Identification of Positive Allosteric Modulators of Glycine Receptors from a High-Throughput Screen Using a Fluorescent Membrane Potential Assay
Stead, Clara, Brown, Adam, Adams, Cathryn, Nickolls, Sarah J, Young, Gareth, Kammonen, Juha, Pryde, David, Cawkill, Darren
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Published in Journal of biomolecular screening (01.12.2016)
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Design and Identification of a Novel, Functionally Subtype Selective GABAA Positive Allosteric Modulator (PF-06372865)
Owen, Robert M, Blakemore, David, Cao, Lishuang, Flanagan, Neil, Fish, Rebecca, Gibson, Karl R, Gurrell, Rachel, Huh, Chan Woo, Kammonen, Juha, Mortimer-Cassen, Elisabeth, Nickolls, Sarah A, Omoto, Kiyoyuki, Owen, Dafydd, Pike, Andy, Pryde, David C, Reynolds, David S, Roeloffs, Rosemarie, Rose, Colin, Stead, Clara, Takeuchi, Mifune, Warmus, Joseph S, Watson, Christine
Published in Journal of medicinal chemistry (27.06.2019)
Published in Journal of medicinal chemistry (27.06.2019)
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Pharmacology in translation: the preclinical and early clinical profile of the novel α2/3 functionally selective GABAA receptor positive allosteric modulator PF‐06372865
Nickolls, Sarah A, Gurrell, Rachel, Amerongen, Guido, Kammonen, Juha, Cao, Lishuang, Brown, Adam R, Stead, Clara, Mead, Andy, Watson, Christine, Hsu, Cathleen, Owen, Robert M, Pike, Andy, Fish, Rebecca L, Chen, Laigao, Qiu, Ruolun, Morris, Evan D, Feng, Gang, Whitlock, Mark, Gorman, Donal, Gerven, Joop, Reynolds, David S, Dua, Pinky, Butt, Richard P
Published in British journal of pharmacology (01.02.2018)
Published in British journal of pharmacology (01.02.2018)
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Design and Identification of a Novel, Functionally Subtype Selective GABA(A) Positive Allosteric Modulator (PF-06372865)
Owen, Robert M., Blakemore, David, Cao, Lishuan, Flanagan, Neil, Fish, Rebecca, Gibson, Karl R., Gurrell, Rachel, Huh, Chan Woo, Kammonen, Juha, Mortimer-Cassen, Elisabeth, Nickolls, Sarah A., Omoto, Kiyoyuki, Owen, Dafydd, Pike, Andy, Pryde, David C., Reynolds, David S., Roeloffs, Rosemarie, Rose, Colin, Stead, Clara, Takeuchi, Mifune, Warmus, Joseph S., Watson, Christine
Published in Journal of medicinal chemistry (27.06.2019)
Published in Journal of medicinal chemistry (27.06.2019)
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Journal Article
Pharmacology in translation: the preclinical and early clinical profile of the novel α2/3 functionally selective GABA A receptor positive allosteric modulator PF-06372865
Nickolls, Sarah A, Gurrell, Rachel, van Amerongen, Guido, Kammonen, Juha, Cao, Lishuang, Brown, Adam R, Stead, Clara, Mead, Andy, Watson, Christine, Hsu, Cathleen, Owen, Robert M, Pike, Andy, Fish, Rebecca L, Chen, Laigao, Qiu, Ruolun, Morris, Evan D, Feng, Gang, Whitlock, Mark, Gorman, Donal, van Gerven, Joop, Reynolds, David S, Dua, Pinky, Butt, Richard P
Published in British journal of pharmacology (01.02.2018)
Published in British journal of pharmacology (01.02.2018)
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