Macrocyclic Carbon-Linked Pyrazoles As Novel Inhibitors of MCL‑1
Demin, Samuël, Peschiulli, Aldo, Velter, Adriana I., Vos, Ann, De Boeck, Benoît, Miller, Bradley, Rombouts, Frederik J. R., Reuillon, Tristan, Lento, William, Blanco, Maria Dominguez, Jouffroy, Matthieu, Steyvers, Helena, Bekkers, Mariette, Altrocchi, Cristina, Pietrak, Beth, Koo, Seong Joo, Szewczuk, Lawrence, Attar, Ricardo, Philippar, Ulrike
Published in ACS medicinal chemistry letters (13.07.2023)
Published in ACS medicinal chemistry letters (13.07.2023)
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Abstract 2133: In pursuit of MCL-1 inhibitors with improved therapeutic window for the treatment of hematological malignancies: Discovery of JNJ-4355
Rombouts, Frederik J., William, Lento, Velter, Ingrid, Vos, Ann, Peschiulli, Aldo, Tristan, Reuillon, Blanco, Maria Dominguez, Jouffroy, Matthieu, McQueen, Lisa, Steyvers, Helena, Bekkers, Mariette, Altrocchi, Cristina, Pietrak, Beth, Koo, Seong Joo, Szewczuk, Lawrence, Walker, David, Packman, Kathryn, Bueters, Ruud, Vinken, Petra, Johnson, Amy, Attar, Ricardo, Philippar, Ulrike
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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