POST, partner of stromal interaction molecule 1 (STIM1), targets STIM1 to multiple transporters
Krapivinsky, Grigory, Krapivinsky, Luba, Stotz, Stephanie C, Manasian, Yunona, Clapham, David E
Published in Proceedings of the National Academy of Sciences - PNAS (29.11.2011)
Published in Proceedings of the National Academy of Sciences - PNAS (29.11.2011)
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Citral sensing by Transient [corrected] receptor potential channels in dorsal root ganglion neurons
Stotz, Stephanie C, Vriens, Joris, Martyn, Derek, Clardy, Jon, Clapham, David E
Published in PloS one (07.05.2008)
Published in PloS one (07.05.2008)
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Breaking boundaries: Pan BETi disrupt 3D chromatin structure, BD2-selective BETi are strictly epigenetic transcriptional regulators
Tsujikawa, Laura M., Kharenko, Olesya A., Stotz, Stephanie C., Rakai, Brooke D., Sarsons, Christopher D., Gilham, Dean, Wasiak, Sylwia, Fu, Li, Sweeney, Michael, Johansson, Jan O., Wong, Norman C.W., Kulikowski, Ewelina
Published in Biomedicine & pharmacotherapy (01.08.2022)
Published in Biomedicine & pharmacotherapy (01.08.2022)
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CACNA1H Mutations in Autism Spectrum Disorders
Splawski, Igor, Yoo, Dana S., Stotz, Stephanie C., Cherry, Allison, Clapham, David E., Keating, Mark T.
Published in The Journal of biological chemistry (04.08.2006)
Published in The Journal of biological chemistry (04.08.2006)
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Inhibition of epigenetic reader proteins by apabetalone counters inflammation in activated innate immune cells from Fabry disease patients receiving enzyme replacement therapy
Fu, Li, Wasiak, Sylwia, Tsujikawa, Laura M., Rakai, Brooke D., Stotz, Stephanie C., Wong, Norman C. W., Johansson, Jan O., Sweeney, Michael, Mohan, Connie M., Khan, Aneal, Kulikowski, Ewelina
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Published in Pharmacology research & perspectives (01.06.2022)
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Bromodomain and Extraterminal Protein Inhibitor, Apabetalone (RVX-208), Reduces ACE2 Expression and Attenuates SARS-Cov-2 Infection In Vitro
Gilham, Dean, Smith, Audrey L, Fu, Li, Moore, Dalia Y, Muralidharan, Abenaya, Reid, St Patrick M, Stotz, Stephanie C, Johansson, Jan O, Sweeney, Michael, Wong, Norman C W, Kulikowski, Ewelina, El-Gamal, Dalia
Published in Biomedicines (18.04.2021)
Published in Biomedicines (18.04.2021)
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Axo-glial communication through neurexin-neuroligin signaling regulates myelination and oligodendrocyte differentiation
Proctor, Dustin T., Stotz, Stephanie C., Scott, Lucas O. M., de la Hoz, Cristiane L. R., Poon, Kelvin W. C., Stys, Peter K., Colicos, Michael A.
Published in Glia (01.11.2015)
Published in Glia (01.11.2015)
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Apabetalone, a Clinical-Stage, Selective BET Inhibitor, Opposes DUX4 Target Gene Expression in Primary Human FSHD Muscle Cells
Sarsons, Christopher D, Gilham, Dean, Tsujikawa, Laura M, Wasiak, Sylwia, Fu, Li, Rakai, Brooke D, Stotz, Stephanie C, Carestia, Agostina, Sweeney, Michael, Kulikowski, Ewelina
Published in Biomedicines (30.09.2023)
Published in Biomedicines (30.09.2023)
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The BET inhibitor apabetalone decreases neuroendothelial proinflammatory activation in vitro and in a mouse model of systemic inflammation
Wasiak, Sylwia, Fu, Li, Daze, Emily, Gilham, Dean, Rakai, Brooke D., Stotz, Stephanie C., Tsujikawa, Laura M., Sarsons, Chris D., Studer, Deborah, Rinker, Kristina D., Jahagirdar, Ravi, Wong, Norman C. W., Sweeney, Michael, Johansson, Jan O., Kulikowski, Ewelina
Published in Translational neuroscience (01.01.2023)
Published in Translational neuroscience (01.01.2023)
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Epigenetic Modulation by Apabetalone Counters Cytokine-Driven Acute Phase Response In Vitro, in Mice and in Patients with Cardiovascular Disease
