Dihydropyrancarboxamides Related to Zanamivir: A New Series of Inhibitors of Influenza Virus Sialidases. 1. Discovery, Synthesis, Biological Activity, and Structure−Activity Relationships of 4-Guanidino- and 4-Amino-4H-pyran-6-carboxamides
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Synthesis and influenza virus sialidase inhibitory activity of analogues of 4-guanidino-Neu5Ac2en (GG167) with modified 5-substituents
Smith, PW, Starkey, ID, Howes, PD, Sollis, SL, Keeling, SP, Cherry, PC, von Itzstein, M, Wu, WY, Jin, B
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Synthesis and influenza virus sialidase inhibitory activity of the 5-desacetamido analogue of 2,3-didehydro-2,4-dideoxy-4-guanidinyl-N-acetylneuraminic acid (GG167)
Starkey, Ian D., Mahmoudian, Mahmoud, Noble, David, Smith, Paul W., Cherry, Peter C., Howes, Peter D., Sollis, Steven L.
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Published in Tetrahedron letters (09.01.1995)
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KITCHIN, J, BETHELL, RC, CAMMACK, N, DOLAN, S, EVANS, DN, HOLMAN, S, HOLMES, DS, MCMEEKIN, P, MO, CL, NIELAND, N, ORR, DC, SAUNDERS, J, SHENOY, BEV, STARKEY, ID, STORER, R
Published in Journal of medicinal chemistry (28.10.1994)
Published in Journal of medicinal chemistry (28.10.1994)
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