Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa
Cotman, Andrej Emanuel, Durcik, Martina, Benedetto Tiz, Davide, Fulgheri, Federica, Secci, Daniela, Sterle, Maša, Možina, Štefan, Skok, Žiga, Zidar, Nace, Zega, Anamarija, Ilaš, Janez, Peterlin Mašič, Lucija, Tomašič, Tihomir, Hughes, Diarmaid, Huseby, Douglas L., Cao, Sha, Garoff, Linnéa, Berruga Fernández, Talía, Giachou, Paraskevi, Crone, Lisa, Simoff, Ivailo, Svensson, Richard, Birnir, Bryndis, Korol, Sergiy V., Jin, Zhe, Vicente, Francisca, Ramos, Maria C., de la Cruz, Mercedes, Glinghammar, Björn, Lenhammar, Lena, Henderson, Sara R., Mundy, Julia E. A., Maxwell, Anthony, Stevenson, Clare E. M., Lawson, David M., Janssen, Guido V., Sterk, Geert Jan, Kikelj, Danijel
Published in Journal of medicinal chemistry (26.01.2023)
Published in Journal of medicinal chemistry (26.01.2023)
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Journal Article
Development of narrow-spectrum topoisomerase-targeting antibacterials against mycobacteria
Sterle, Maša, Habjan, Eva, Piga, Martina, Peršolja, Peter, Durcik, Martina, Dernovšek, Jaka, Szili, Petra, Czikkely, Marton Simon, Zidar, Nace, Janez, Ilaš, Pal, Csaba, Accetto, Tomaž, Pardo, Luis A., Kikelj, Danijel, Peterlin Mašič, Lucija, Tomašič, Tihomir, Bitter, Wilbert, Cotman, Andrej Emanuel, Speer, Alexander, Zega, Anamarija
Published in European journal of medicinal chemistry (05.10.2024)
Published in European journal of medicinal chemistry (05.10.2024)
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Journal Article
Practical Synthesis and Application of Halogen-Doped Pyrrole Building Blocks
Cotman, Andrej Emanuel, Guérin, Thomas, Kovačević, Ivana, Benedetto Tiz, Davide, Durcik, Martina, Fulgheri, Federica, Možina, Štefan, Secci, Daniela, Sterle, Maša, Ilaš, Janez, Zega, Anamarija, Zidar, Nace, Mašič, Lucija Peterlin, Tomašič, Tihomir, Leroux, Frédéric R, Hanquet, Gilles, Kikelj, Danijel
Published in ACS omega (13.04.2021)
Published in ACS omega (13.04.2021)
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Journal Article
Exploring the 5‑Substituted 2‑Aminobenzothiazole-Based DNA Gyrase B Inhibitors Active against ESKAPE Pathogens
Sterle, Maša, Durcik, Martina, Stevenson, Clare E. M., Henderson, Sara R., Szili, Petra Eva, Czikkely, Marton, Lawson, David M., Maxwell, Anthony, Cahard, Dominique, Kikelj, Danijel, Zidar, Nace, Pal, Csaba, Mašič, Lucija Peterlin, Ilaš, Janez, Tomašič, Tihomir, Cotman, Andrej Emanuel, Zega, Anamarija
Published in ACS omega (11.07.2023)
Published in ACS omega (11.07.2023)
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Journal Article
Hydrogen-Bonding Ability of Noyori–Ikariya Catalysts Enables Stereoselective Access to CF3‑Substituted syn-1,2-Diols via Dynamic Kinetic Resolution
Sterle, Maša, Huš, Matej, Lozinšek, Matic, Zega, Anamarija, Cotman, Andrej Emanuel
Published in ACS catalysis (05.05.2023)
Published in ACS catalysis (05.05.2023)
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Journal Article
Catalytic Stereoconvergent Synthesis of Homochiral β‑CF3, β‑SCF3, and β‑OCF3 Benzylic Alcohols
Cotman, Andrej Emanuel, Dub, Pavel A., Sterle, Maša, Lozinšek, Matic, Dernovšek, Jaka, Zajec, Živa, Zega, Anamarija, Tomašič, Tihomir, Cahard, Dominique
Published in ACS Organic & Inorganic Au (05.10.2022)
Published in ACS Organic & Inorganic Au (05.10.2022)
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Journal Article
New Quinolinone O-GlcNAc Transferase Inhibitors Based on Fragment Growth
Weiss, Matjaž, Loi, Elena M, Sterle, Maša, Balsollier, Cyril, Tomašič, Tihomir, Pieters, Roland J, Gobec, Martina, Anderluh, Marko
Published in Frontiers in chemistry (14.04.2021)
Published in Frontiers in chemistry (14.04.2021)
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Journal Article
Hydrogen-Bonding Ability of Noyori-Ikariya Catalysts Enables Stereoselective Access to CF 3 -Substituted syn -1,2-Diols via Dynamic Kinetic Resolution
Sterle, Maša, Huš, Matej, Lozinšek, Matic, Zega, Anamarija, Cotman, Andrej Emanuel
Published in ACS catalysis (05.05.2023)
Published in ACS catalysis (05.05.2023)
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Journal Article
Discovery of KV1.3 ion channel inhibitors: Medicinal chemistry approaches and challenges
Gubič, Špela, Hendrickx, Louise A., Toplak, Žan, Sterle, Maša, Peigneur, Steve, Tomašič, Tihomir, Pardo, Luis A., Tytgat, Jan, Zega, Anamarija, Mašič, Lucija P.
Published in Medicinal research reviews (01.07.2021)
Published in Medicinal research reviews (01.07.2021)
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Journal Article
New N -phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity
Cotman, Andrej Emanuel, Fulgheri, Federica, Piga, Martina, Peršolja, Peter, Tiz, Davide Benedetto, Skok, Žiga, Durcik, Martina, Sterle, Maša, Dernovšek, Jaka, Cruz, Cristina D., Tammela, Päivi, Szili, Petra Éva, Daruka, Lejla, Pál, Csaba, Zega, Anamarija, Mašič, Lucija Peterlin, Ilaš, Janez, Tomašič, Tihomir, Kikelj, Danijel, Zidar, Nace
Published in RSC advances (04.09.2024)
Published in RSC advances (04.09.2024)
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Journal Article
Discovery of K V 1.3 ion channel inhibitors: Medicinal chemistry approaches and challenges
Gubič, Špela, Hendrickx, Louise A, Toplak, Žan, Sterle, Maša, Peigneur, Steve, Tomašič, Tihomir, Pardo, Luis A, Tytgat, Jan, Zega, Anamarija, Mašič, Lucija P
Published in Medicinal research reviews (01.07.2021)
Published in Medicinal research reviews (01.07.2021)
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Journal Article
Catalytic Stereoconvergent Synthesis of Homochiral β-CF 3 , β-SCF 3 , and β-OCF 3 Benzylic Alcohols
Cotman, Andrej Emanuel, Dub, Pavel A., Sterle, Maša, Lozinšek, Matic, Dernovšek, Jaka, Zajec, Živa, Zega, Anamarija, Tomašič, Tihomir, Cahard, Dominique
Published in ACS Organic & Inorganic Au (05.10.2022)
Published in ACS Organic & Inorganic Au (05.10.2022)
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Journal Article