Selective USP7 inhibition elicits cancer cell killing through a p53-dependent mechanism
Schauer, Nathan J, Liu, Xiaoxi, Magin, Robert S, Doherty, Laura M, Chan, Wai Cheung, Ficarro, Scott B, Hu, Wanyi, Roberts, Rebekka M, Iacob, Roxana E, Stolte, Björn, Giacomelli, Andrew O, Perera, Sumner, McKay, Kyle, Boswell, Sarah A, Weisberg, Ellen L, Ray, Arghya, Chauhan, Dharminder, Dhe-Paganon, Sirano, Anderson, Ken C, Griffin, James D, Li, Jianing, Hahn, William C, Sorger, Peter K, Engen, John R, Stegmaier, Kimberly, Marto, Jarrod A, Buhrlage, Sara J
Published in Scientific reports (24.03.2020)
Published in Scientific reports (24.03.2020)
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Journal Article
TRIM8 modulates the EWS/FLI oncoprotein to promote survival in Ewing sarcoma
Seong, Bo Kyung A., Dharia, Neekesh V., Lin, Shan, Donovan, Katherine A., Chong, Shasha, Robichaud, Amanda, Conway, Amy, Hamze, Amanda, Ross, Linda, Alexe, Gabriela, Adane, Biniam, Nabet, Behnam, Ferguson, Fleur M., Stolte, Björn, Wang, Emily Jue, Sun, Jialin, Darzacq, Xavier, Piccioni, Federica, Gray, Nathanael S., Fischer, Eric S., Stegmaier, Kimberly
Published in Cancer cell (13.09.2021)
Published in Cancer cell (13.09.2021)
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Journal Article
Genome-scale CRISPR-Cas9 screen identifies druggable dependencies in TP53 wild-type Ewing sarcoma
Stolte, Björn, Iniguez, Amanda Balboni, Dharia, Neekesh V, Robichaud, Amanda L, Conway, Amy Saur, Morgan, Ann M, Alexe, Gabriela, Schauer, Nathan J, Liu, Xiaoxi, Bird, Gregory H, Tsherniak, Aviad, Vazquez, Francisca, Buhrlage, Sara J, Walensky, Loren D, Stegmaier, Kimberly
Published in The Journal of experimental medicine (06.08.2018)
Published in The Journal of experimental medicine (06.08.2018)
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Journal Article
EWS/FLI Confers Tumor Cell Synthetic Lethality to CDK12 Inhibition in Ewing Sarcoma
Iniguez, Amanda Balboni, Stolte, Björn, Wang, Emily Jue, Conway, Amy Saur, Alexe, Gabriela, Dharia, Neekesh V., Kwiatkowski, Nicholas, Zhang, Tinghu, Abraham, Brian J., Mora, Jaume, Kalev, Peter, Leggett, Alan, Chowdhury, Dipanjan, Benes, Cyril H., Young, Richard A., Gray, Nathanael S., Stegmaier, Kimberly
Published in Cancer cell (12.02.2018)
Published in Cancer cell (12.02.2018)
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Resistance to Epigenetic-Targeted Therapy Engenders Tumor Cell Vulnerabilities Associated with Enhancer Remodeling
Iniguez, Amanda Balboni, Alexe, Gabriela, Wang, Emily Jue, Roti, Giovanni, Patel, Sarvagna, Chen, Liying, Kitara, Samuel, Conway, Amy, Robichaud, Amanda L., Stolte, Björn, Bandopadhayay, Pratiti, Goodale, Amy, Pantel, Sasha, Lee, Yenarae, Cheff, Dorian M., Hall, Matthew D., Guha, Rajarshi, Davis, Mindy I., Menard, Marie, Nasholm, Nicole, Weiss, William A., Qi, Jun, Beroukhim, Rameen, Piccioni, Federica, Johannessen, Cory, Stegmaier, Kimberly
Published in Cancer cell (10.12.2018)
Published in Cancer cell (10.12.2018)
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Abstract 2441: CDK12/13 inhibition cooperates with the Ewing sarcoma oncoprotein EWS/FLI to attenuate homologous recombination repair in Ewing sarcoma cells
Balboni, Amanda, Stolte, Björn, Kalev, Peter, Kwiatkowski, Nicholas, Zhang, Tinghu, Abraham, Brian, Alexe, Gabriela, Chowdhury, Dipanjan, Young, Richard A., Gray, Nathanael S., Stegmaier, Kimberly
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
Abstract B50: Targeting EWS/FLI fusion oncoprotein stability/degradation in Ewing sarcoma
Seong, Bo Kyung Alex, Lin, Shan, Donovan, Katherine, Robichaud, Amanda, Stolte, Bjorn, Wang, Emily, Dharia, Neekesh, Nabet, Behnam, Piccioni, Federica, Gray, Nathanael, Fischer, Eric, Stegmaier, Kimberly
Published in Cancer research (Chicago, Ill.) (15.07.2020)
Published in Cancer research (Chicago, Ill.) (15.07.2020)
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Abstract 1118: Synthetic lethality of CDK12 inhibition in tumors with EWS/FLI rearrangements
Balboni, Amanda L., Stolte, Bjorn, Conway, Amy Saur, Alexe, Gabriela, Wang, Emily Jue, Kwiatkowski, Nicholas, Zhang, Tinghu, Abraham, Brian J., Kalev, Peter, Chowdhury, Dipanjan, Benes, Cyril H., Young, Richard A., Gray, Nathanael S., Stegmaier, Kimberly
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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