Spiro-1-benzofuranpiperidinylalkanoic acids as a novel and selective sphingosine S1P5 receptor agonist chemotype
Stoit, Axel R., Lange, Jos H.M., Coolen, Hein K.A.C., Rensink, Annemieke, van den Hoogenband, Adri, den Hartog, Arnold P., van Schaik, Sjoerd, Kruse, Chris G.
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
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Journal Article
Design, Synthesis and Biological Activity of Rigid Cannabinoid CB1 Receptor Antagonists
Stoit, Axel Reinhard, Lange, Jos Hubertus Maria, Hartog, Arnold Peter den, Ronken, Eric, Tipker, Koos, Stuivenberg, Herman Heinrich van, Dijksman, Jessica Adriana Rigtje, Wals, Henri Cornelis, Kruse, Chris Gerrit
Published in Chemical & pharmaceutical bulletin (01.08.2002)
Published in Chemical & pharmaceutical bulletin (01.08.2002)
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Journal Article
7-Azaindole derivatives as potential partial nicotinic agonists
Stoit, Axel R., den Hartog, Arnold P., Mons, Harry, van Schaik, Sjoerd, Barkhuijsen, Nynke, Stroomer, Cees, Coolen, Hein K.A.C., Reinders, Jan Hendrik, Adolfs, Tiny J.P., van der Neut, Martina, Keizer, Hiskias, Kruse, Chris G.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Journal Article
Spiro-1-benzofuranpiperidinylalkanoic acids as a novel and selective sphingosine S1P(5) receptor agonist chemotype
Stoit, Axel R., Lange, Jos H. M., Coolen, Hein K. A. C., Rensink, Annemieke, van den Hoogenband, Adri, den Hartog, Arnold P., van Schaik, Sjoerd, Kruse, Chris G.
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
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Journal Article
Synthesis and differential functionalisation of pyrrolidine and piperidine based spirodiamine scaffolds
Weinberg, Kamil, Stoit, Axel, Kruse, Chris G., Haddow, Mairi F., Gallagher, Timothy
Published in Tetrahedron (10.06.2013)
Published in Tetrahedron (10.06.2013)
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Journal Article
Spiro-1-benzofuranpiperidinylalkanoic acids as a novel and selective sphingosine S1P 5 receptor agonist chemotype
Stoit, Axel R, Lange, Jos H M, Coolen, Hein K A C, Rensink, Annemieke, van den Hoogenband, Adri, den Hartog, Arnold P, van Schaik, Sjoerd, Kruse, Chris G
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
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Published in Bioorganic & medicinal chemistry letters (01.02.2018)
Journal Article
SPIRO-CYCLIC AMINE DERIVATIVES AS S1P MODULATORS
VAN DONGEN MARIA J.P, STOIT AXEL, COOLEN HEIN K.A.C, IWEMA BAKKER WOUTER I, LEFLEMME NICOLAS J. L.D
Year of Publication 15.05.2013
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Year of Publication 15.05.2013
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(THIO)MORPHOLINE DERIVATIVES AS S1P MODULATORS
RONKEN ERIC, COOLEN HEIN K.A.C, STOIT AXEL, IWEMA BAKKER WOUTER I, VAN DER KAM ELIZABETH, MONS HARMEN, FRANKENA JURJEN
Year of Publication 20.08.2012
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Year of Publication 20.08.2012
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SILDENAFIL N-OXIDE AS PRODRUG
TULP MARTINUS TH. M, TURSKI LECHOSLAW A, KRUSE CORNELIS G, STOIT AXEL, VADER SANDER
Year of Publication 13.05.2010
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Year of Publication 13.05.2010
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N-OXIDES OF VENLAFAXINE AND O-DESMETHYLVENLAFAXINE AS PRODRUGS
TURSKI LECHOSLAW A, KRUSE CORNELIS G, STOIT AXEL, VADER SANDER, TULP MARTINUS TH.M
Year of Publication 21.04.2010
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Year of Publication 21.04.2010
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Spiro-cyclic amine derivatives as S1P modulators
Stoit, Axel, Iwema Bakker, Wouter I, Coolen, Hein K. A. C, Hobson, Adrian, Leflemme, Nicolas J.-L. D, van Dongen, Maria J. P
Year of Publication 30.08.2022
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Year of Publication 30.08.2022
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SPIRO-CYCLIC AMINE DERIVATIVES AS S1P MODULATORS
Leflemme, Nicolas J.-L.D, Stoit, Axel, Iwema Bakker, Wouter I, van Dongen, Maria J.P, Hobson, Adrian, Coolen, Hein K.A.C
Year of Publication 06.05.2021
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Year of Publication 06.05.2021
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SPIRO-CYCLIC AMINE DERIVATIVES AS S1P MODULATORS
IWEMA BAKKER, WOUTER I, HOBSON, ADRIAN D, COOLEN, HEIN K.A.C, VAN DONGEN, MARIA J.P, STOIT, AXEL, LEFLEMME, NICOLAS J.-L.D
Year of Publication 10.03.2020
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Year of Publication 10.03.2020
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Spiro-cyclic amine derivatives as S1P modulators
Stoit, Axel, Iwema Bakker, Wouter I, Coolen, Hein K. A. C, Hobson, Adrian, Leflemme, Nicolas J.-L. D, van Dongen, Maria J. P
Year of Publication 20.10.2020
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Year of Publication 20.10.2020
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SPIRO-CYCLIC AMINE DERIVATIVES AS S1P MODULATORS
Leflemme, Nicolas J.-L.D, Stoit, Axel, Iwema Bakker, Wouter I, van Dongen, Maria J.P, Hobson, Adrian, Coolen, Hein K.A.C
Year of Publication 18.07.2019
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Year of Publication 18.07.2019
Patent
Spiro-cyclic amine derivatives as S1P modulators
Stoit, Axel, Iwema Bakker, Wouter I, Coolen, Hein K. A. C, Hobson, Adrian, Leflemme, Nicolas J.-L. D, van Dongen, Maria J. P
Year of Publication 15.01.2019
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Year of Publication 15.01.2019
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SPIRO-CYCLIC AMINE DERIVATIVES AS S1P MODULATORS
LEFLEMME NICOLAS J-LD, STOIT AXEL, VAN DONGEN MARIA J P, IWENA BAKKER WOUTER I, COOLEN HEIN K A C, HOBSON ADRIAN D
Year of Publication 19.12.2018
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Year of Publication 19.12.2018
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