Discovery of Mer kinase inhibitors by virtual screening using Structural Protein–Ligand Interaction Fingerprints
Da, C., Stashko, M., Jayakody, C., Wang, X., Janzen, W., Frye, S., Kireev, D.
Published in Bioorganic & medicinal chemistry (01.03.2015)
Published in Bioorganic & medicinal chemistry (01.03.2015)
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Nonsteroidal Selective Glucocorticoid Modulators: the Effect of C-5 Alkyl Substitution on the Transcriptional Activation/Repression Profile of 2,5-Dihydro-10-methoxy-2,2,4-trimethyl-1H-[1]benzopyrano[3,4-f]quinolines
Elmore, Steven W, Coghlan, Michael J, Anderson, David D, Pratt, John K, Green, Brian E, Wang, Alan X, Stashko, Michael A, Lin, Chun W, Tyree, Curtis M, Miner, Jeffery N, Jacobson, Peer B, Wilcox, Denise M, Lane, Benjamin C
Published in Journal of medicinal chemistry (06.12.2001)
Published in Journal of medicinal chemistry (06.12.2001)
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Synthesis and Characterization of Non-Steroidal Ligands for the Glucocorticoid Receptor: Selective Quinoline Derivatives with Prednisolone-Equivalent Functional Activity
Coghlan, Michael J, Kym, Philip R, Elmore, Steven W, Wang, Alan X, Luly, Jay R, Wilcox, Denise, Stashko, Michael, Lin, Chun-Wei, Miner, Jeffrey, Tyree, Curtis, Nakane, Masaki, Jacobson, Peer, Lane, Benjamin C
Published in Journal of medicinal chemistry (30.08.2001)
Published in Journal of medicinal chemistry (30.08.2001)
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ABT-431: the diacetyl prodrug of A-86929, a potent and selective dopamine D1 receptor agonist: in vitro characterization and effects in animal models of Parkinson's disease
Shiosaki, K, Jenner, P, Asin, K E, Britton, D R, Lin, C W, Michaelides, M, Smith, L, Bianchi, B, Didomenico, S, Hodges, L, Hong, Y, Mahan, L, Mikusa, J, Miller, T, Nikkel, A, Stashko, M, Witte, D, Williams, M
Published in The Journal of pharmacology and experimental therapeutics (01.01.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1996)
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Characterization of cloned human dopamine D1 receptor-mediated calcium release in 293 cells
Lin, C W, Miller, T R, Witte, D G, Bianchi, B R, Stashko, M, Manelli, A M, Frail, D E
Published in Molecular pharmacology (01.01.1995)
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Published in Molecular pharmacology (01.01.1995)
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In vitro enzymatic assays of protein tyrosine phosphatase 1B
Lubben, T, Clampit, J, Stashko, M, Trevillyan, J, Jirousek, M R
Published in Current protocols in pharmacology (01.08.2001)
Published in Current protocols in pharmacology (01.08.2001)
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Persistent activation of the dopamine D1 receptor contributes to prolonged receptor desensitization: studies with A-77636
Lin, C W, Bianchi, B R, Miller, T R, Stashko, M A, Wang, S S, Curzon, P, Bednarz, L, Asin, K E, Britton, D R
Published in The Journal of pharmacology and experimental therapeutics (01.03.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1996)
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Novel Asp32-Replacement Tetrapeptide Analogs as Potent and Selective CCK-A Agonists
Elliott, Richard L, Kopecka, Hana, Tufano, Michael D, Shue, Youe-Kong, Gauri, Andre J, Lin, Chun-Wel, Bianchi, Bruce R, Miller, Thomas R, Witte, David G
Published in Journal of medicinal chemistry (01.05.1994)
Published in Journal of medicinal chemistry (01.05.1994)
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Tetrapeptide CCK agonists: structure-activity studies on modifications at the N-terminus
Elliott, Richard L, Kopecka, Hana, Bennett, Michael J, Shue, Youe Kong, Craig, Richard, Lin, Chun Wel, Bianchi, Bruce R, Miller, Thomas R, Witte, David G
Published in Journal of medicinal chemistry (01.01.1994)
Published in Journal of medicinal chemistry (01.01.1994)
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trans-Activation and Repression Properties of the Novel Nonsteroid Glucocorticoid Receptor Ligand 2,5-Dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5-(1-methylcyclohexen-3-y1)-1H-[1]benzopyrano[3,4-f]quinoline (A276575) and Its Four Stereoisomers
Lin, Chun Wel, Nakane, Masaki, Stashko, Mike, Falls, Doug, Kuk, Jane, Miller, Loan, Huang, Ruth, Tyree, Curtis, Miner, Jeffrey N, Rosen, John, Kym, Philip R, Coghlan, Mike J, Carter, George, Lane, Ben C
Published in Molecular pharmacology (01.08.2002)
Published in Molecular pharmacology (01.08.2002)
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Discovery of a Potent, Selective Protein Tyrosine Phosphatase 1B Inhibitor Using a Linked-Fragment Strategy
Szczepankiewicz, Bruce G, Liu, Gang, Hajduk, Philip J, Abad-Zapatero, Cele, Pei, Zhonghua, Xin, Zhili, Lubben, Thomas H, Trevillyan, James M, Stashko, Michael A, Ballaron, Stephen J, Liang, Heng, Huang, Flora, Hutchins, Charles W, Fesik, Stephen W, Jirousek, Michael R
Published in Journal of the American Chemical Society (09.04.2003)
