Stereochemistry and molecular pharmacology of ( S)-thio-ATPA, a new potent and selective GluR5 agonist
Stensbøl, Tine B., Jensen, Henrik S., Nielsen, Birgitte, Johansen, Tommy N., Egebjerg, Jan, Frydenvang, Karla, Krogsgaard-Larsen, Povl
Published in European journal of pharmacology (12.01.2001)
Published in European journal of pharmacology (12.01.2001)
Get full text
Journal Article
Genetic predictors of response to serotonergic and noradrenergic antidepressants in major depressive disorder: a genome-wide analysis of individual-level data and a meta-analysis
Tansey, Katherine E, Guipponi, Michel, Perroud, Nader, Bondolfi, Guido, Domenici, Enrico, Evans, David, Hall, Stephanie K, Hauser, Joanna, Henigsberg, Neven, Hu, Xiaolan, Jerman, Borut, Maier, Wolfgang, Mors, Ole, O'Donovan, Michael, Peters, Tim J, Placentino, Anna, Rietschel, Marcella, Souery, Daniel, Aitchison, Katherine J, Craig, Ian, Farmer, Anne, Wendland, Jens R, Malafosse, Alain, Holmans, Peter, Lewis, Glyn, Lewis, Cathryn M, Stensbøl, Tine Bryan, Kapur, Shitij, McGuffin, Peter, Uher, Rudolf
Published in PLoS medicine (01.10.2012)
Published in PLoS medicine (01.10.2012)
Get full text
Journal Article
Novel class of potent 4-arylalkyl substituted 3-isoxazolol GABA(A) antagonists: Synthesis, pharmacology, and molecular modeling
Frolund, B, Jorgensen, AT, Tagmose, L, Stensbol, TB, Vestergaard, HT, Engblom, C, Kristiansen, U, Sanchez, C, Krogsgaard-Larsen, P, Liljefors, T
Published in Journal of medicinal chemistry (06.06.2002)
Published in Journal of medicinal chemistry (06.06.2002)
Get full text
Journal Article
Potent 4-aryl- or 4-arylalkyl-substituted 3-isoxazolol GABA(A) antagonists: Synthesis, pharmacology, and molecular modeling
Frolund, B, Jensen, LS, Guandalini, L, Canillo, C, Vestergaard, HT, Kristiansen, U, Nielsen, B, Stensbol, TB, Madsen, C, Krogsgaard-Larszen, P, Liljefors, T
Published in Journal of medicinal chemistry (27.01.2005)
Published in Journal of medicinal chemistry (27.01.2005)
Get full text
Journal Article
Ibotenic acid and thioibotenic acid: a remarkable difference in activity at group III metabotropic glutamate receptors
Hermit, Mette B., Greenwood, Jeremy R., Nielsen, Birgitte, Bunch, Lennart, Jørgensen, Charlotte G., Vestergaard, Henrik T., Stensbøl, Tine B., Sanchez, Connie, Krogsgaard-Larsen, Povl, Madsen, Ulf, Bräuner-Osborne, Hans
Published in European journal of pharmacology (23.02.2004)
Published in European journal of pharmacology (23.02.2004)
Get full text
Journal Article
Three-Dimensional Structure of the Ligand-Binding Core of GluR2 in Complex with the Agonist (S)-ATPA: Implications for Receptor Subunit Selectivity
Lunn, Marie-Louise, Hogner, Anders, Stensbøl, Tine B, Gouaux, Eric, Egebjerg, Jan, Kastrup, Jette S
Published in Journal of medicinal chemistry (27.02.2003)
Published in Journal of medicinal chemistry (27.02.2003)
Get full text
Journal Article
The AMPA Receptor Binding Site: Focus on Agonists and Competitive Antagonists
Stensbol, Tine, Madsen, Ulf, Krogsgaard-Larsen, Povl
Published in Current pharmaceutical design (01.05.2002)
Published in Current pharmaceutical design (01.05.2002)
Get full text
Journal Article
Synthesis and Anticonvulsant Activity of Novel Bicyclic Acidic Amino Acids
Conti, Paola, De Amici, Marco, Joppolo di Ventimiglia, Samuele, Stensbøl, Tine B, Madsen, Ulf, Bräuner-Osborne, Hans, Russo, Emilio, De Sarro, Giovambattista, Bruno, Giuseppe, Micheli, Carlo De
Published in Journal of medicinal chemistry (03.07.2003)
Published in Journal of medicinal chemistry (03.07.2003)
Get full text
Journal Article
Design, Synthesis, and Pharmacological Characterization of Novel, Potent NMDA Receptor Antagonists
Conti, Paola, De Amici, Marco, Grazioso, Giovanni, Roda, Gabriella, Barberis Negra, Federico F, Nielsen, Birgitte, Stensbøl, Tine B, Madsen, Ulf, Bräuner-Osborne, Hans, Frydenvang, Karla, De Sarro, Giovambattista, Toma, Lucio, De Micheli, Carlo
Published in Journal of medicinal chemistry (30.12.2004)
