Design, synthesis, and neuraminidase inhibitory activity of GS-4071 analogues that utilize a novel hydrophobic paradigm
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Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
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Design and characterization of an engineered gp41 protein from human immunodeficiency virus-1 as a tool for drug discovery
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Published in Journal of computer-aided molecular design (01.01.2007)
Published in Journal of computer-aided molecular design (01.01.2007)
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An Unusual Intramolecular Hetero-Diels−Alder Cycloaddition
Stoner, Eric J, Allen, Michael S, Christesen, Alan C, Henry, Rodger F, Hollis, L. Steven, Keyes, Robert, Marsden, Ian, Rehm, Tamara C, Shiroor, Sandeep G, Soni, Niru B, Stewart, Kent D
Published in Journal of organic chemistry (15.04.2005)
Published in Journal of organic chemistry (15.04.2005)
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NOVEL TRICYCLIC COMPOUNDS
WOLLER KEVIN R, FRANK KRISTINE E, ERICSSON ANNA M, VOSS JEFFREY W, FRIEDMAN MICHAEL, WISHART NEIL, MORYTKO MICHAEL J, CALDERWOOD DAVID J, FIAMENGO BRYAN A, WALLACE GRIER A, WANG LU, JOSEPHSOHN NATHAN S, ARGIRIADI MARIA A, GOEDKEN ERIC R, GEORGE DAWN M, LI BIQIN C, STEWART KENT D
Year of Publication 12.09.2018
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Year of Publication 12.09.2018
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A Novel, Picomolar Inhibitor of Human Immunodeficiency Virus Type 1 Protease
Sham, Hing L, Zhao, Chen, Stewart, Kent D, Betebenner, David A, Lin, Shuqun, Park, Chang H, Kong, Xiang-P, Rosenbrook, William, Herrin, Thomas, Madigan, Darold, Vasavanonda, Suthida, Lyons, Nicholas, Molla, Akhter, Saldivar, Ayda, Marsh, Kennan C, McDonald, Edith, Wideburg, Norman E, Denissen, Jon F, Robins, Terrel, Kempf, Dale J, Plattner, Jacob J, Norbeck, Daniel W
Published in Journal of medicinal chemistry (19.01.1996)
Published in Journal of medicinal chemistry (19.01.1996)
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NOVEL TRICYCLIC COMPOUNDS
WOLLER KEVIN R, FRANK KRISTINE E, ERICSSON ANNA M, VOSS JEFFREY W, FRIEDMAN MICHAEL, WISHART NEIL, MORYTKO MICHAEL J, CALDERWOOD DAVID J, FIAMENGO BRYAN A, WALLACE GRIER A, WANG LU, JOSEPHSOHN NATHAN S, ARGIRIADI MARIA A, GOEDKEN ERIC R, GEORGE DAWN M, LI BIQIN C, STEWART KENT D
Year of Publication 24.10.2017
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Year of Publication 24.10.2017
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Novel tricyclic compounds
WOLLER KEVIN R, FRANK KRISTINE E, ERICSSON ANNA M, VOSS JEFFREY W, FRIEDMAN MICHAEL, WISHART NEIL, MORYTKO MICHAEL J, CALDERWOOD DAVID J, FIAMENGO BRYAN A, WALLACE GRIER A, WANG LU, JOSEPHSOHN NATHAN S, ARGIRIADI MARIA A, GOEDKEN ERIC R, GEORGE DAWN M, LI BIQIN C, STEWART KENT D
Year of Publication 23.12.2016
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Year of Publication 23.12.2016
Patent
Host-guest complexation. 42. Preorganization strongly enhances the tendancy of hemispherands to form hemispheraplexes
Doxsee, Kenneth M, Feigel, Martin, Stewart, Kent D, Canary, Jimmy W, Knobler, Carolyn B, Cram, Donald J
Published in Journal of the American Chemical Society (01.05.1987)
Published in Journal of the American Chemical Society (01.05.1987)
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URACIL OR THYMINE DERIVATIVE FOR TREATING HEPATITIS C
HENRY RODGER F, LIU YAYA, LOU XIAOCHUN, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, FRANCZYK II THADDEUS S, ROCKWAY TODD W, HUANG PEGGY P, FLENTGE CHARLES A, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, MARING CLARENCE J, BARNES DAVID M, PRATT JOHN K, DONNER PAMELA L, CHEN SHUANG, WAGNER ROLF, HENGEVELD JOHN E, RANDOLPH JOHN T, TUFANO MICHAEL D, LONGENECKER KENTON L, MOTTER CHRISTOPHER E, LIU DACHUN, KRUEGER ALLAN C, KOTECKI BRIAN J, HAIGHT ANTHONY R, ZHANG GEOFF G. Z, STEWART KENT D
Year of Publication 20.10.2015
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Year of Publication 20.10.2015
Patent
Discovery of 3H-Benzo[4,5]thieno[3,2-d)pyrimidin-4-ones as Potent, Highly Selective, and Orally Bioavailable Inhibitors of the Human Protooncogene Proviral Insertion Site in Moloney Murine Leukemia Virus (PIM) Kinases
Tao, Zhi-Fu, Hasvold, Lisa A., Leverson, Joel D., Han, Edward K., Guan, Ran, Johnson, Eric F., Stoll, Vincent S., Stewart, Kent D., Stamper, Geoff, Soni, Nirupama, Bouska, Jennifer J., Luo, Yan, Sowin, Thomas J., Lin, Nan-Horng, Giranda, Vincent S., Rosenberg, Saul H., Penning, Thomas D.