Published in Journal of the American Chemical Society (09.04.2003)
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Selective Protein Tyrosine Phosphatase 1B Inhibitors: Targeting the Second Phosphotyrosine Binding Site with Non-Carboxylic Acid-Containing Ligands
Liu, Gang, Xin, Zhili, Liang, Heng, Abad-Zapatero, Cele, Hajduk, Philip J, Janowick, David A, Szczepankiewicz, Bruce G, Pei, Zhonghua, Hutchins, Charles W, Ballaron, Stephen J, Stashko, Michael A, Lubben, Thomas H, Berg, Cathy E, Rondinone, Cristina M, Trevillyan, James M, Jirousek, Michael R
Published in Journal of medicinal chemistry (31.07.2003)
Published in Journal of medicinal chemistry (31.07.2003)
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Nonsteroidal Selective Glucocorticoid Modulators: The Effect of C-10 Substitution on Receptor Selectivity and Functional Potency of 5-Allyl-2,5-dihydro-2,2,4-trimethyl-1H-[1]benzopyrano[3,4-f]quinolines
Kym, Philip R, Kort, Michael E, Coghlan, Michael J, Moore, Jimmie L, Tang, Rui, Ratajczyk, James D, Larson, Daniel P, Elmore, Steven W, Pratt, John K, Stashko, Michael A, Falls, H. Douglass, Lin, Chun W, Nakane, Masake, Miller, Loan, Tyree, Curtis M, Miner, Jeffery N, Jacobson, Peer B, Wilcox, Denise M, Nguyen, Phong, Lane, Benjamin C
Published in Journal of medicinal chemistry (13.03.2003)
Published in Journal of medicinal chemistry (13.03.2003)
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Discovery of ((4R,5S)-5-Amino-4-(2,4,5- trifluorophenyl)cyclohex-1-enyl)-(3- (trifluoromethyl)-5,6-dihydro- [1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)methanone (ABT-341), a Highly Potent, Selective, Orally Efficacious, and Safe Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes
Pei, Zhonghua, Li, Xiaofeng, von Geldern, Thomas W, Madar, David J, Longenecker, Kenton, Yong, Hong, Lubben, Thomas H, Stewart, Kent D, Zinker, Bradley A, Backes, Bradley J, Judd, Andrew S, Mulhern, Mathew, Ballaron, Stephen J, Stashko, Michael A, Mika, Amanda K, Beno, David W. A, Reinhart, Glenn A, Fryer, Ryan M, Preusser, Lee C, Kempf-Grote, Anita J, Sham, Hing L, Trevillyan, James M
Published in Journal of medicinal chemistry (02.11.2006)
Published in Journal of medicinal chemistry (02.11.2006)
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Minor Structural Differences in Boc-CCK-4 Derivatives Dictate Affinity and Selectivity for CCK-A and CCK-B Receptors
Shiosaki, Kazumi, Lin, Chun Wel, Kopecka, Hana, Bianchi, Bruce, Miller, Thomas, Stashko, Michael, Witte, David
Published in Journal of medicinal chemistry (28.03.1997)
Published in Journal of medicinal chemistry (28.03.1997)
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Identification of a monoacid-Based, cell permeable, selective inhibitor of protein tyrosine phosphatase 1B
Xin, Zhili, Liu, Gang, Abad-Zapatero, Cele, Pei, Zhonghua, Szczepankiewicz, Bruce G., Li, Xiaofeng, Zhang, Tianyuan, Hutchins, Charles W., Hajduk, Philip J., Ballaron, Stephen J., Stashko, Michael A., Lubben, Thomas H., Trevillyan, James M., Jirousek, Michael R.
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
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Journal Article
Potent, selective inhibitors of protein tyrosine phosphatase 1B
Xin, Zhili, Oost, Thorsten K, Abad-Zapatero, Cele, Hajduk, Philip J, Pei, Zhonghua, Szczepankiewicz, Bruce G, Hutchins, Charles W, Ballaron, Steve J, Stashko, Mike A, Lubben, Tom, Trevillyan, James M, Jirousek, Mike R, Liu, Gang
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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Journal Article
Differentiation of in vitro transcriptional repression and activation profiles of selective glucocorticoid modulators
Elmore, Steven W, Pratt, John K, Coghlan, Michael J, Mao, Yue, Green, Brian E, Anderson, David D, Stashko, Michael A, Lin, Chun W, Falls, Douglas, Nakane, Masaki, Miller, Loan, Tyree, Curtis M, Miner, Jeffrey N, Lane, Ben
Published in Bioorganic & medicinal chemistry letters (05.04.2004)
Published in Bioorganic & medicinal chemistry letters (05.04.2004)
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Journal Article
A-86929: A selective dopamine D 1 receptor agonist with anti-Parkinsonian efficacy in MPTP-lesioned primate models
Shiosaki, K., Jenner, P., Bedard, P., Lin, C.W., Britton, D., Bianchi, B., Grondin, R., Hong, Y., Michaelides, M., Miller, T., Smith, L., Stashko, M., Williams, M.
Published in Pharmacological research (1995)
Published in Pharmacological research (1995)
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Journal Article
A-86929: A selective dopamine D1 receptor agonist with anti-Parkinsonian efficacy in MPTP-lesioned primate models
Shiosaki, K., Jenner, P., Bedard, P., Lin, C.W., Britton, D., Bianchi, B., Grondin, R., Hong, Y., Michaelides, M., Miller, T., Smith, L., Stashko, M., Williams, M.
Published in Pharmacological research (01.01.1995)
Published in Pharmacological research (01.01.1995)
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