Substrate-Dependent Modulation of CYP3A4 Catalytic Activity: Analysis of 27 Test Compounds with Four Fluorometric Substrates
STRESSER, David M, BLANCHARD, Andrew P, TURNER, Stephanie D, ERVE, John C. L, DANDENEAU, Andre A, MILLER, Vaughn P, CRESPI, Charles L
Published in Drug metabolism and disposition (01.12.2000)
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Published in Drug metabolism and disposition (01.12.2000)
Journal Article
Concurrent Flavin-Containing Monooxygenase Down-Regulation and Cytochrome P-450 Induction by Dietary Indoles in Rat: Implications for Drug-Drug Interaction
KATCHAMART, S, STRESSER, D. M, DEHAL, S. S, KUPFER, D, WILLIAMS, D. E
Published in Drug metabolism and disposition (01.08.2000)
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Published in Drug metabolism and disposition (01.08.2000)
Journal Article
Validation of cytochrome P450 time-dependent inhibition assays: a two-time point IC50 shift approach facilitates kinact assay design
Perloff, E. S., Mason, A. K., Dehal, S. S., Blanchard, A. P., Morgan, L., Ho, T., Dandeneau, A., Crocker, R. M., Chandler, C. M., Boily, N., Crespi, C. L., Stresser, D. M.
Published in Xenobiotica (01.02.2009)
Published in Xenobiotica (01.02.2009)
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The Use of 3-[2-(N,N-Diethyl-N-methylammonium)ethyl]-7-methoxy-4-methylcoumarin (AMMC) as a Specific CYP2D6 Probe in Human Liver Microsomes
CHAURET, Nathalie, DOBBS, Barry, LACKMAN, Rebecca L, BATEMAN, Kevin, NICOLL-GRIFFITH, Deborah A, STRESSER, David M, ACKERMANN, Joseph M, TURNER, Stephanie D, MILLER, Vaughn P, CRESPI, Charles L
Published in Drug metabolism and disposition (01.09.2001)
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Published in Drug metabolism and disposition (01.09.2001)
Journal Article
Indole-3-carbinol induces a rat liver glutathione transferase subunit (Yc2) with high activity toward aflatoxin B1 exo-epoxide. Association with reduced levels of hepatic aflatoxin-DNA adducts in vivo
Stresser, D M, Williams, D E, McLellan, L I, Harris, T M, Bailey, G S
Published in Drug metabolism and disposition (01.05.1994)
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Published in Drug metabolism and disposition (01.05.1994)
Journal Article
In vitro and pharmacophore insights into CYP3A enzymes
Ekins, Sean, Stresser, David M., Andrew Williams, J.
Published in Trends in pharmacological sciences (Regular ed.) (01.04.2003)
Published in Trends in pharmacological sciences (Regular ed.) (01.04.2003)
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Journal Article
Biotransformation and estrogenic activity of Methoxychlor and its metabolites in channel catfish ( Ictalurus punctatus)
Schlenk, D., Stresser, D.M., Rimoldi, J., Arcand, L., McCants, J., Nimrod, A.C., Bensorr, W.H.
Published in Marine environmental research (01.07.1998)
Published in Marine environmental research (01.07.1998)
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Journal Article
Conference Proceeding
Influence of β-Naphthoflavone and Methoxychlor Pretreatment on the Biotransformation and Estrogenic Activity of Methoxychlor in Channel Catfish (Ictalurus punctatus)
Schlenk, Daniel, Stresser, David M., McCants, John C., Nimrod, Alison C., Benson, William H.
Published in Toxicology and applied pharmacology (01.08.1997)
Published in Toxicology and applied pharmacology (01.08.1997)
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Fluorometric screening for metabolism-based drug–drug interactions
Crespi, Charles L., Stresser, David M.
Published in Journal of pharmacological and toxicological methods (01.07.2000)
Published in Journal of pharmacological and toxicological methods (01.07.2000)
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Journal Article
Cytochrome P450 Fluorometric Substrates: Identification of Isoform-Selective Probes for Rat CYP2D2 and Human CYP3A4
STRESSER, David M, TURNER, Stephanie D, BLANCHARD, Andrew P, MILLER, Vaughn P, CRESPI, Charles L
Published in Drug metabolism and disposition (01.07.2002)
Published in Drug metabolism and disposition (01.07.2002)
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Journal Article
Selective Time- and NADPH-Dependent Inhibition of Human CYP2E1 by Clomethiazole
Stresser, David M, Perloff, Elke S, Mason, Andrew K, Blanchard, Andrew P, Dehal, Shangara S, Creegan, Timothy P, Singh, Ritu, Gangl, Eric T
Published in Drug metabolism and disposition (01.08.2016)
Published in Drug metabolism and disposition (01.08.2016)
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