Identification of phosphorylase kinase as a novel therapeutic target through high-throughput screening for anti-angiogenesis compounds in zebrafish
Camus, S, Quevedo, C, Menéndez, S, Paramonov, I, Stouten, P F W, Janssen, R A J, Rueb, S, He, S, Snaar-Jagalska, B E, Laricchia-Robbio, L, Izpisua Belmonte, J C
Published in Oncogene (27.09.2012)
Published in Oncogene (27.09.2012)
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A fast immunoassay for the screening of β-agonists in hair
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Conference Proceeding
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Design, Synthesis, and Biological Evaluation of Potent and Selective Amidino Bicyclic Factor Xa Inhibitors
Han, Qi, Dominguez, Celia, Stouten, Pieter F. W, Park, Jeongsook M, Duffy, Daniel E, Galemmo, Robert A, Rossi, Karen A, Alexander, Richard S, Smallwood, Angela M, Wong, Pancras C, Wright, Matthew M, Luettgen, Joseph M, Knabb, Robert M, Wexler, Ruth R
Published in Journal of medicinal chemistry (16.11.2000)
Published in Journal of medicinal chemistry (16.11.2000)
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How does the switch II region of G-domains work?
Stouten, Pieter F.W., Sander, Chris, Wittinghofer, Alfred, Valencia, Alfonso
Published in FEBS Letters (29.03.1993)
Published in FEBS Letters (29.03.1993)
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A comparison of structural and dynamic properties of different simulation methods applied to SH3
van Aalten, D.M., Amadei, A., Bywater, R., Findlay, J.B., Berendsen, H.J., Sander, C., Stouten, P.F.
Published in Biophysical journal (01.02.1996)
Published in Biophysical journal (01.02.1996)
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New triple-helical model for the shaft of the adenovirus fibre
Stouten, Pieter F.W., Sander, Chris, Ruigrok, Rob W.H., Cusack, Stephen
Published in Journal of molecular biology (20.08.1992)
Published in Journal of molecular biology (20.08.1992)
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Does a diol cyclic urea inhibitor of HIV-1 protease bind tighter than its corresponding alcohol form? A study by free energy perturbation and continuum electrostatics calculations
Wang, L, Duan, Y, Stouten, P, De Lucca, G V, Klabe, R M, Kollman, P A
Published in Journal of computer-aided molecular design (01.02.2001)
Published in Journal of computer-aided molecular design (01.02.2001)
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Bisbenzamidine isoxazoline derivatives as factor Xa inhibitors
Quan, M.L., Pruitt, J.R., Ellis, C.D., Liauw, A.Y., Galemmo, R.A., Stouten, P.F.W., Wityak, J., Knabb, R.M., Thoolen, M.J., Wong, P.C., Wexler, R.R.
Published in Bioorganic & medicinal chemistry letters (04.11.1997)
Published in Bioorganic & medicinal chemistry letters (04.11.1997)
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The de novo design and synthesis of cyclic urea inhibitors of factor Xa: Initial sar studies
Galemmo, Robert A., Maduskuie, Thomas P., Dominguez, Celia, Rossi, Karen A., Knabb, Robert M., Wexler, Ruth R., Stouten, Pieter F.W.
Published in Bioorganic & medicinal chemistry letters (06.10.1998)
Published in Bioorganic & medicinal chemistry letters (06.10.1998)
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Preparation of pyrrolidine and isoxazolidine benzamidines as potent inhibitors of coagulation factor Xa
Fevig, John M., Buriak, Joseph, Stouten, Pieter F.W., Knabb, Robert M., Lam, Gilbert N., Wong, Pancras C., Wexler, Ruth R.
Published in Bioorganic & medicinal chemistry letters (19.04.1999)
Published in Bioorganic & medicinal chemistry letters (19.04.1999)
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Journal Article
The de novo design and synthesis of cyclic urea inhibitors of factor Xa : Optimization of the S4 ligand
GALEMMO, R. A, WELLS, B. L, KNABB, R. M, WEXLER, R. R, ROSSI, K. A, ALEXANDER, R. S, DOMINGUEZ, C, MADUSKUIE, T. P, STOUTEN, P. F. W, WRIGHT, M. R, AUNGST, B. J, WONG, P. C
Published in Bioorganic & medicinal chemistry letters (07.02.2000)
Published in Bioorganic & medicinal chemistry letters (07.02.2000)
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Interchain cysteine bridges control entry of progesterone to the central cavity of the uteroglobin dimer
Peter, W, Dunkel, R, Stouten, P F, Vriend, G, Beato, M, Suske, G
Published in Protein engineering (01.06.1992)
Published in Protein engineering (01.06.1992)
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Journal Article
Synthesis and Biological Evaluation of 1-Aryl-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-4-one Inhibitors of Cyclin-Dependent Kinases
Markwalder, Jay A, Arnone, Marc R, Benfield, Pamela A, Boisclair, Michael, Burton, Catherine R, Chang, Chong-Hwan, Cox, Sarah S, Czerniak, Philip M, Dean, Charity L, Doleniak, Deborah, Grafstrom, Robert, Harrison, Barbara A, Kaltenbach, Robert F, Nugiel, David A, Rossi, Karen A, Sherk, Susan R, Sisk, Lisa M, Stouten, Pieter, Trainor, George L, Worland, Peter, Seitz, Steven P
Published in Journal of medicinal chemistry (18.11.2004)
Published in Journal of medicinal chemistry (18.11.2004)
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Structure-function relationship for the highly toxic crotoxin from Crotalus durissus terrificus
MASCARENHAS, Y. P, STOUTEN, P. F. W, BELTRAN, J. R, LAURE, C. J, VRIEND, G
Published in European biophysics journal (01.07.1992)
Published in European biophysics journal (01.07.1992)
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Development of a one step strip test for the detection of sulfadimidine residues
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Conference Proceeding
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