Sweeney, Michael, Johansson, Jan O., Wong, Norman C. W., Kulikowski, Ewelina, Fu, Li, Rakai, Brooke D., Stotz, Stephanie C., Halliday, Christopher, Tsujikawa, Laura M., Daze, Emily, Gilham, Dean, Wasiak, Sylwia, Jahagirdar, Ravi
Published in Cardiovascular therapeutics (2020)
Published in Cardiovascular therapeutics (2020)
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Benefit of Apabetalone on Plasma Proteins in Renal Disease
Wasiak, Sylwia, Tsujikawa, Laura M., Halliday, Christopher, Stotz, Stephanie C., Gilham, Dean, Jahagirdar, Ravi, Kalantar-Zadeh, Kamyar, Robson, Richard, Sweeney, Michael, Johansson, Jan O., Wong, Norman C., Kulikowski, Ewelina
Published in Kidney international reports (01.05.2018)
Published in Kidney international reports (01.05.2018)
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Inorganic polyphosphate regulates neuronal excitability through modulation of voltage-gated channels
Stotz, Stephanie C, Scott, Lucas Om, Drummond-Main, Christopher, Avchalumov, Yosef, Girotto, Fernando, Davidsen, Jörn, Gómez-Gárcia, Maria R, Rho, Jong M, Pavlov, Evgeny V, Colicos, Michael A
Published in Molecular brain (31.05.2014)
Published in Molecular brain (31.05.2014)
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Integrin Receptor Activation Triggers Converging Regulation of Cav1.2 Calcium Channels by c-Src and Protein Kinase A Pathways
Gui, Peichun, Wu, Xin, Ling, Shizhang, Stotz, Stephanie C., Winkfein, Robert J., Wilson, Emily, Davis, George E., Braun, Andrew P., Zamponi, Gerald W., Davis, Michael J.
Published in The Journal of biological chemistry (19.05.2006)
Published in The Journal of biological chemistry (19.05.2006)
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Apabetalone downregulates factors and pathways associated with vascular calcification
Gilham, Dean, Tsujikawa, Laura M., Sarsons, Christopher D., Halliday, Christopher, Wasiak, Sylwia, Stotz, Stephanie C., Jahagirdar, Ravi, Sweeney, Michael, Johansson, Jan O., Wong, Norman C.W., Kalantar-Zadeh, Kamyar, Kulikowski, Ewelina
Published in Atherosclerosis (01.01.2019)
Published in Atherosclerosis (01.01.2019)
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AKAP79 modulation of L-type channels involves disruption of intramolecular interactions in the CaV1.2 subunit
Altier, Christophe, Dubel, Stefan J., Barrere, Christian, Jarvis, Scott E., Stotz, Stephanie C., Scott, John D., Nargeot, Joel, Zamponi, Gerald W., Bourinet, Emmanuel
Published in Channels (Austin, Tex.) (01.05.2012)
Published in Channels (Austin, Tex.) (01.05.2012)
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Epigenetic BET reader inhibitor apabetalone (RVX-208) counters proinflammatory aortic gene expression in a diet induced obesity mouse model and in human endothelial cells
Wasiak, Sylwia, Tsujikawa, Laura M., Daze, Emily, Gilham, Dean, Stotz, Stephanie C., Rakai, Brooke D., Sarsons, Chris D., Fu, Li, Azhar, Salman, Jahagirdar, Ravi, Sweeney, Michael, Johansson, Jan O., Wong, Norman C.W., Kulikowski, Ewelina
Published in Atherosclerosis (01.01.2023)
Published in Atherosclerosis (01.01.2023)
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Apabetalone (RVX-208) reduces vascular inflammation in vitro and in CVD patients by a BET-dependent epigenetic mechanism
Tsujikawa, Laura M, Fu, Li, Das, Shovon, Halliday, Christopher, Rakai, Brooke D, Stotz, Stephanie C, Sarsons, Christopher D, Gilham, Dean, Daze, Emily, Wasiak, Sylwia, Studer, Deborah, Rinker, Kristina D, Sweeney, Michael, Johansson, Jan O, Wong, Norman C W, Kulikowski, Ewelina
Published in Clinical epigenetics (12.07.2019)
Published in Clinical epigenetics (12.07.2019)
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Dual mechanism: Epigenetic inhibitor apabetalone reduces SARS-CoV-2 Delta and Omicron variant spike binding and attenuates SARS-CoV-2 RNA induced inflammation
Fu, Li, Gilham, Dean, Stotz, Stephanie C., Sarsons, Christopher D., Rakai, Brooke D., Tsujikawa, Laura M., Wasiak, Sylwia, Johansson, Jan O., Sweeney, Michael, Wong, Norman C.W., Kulikowski, Ewelina
Published in International immunopharmacology (01.04.2023)
Published in International immunopharmacology (01.04.2023)
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