hong, Lin, Kenney, S.Ray, Phillips, Genevieve K., Simpson, Denise, Schroeder, Chad E., Nöth, Julica, Romero, Elsa, Swanson, Scarlett, Waller, Anna, Strouse, J.Jacob, Carter, Mark, Chigaev, Alexandre, Ursu, Oleg, Oprea, Tudor, Hjelle, Brian, Golden, Jennifer E., Aubé, Jeffrey, Hudson, Laurie G., Buranda, Tione, Sklar, Larry A., Wandinger-Ness, Angela
Published in The Journal of biological chemistry (22.03.2013)
Published in The Journal of biological chemistry (22.03.2013)
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A Competitive Nucleotide Binding Inhibitor: In Vitro Characterization of Rab7 GTPase Inhibition
Agola, Jacob O, Hong, Lin, Surviladze, Zurab, Ursu, Oleg, Waller, Anna, Strouse, J. Jacob, Simpson, Denise S, Schroeder, Chad E, Oprea, Tudor I, Golden, Jennifer E, Aubé, Jeffrey, Buranda, Tione, Sklar, Larry A, Wandinger-Ness, Angela
Published in ACS chemical biology (15.06.2012)
Published in ACS chemical biology (15.06.2012)
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Discovery of regulators of receptor internalization with high-throughput flow cytometry
Wu, Yang, Tapia, Phillip H, Fisher, Gregory W, Simons, Peter C, Strouse, J Jacob, Foutz, Terry, Waggoner, Alan S, Jarvik, Jonathan, Sklar, Larry A
Published in Molecular pharmacology (01.10.2012)
Published in Molecular pharmacology (01.10.2012)
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Identification of a Small Molecule Yeast TORC1 Inhibitor with a Multiplex Screen Based on Flow Cytometry
Chen, Jun, Young, Susan M, Allen, Chris, Seeber, Andrew, Péli-Gulli, Marie-Pierre, Panchaud, Nicolas, Waller, Anna, Ursu, Oleg, Yao, Tuanli, Golden, Jennifer E, Strouse, J. Jacob, Carter, Mark B, Kang, Huining, Bologa, Cristian G, Foutz, Terry D, Edwards, Bruce S, Peterson, Blake R, Aubé, Jeffrey, Werner-Washburne, Margaret, Loewith, Robbie J, De Virgilio, Claudio, Sklar, Larry A
Published in ACS chemical biology (20.04.2012)
Published in ACS chemical biology (20.04.2012)
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Detection of Intracellular Granularity Induction in Prostate Cancer Cell Lines by Small Molecules Using the HyperCyt® High-Throughput Flow Cytometry System
Haynes, Mark K., Strouse, J. Jacob, Waller, Anna, Leitao, Andrei, Curpan, Ramona F., Bologa, Cristian, Oprea, Tudor I., Prossnitz, Eric R., Edwards, Bruce S., Sklar, Larry A., Thompson, Todd A.
Published in Journal of biomolecular screening (01.07.2009)
Published in Journal of biomolecular screening (01.07.2009)
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Synthesis and anti-Hantaan virus activity of N(1)-3-fluorophenyl-inosine
Chung, Dong-Hoon, Strouse, J Jacob, Sun, Yanjie, Arterburn, Jeffrey B, Parker, William B, Jonsson, Colleen B
Published in Antiviral research (01.07.2009)
Published in Antiviral research (01.07.2009)
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Journal Article
Characterization of a Cdc42 protein inhibitor and its use as a molecular probe
Hong, Lin, Kenney, S. Ray, Phillips, Genevieve K., Simpson, Denise, Schroeder, Chad E., Nöth, Julica, Romero, Elsa, Swanson, Scarlett, Waller, Anna, Strouse, J. Jacob, Carter, Mark, Chigaev, Alexandre, Ursu, Oleg, Oprea, Tudor, Hjelle, Brian, Golden, Jennifer E., Aubé, Jeffrey, Hudson, Laurie G., Buranda, Tione, Sklar, Larry A., Wandinger-Ness, Angela
Published in The Journal of biological chemistry (07.03.2014)
Published in The Journal of biological chemistry (07.03.2014)
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Synthesis and anti-Hantaan virus activity of N 1-3-fluorophenyl-inosine
Chung, Dong-Hoon, Strouse, J. Jacob, Sun, Yanjie, Arterburn, Jeffrey B., Parker, William B., Jonsson, Colleen B.
Published in Antiviral research (01.07.2009)
Published in Antiviral research (01.07.2009)
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Journal Article
Identification of a small molecule yeast TORC1 inhibitor with a flow cytometry-based multiplex screen
Chen, Jun, Young, Susan M., Allen, Chris, Seeber, Andrew, Péli-Gulli, Marie-Pierre, Panchaud, Nicolas, Waller, Anna, Ursu, Oleg, Yao, Tuanli, Golden, Jennifer E., Strouse, J. Jacob, Carter, Mark B., Kang, Huining, Bologa, Cristian G., Foutz, Terry D., Edwards, Bruce S., Peterson, Blake R., Aubé, Jeffrey, Werner-Washburne, Margaret, Loewith, Robbie J., De Virgilio, Claudio, Sklar, Larry A.
Published in ACS chemical biology (01.02.2012)
Published in ACS chemical biology (01.02.2012)
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Synthesis and anti-Hantaan virus activity of N1-3-fluorophenyl-inosine
CHUNG, Dong-Hoon, STROUSE, J. Jacob, YANJIE SUN, ARTERBURN, Jeffrey B, PARKER, William B, JONSSON, Colleen B
Published in Antiviral research (01.07.2009)
Published in Antiviral research (01.07.2009)
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Journal Article
A Novel Fluorescent Cross-Reactive Formylpeptide Receptor/Formylpeptide Receptor-Like 1 Hexapeptide Ligand1
Strouse, J. Jacob, Young, Susan M., Mitchell, Hugh D., Ye, Richard D., Prossnitz, Eric R., Sklar, Larry A., Edwards, Bruce S.
Published in Cytometry. Part A (01.03.2009)
Published in Cytometry. Part A (01.03.2009)
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