Allosteric PI3Kα Inhibition Overcomes On-target Resistance to Orthosteric Inhibitors Mediated by Secondary PIK3CA Mutations
Varkaris, Andreas, Fece de la Cruz, Ferran, Martin, Elizabeth E, Norden, Bryanna L, Chevalier, Nicholas, Kehlmann, Allison M, Leshchiner, Ignaty, Barnes, Haley, Ehnstrom, Sara, Stavridi, Anastasia-Maria, Yuan, Xin, Kim, Janice S, Ellis, Haley, Papatheodoridi, Alkistis, Gunaydin, Hakan, Danysh, Brian P, Parida, Laxmi, Sanidas, Ioannis, Ji, Yongli, Lau, Kayao, Wulf, Gerburg M, Bardia, Aditya, Spring, Laura M, Isakoff, Steven J, Lennerz, Jochen K, Del Vecchio, Kathryn, Pierce, Levi, Pazolli, Ermira, Getz, Gad, Corcoran, Ryan B, Juric, Dejan
Published in Cancer discovery (08.02.2024)
Published in Cancer discovery (08.02.2024)
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