Published in Journal of medicinal chemistry (12.11.2009)
Published in Journal of medicinal chemistry (12.11.2009)
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NOVEL TRICYCLIC COMPOUNDS
WOLLER KEVIN R, FRANK KRISTINE E, ERICSSON ANNA M, VOSS JEFFREY W, FRIEDMAN MICHAEL, WISHART NEIL, MORYTKO MICHAEL J, CALDERWOOD DAVID J, FIAMENGO BRYAN A, WALLACE GRIER A, WANG LU, JOSEPHSOHN NATHAN S, ARGIRIADI MARIA A, GOEDKEN ERIC R, GEORGE DAWN M, LI BIQIN C, STEWART KENT D
Year of Publication 06.02.2014
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Year of Publication 06.02.2014
Patent
NOVEL TRICYCLIC COMPOUNDS
WOLLER KEVIN R, FRANK KRISTINE E, HOEMANN MICHAEL Z, ERICSSON ANNA M, VOSS JEFFREY W, FRIEDMAN MICHAEL, WISHART NEIL, MORYTKO MICHAEL J, CALDERWOOD DAVID J, FIAMENGO BRYAN A, WALLACE GRIER A, WANG LU, JOSEPHSOHN NATHAN S, ARGIRIADI MARIA A, GOEDKEN ERIC R, BREINLINGER ERIC C, GEORGE DAWN M, SOMAL GAGANDEEP, MULLEN KELLY D, LI BIQIN C, STEWART KENT D
Year of Publication 18.09.2012
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Year of Publication 18.09.2012
Patent
NOVEL TRICYCLIC COMPOUNDS
WOLLER KEVIN R, FRANK KRISTINE E, ERICSSON ANNA M, VOSS JEFFREY W, FRIEDMAN MICHAEL, WISHART NEIL, MORYTKO MICHAEL J, CALDERWOOD DAVID J, FIAMENGO BRYAN A, WALLACE GRIER A, WANG LU, JOSEPHSOHN NATHAN S, ARGIRIADI MARIA A, GOEDKEN ERIC R, GEORGE DAWN M, LI BIQIN C, STEWART KENT D
Year of Publication 21.02.2011
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Year of Publication 21.02.2011
Patent
The Drug Guru Project
Stewart, Kent D, Shanley, Jason, Ahmed, Karam B. Alsayyed, Bowen, J. Phillip
Published in Bioisosteres in Medicinal Chemistry (22.08.2012)
Published in Bioisosteres in Medicinal Chemistry (22.08.2012)
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Book Chapter
URACIL OR THYMINE DERIVATIVE FOR TREATING HEPATITIS C
HENRY RODGER F, LIU YAYA, LOU XIAOCHUN, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, FRANCZYK II THADDEUS S, ROCKWAY TODD W, HUANG PEGGY P, FLENTGE CHARLES A, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, MARING CLARENCE J, BARNES DAVID M, PRATT JOHN K, DONNER PAMELA L, CHEN SHUANG, WAGNER ROLF, HENGEVELD JOHN E, RANDOLPH JOHN T, TUFANO MICHAEL D, LONGENECKER KENTON L, MOTTER CHRISTOPHER E, LIU DACHUN, KRUEGER ALLAN C, KOTECKI BRIAN J, HAIGHT ANTHONY R, ZHANG GEOFF G. Z, STEWART KENT D
Year of Publication 22.06.2010
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Year of Publication 22.06.2010
Patent
Abstract C202: Discovery and initial characterization of the clinical compound ABT-348, a potent inhibitor of the VEGF, PDGF, and Aurora kinase families
Curtin, Michael L., Heyman, Robin, Frey, Robin R., Soni, Niru B., Marcotte, Patick A., Pease, Lori J., Glaser, Keith B., Magoc, Terrance J., Tapang, Paul, Albert, Daniel H., Osterling, Donald J., Olson, Amanda M., Bouska, Jennifer J., Guan, Zhiwen, Martin, Ruth L., Stewart, Kent D., Tse, Chris, Davidsen, Steven K., Michaelides, Michael R.
Published in Molecular cancer therapeutics (12.11.2011)
Published in Molecular cancer therapeutics (12.11.2011)
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