Published in Journal of medicinal chemistry (30.12.2004)
Get full text
Journal Article
A novel class of potent 3-isoxazolol GABA(A) antagonists: design, synthesis, and pharmacology
Frolund, B, Tagmose, L, Liljefors, T, Stensbol, TB, Engblom, C, Kristiansen, U, Krogsgaard-Larsen, P
Published in Journal of medicinal chemistry (28.12.2000)
Published in Journal of medicinal chemistry (28.12.2000)
Get full text
Journal Article
Tetrazolyl isoxazole amino acids as ionotropic glutamate receptor antagonists: Synthesis, modelling and molecular pharmacology
Frølund, Bente, Greenwood, Jeremy R., Holm, Mai M., Egebjerg, Jan, Madsen, Ulf, Nielsen, Birgitte, Bräuner-Osborne, Hans, Stensbøl, Tine B., Krogsgaard-Larsen, Povl
Published in Bioorganic & medicinal chemistry (15.09.2005)
Published in Bioorganic & medicinal chemistry (15.09.2005)
Get full text
Journal Article
(S)-Homo-AMPA, a specific agonist at the mGlu(6) subtype of metabotropic glutamic acid receptors
Ahmadian, H, Nielsen, B, Brauner-Osborne, H, Johansen, TN, Stensbol, TB, Slok, FA, Sekiyama, N, Nakanishi, S, KrogsgaardLarsen, P, Madsen, U
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
Get full text
Journal Article
Novel 1-Hydroxyazole Bioisosteres of Glutamic Acid. Synthesis, Protolytic Properties, and Pharmacology
Stensbøl, Tine B, Uhlmann, Peter, Morel, Sandrine, Eriksen, Birgitte L, Felding, Jakob, Kromann, Hasse, Hermit, Mette B, Greenwood, Jeremy R, Braüner-Osborne, Hans, Madsen, Ulf, Junager, Finn, Krogsgaard-Larsen, Povl, Begtrup, Mikael, Vedsø, Per
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
Get full text
Journal Article
(S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid, a Potent and Selective Agonist at the GluR5 Subtype of Ionotropic Glutamate Receptors. Synthesis, Modeling, and Molecular Pharmacology
Brehm, Lotte, Greenwood, Jeremy R, Hansen, Kasper B, Nielsen, Birgitte, Egebjerg, Jan, Stensbøl, Tine B, Bräuner-Osborne, Hans, Sløk, Frank A, Kronborg, Tine T. A, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (10.04.2003)
Published in Journal of medicinal chemistry (10.04.2003)
Get full text
Journal Article
Synthesis and Enantiopharmacology of New AMPA-Kainate Receptor Agonists
Conti, Paola, De Amici, Marco, De Sarro, Giovambattista, Rizzo, Milena, Stensbøl, Tine Bryan, Bräuner-Osborne, Hans, Madsen, Ulf, Toma, Lucio, De Micheli, Carlo
Published in Journal of medicinal chemistry (07.10.1999)
Published in Journal of medicinal chemistry (07.10.1999)
Get full text
Journal Article
Inhibitors of AMPA and Kainate Receptors
Madsen, U., Stensbol, T., Krogsgaard-Larsen, P.
Published in Current medicinal chemistry (01.09.2001)
Published in Current medicinal chemistry (01.09.2001)
Get full text
Journal Article
Structural Determinants of AMPA Agonist Activity in Analogues of 2-Amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic Acid: Synthesis and Pharmacology
Bang-Andersen, Benny, Ahmadian, Haleh, Lenz, Sibylle M, Stensbøl, Tine B, Madsen, Ulf, Bøgesø, Klaus P, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (14.12.2000)
Published in Journal of medicinal chemistry (14.12.2000)
Get full text
Journal Article
2-Amino-3-(3-hydroxy-1,2,5-thiadiazol-4-yl)propionic acid: Resolution, absolute stereochemistry and enantiopharmacology at glutamate receptors
JOHANSEN, Tommy N, JANIN, Yves L, NIELSEN, Birgitte, FRYDENVANG, Karla, BRÄUNER-OSBORNE, Hans, STENSBØL, Tine B, VOGENSEN, Stine B, MADSEN, Ulf, KROGSGAARD-LARSEN, Povl
Published in Bioorganic & medicinal chemistry (01.07.2002)
Published in Bioorganic & medicinal chemistry (01.07.2002)
Get full text
Journal Article
Design of novel conformationally restricted analogues of glutamic acid
Conti, Paola, De Amici, Marco, Roda, Gabriella, Vistoli, Giulio, Stensbøl, Tine Bryan, Bräuner-Osborne, Hans, Madsen, Ulf, Toma, Lucio, De Micheli, Carlo
Published in Tetrahedron (24.02.2003)
Published in Tetrahedron (24.02.2003)
Get full text
Journal Article