TCFH–NMI: Direct Access to N‑Acyl Imidazoliums for Challenging Amide Bond Formations
Beutner, Gregory L, Young, Ian S, Davies, Merrill L, Hickey, Matthew R, Park, Hyunsoo, Stevens, Jason M, Ye, Qingmei
Published in Organic letters (20.07.2018)
Published in Organic letters (20.07.2018)
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Journal Article
A Multi-Objective Active Learning Platform and Web App for Reaction Optimization
Torres, Jose Antonio Garrido, Lau, Sii Hong, Anchuri, Pranay, Stevens, Jason M., Tabora, Jose E., Li, Jun, Borovika, Alina, Adams, Ryan P., Doyle, Abigail G.
Published in Journal of the American Chemical Society (02.11.2022)
Published in Journal of the American Chemical Society (02.11.2022)
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Journal Article
Identifying general reaction conditions by bandit optimization
Wang, Jason Y., Stevens, Jason M., Kariofillis, Stavros K., Tom, Mai-Jan, Golden, Dung L., Li, Jun, Tabora, Jose E., Parasram, Marvin, Shields, Benjamin J., Primer, David N., Hao, Bo, Del Valle, David, DiSomma, Stacey, Furman, Ariel, Zipp, G. Greg, Melnikov, Sergey, Paulson, James, Doyle, Abigail G.
Published in Nature (London) (29.02.2024)
Published in Nature (London) (29.02.2024)
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Journal Article
Direct Lewis Acid Catalyzed Conversion of Enantioenriched N‑Acyloxazolidinones to Chiral Esters, Amides, and Acids
Stevens, Jason M, Parra-Rivera, Ana Cristina, Dixon, Darryl D, Beutner, Gregory L, DelMonte, Albert J, Frantz, Doug E, Janey, Jacob M, Paulson, James, Talley, Michael R
Published in Journal of organic chemistry (07.12.2018)
Published in Journal of organic chemistry (07.12.2018)
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Journal Article
Utilizing Native Directing Groups: Synthesis of a Selective IKur Inhibitor, BMS-919373, via a Regioselective C–H Arylation
Wisniewski, Steven R, Stevens, Jason M, Yu, Miao, Fraunhoffer, Kenneth J, Romero, Evan O, Savage, Scott A
Published in Journal of organic chemistry (19.04.2019)
Published in Journal of organic chemistry (19.04.2019)
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Journal Article
Coupling-Condensation Strategy for the Convergent Synthesis of an Imidazole-Fused 2‑Aminoquinoline NLRP3 Agonist
Bi, Cong, Chadwick, James, Davies, Merrill L., DelMonte, Albert J., Geng, Peng, Glace, Andrew W., Green, Rebecca A., Gurak, John A., Haley, Matthew W., He, Brian L., Inankur, Bahar, Jamison, Christopher R., Joe, Candice L., Kolotuchin, Sergei, Lin, Dong, Lou, Sha, Nye, Jeffrey, Ortiz, Adrian, Purdum, Geoffrey E., Rosso, Victor W., Shah, Mansi, Simmons, Eric M., Stevens, Jason M., Strotman, Neil A., Tan, Yichen, Zhang, Ling
Published in Journal of organic chemistry (06.01.2023)
Published in Journal of organic chemistry (06.01.2023)
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Journal Article
CITU: A Peptide and Decarboxylative Coupling Reagent
deGruyter, Justine N., Malins, Lara R., Wimmer, Laurin, Clay, Khalyd J., Lopez-Ogalla, Javier, Qin, Tian, Cornella, Josep, Liu, Zhiqing, Che, Guanda, Bao, Denghui, Stevens, Jason M., Qiao, Jennifer X., Allen, Martin P., Poss, Michael A., Baran, Phil S.
Published in Organic letters (17.11.2017)
Published in Organic letters (17.11.2017)
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Journal Article
Systematic Optimization of a Robust Telescoped Process for a BTK Inhibitor with Atropisomer Control by High-Throughput Experimentation, Design of Experiments, and Linear Regression
Gonzalez, Federico Lora, Wisniewski, Steven R, Katipally, Kishta, Stevens, Jason M, Rosso, Victor, Mack, Brendan, Razler, Thomas M
Published in Organic process research & development (21.06.2019)
Published in Organic process research & development (21.06.2019)
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Journal Article
Revisiting the Cleavage of Evans Oxazolidinones with LiOH/H2O2
Beutner, Gregory L, Cohen, Benjamin M, DelMonte, Albert J, Dixon, Darryl D, Fraunhoffer, Kenneth J, Glace, Andrew W, Lo, Ehrlic, Stevens, Jason M, Vanyo, Dale, Wilbert, Christopher
Published in Organic process research & development (19.07.2019)
Published in Organic process research & development (19.07.2019)
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Journal Article
Utilizing Native Directing Groups: Synthesis of a Selective I Kur Inhibitor, BMS-919373, via a Regioselective C-H Arylation
Wisniewski, Steven R, Stevens, Jason M, Yu, Miao, Fraunhoffer, Kenneth J, Romero, Evan O, Savage, Scott A
Published in Journal of organic chemistry (19.04.2019)
Published in Journal of organic chemistry (19.04.2019)
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Journal Article
Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor
Fraunhoffer, Kenneth J, DelMonte, Albert J, Beutner, Gregory L, Bultman, Michael S, Camacho, Kathryn, Cohen, Benjamin, Dixon, Darryl D, Fan, Yu, Fanfair, Dayne, Freitag, Adam J, Glace, Andrew W, Gonzalez-Bobes, Francisco, Gujjar, Manjunath, Haley, Matthew W, Hickey, Matthew R, Ho, Jeanne, Iyer, Vidya, Maity, Prantik, Patel, Sunil, Rosso, Victor W, Schmidt, Michael A, Stevens, Jason M, Tan, Yichen, Wilbert, Christopher, Young, Ian S, Yu, Miao
Published in Organic process research & development (15.11.2019)
Published in Organic process research & development (15.11.2019)
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Journal Article
Synthesis and SAR of vinca alkaloid analogues
Voss, Matthew E., Ralph, Jeffery M., Xie, Dejian, Manning, David D., Chen, Xinchao, Frank, Anthony J., Leyhane, Andrew J., Liu, Lei, Stevens, Jason M., Budde, Cheryl, Surman, Matthew D., Friedrich, Thomas, Peace, Denise, Scott, Ian L., Wolf, Mark, Johnson, Randall
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Journal Article
Advancing Base Metal Catalysis through Data Science: Insight and Predictive Models for Ni-Catalyzed Borylation through Supervised Machine Learning
Stevens, Jason M., Li, Jun, Simmons, Eric M., Wisniewski, Steven R., DiSomma, Stacey, Fraunhoffer, Kenneth J., Geng, Peng, Hao, Bo, Jackson, Erika W.
Published in Organometallics (25.07.2022)
Published in Organometallics (25.07.2022)
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