Synthesis and Serotonergic Activity of 3-[2-(Pyrrolidin-1-yl)ethyl]indoles: Potent Agonists for the h5-HT1D Receptor with High Selectivity over the h5-HT1B Receptor
Sternfeld, Francine, Guiblin, Alexander R, Jelley, Richard A, Matassa, Victor G, Reeve, Austin J, Hunt, Peter A, Beer, Margaret S, Heald, Anne, Stanton, Josephine A, Sohal, Bindi, Watt, Alan P, Street, Leslie J
Published in Journal of medicinal chemistry (25.02.1999)
Published in Journal of medicinal chemistry (25.02.1999)
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3-[3-(Piperidin-1-yl)propyl]indoles as Highly Selective h5-HT1D Receptor Agonists
Russell, Michael G. N, Matassa, Victor G, Pengilley, Roy R, van Niel, Monique B, Sohal, Bindi, Watt, Alan P, Hitzel, Laure, Beer, Margaret S, Stanton, Josephine A, Broughton, Howard B, Castro, José L
Published in Journal of medicinal chemistry (02.12.1999)
Published in Journal of medicinal chemistry (02.12.1999)
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3-(Piperazinylpropyl)indoles: Selective, Orally Bioavailable h5-HT1D Receptor Agonists as Potential Antimigraine Agents
Chambers, Mark S, Street, Leslie J, Goodacre, Simon, Hobbs, Sarah C, Hunt, Peter, Jelley, Richard A, Matassa, Victor G, Reeve, Austin J, Sternfeld, Francine, Beer, Margaret S, Stanton, Josephine A, Rathbone, Denise, Watt, Alan P, MacLeod, Angus M
Published in Journal of medicinal chemistry (25.02.1999)
Published in Journal of medicinal chemistry (25.02.1999)
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Enhancement of Oral Absorption in Selective 5-HT1D Receptor Agonists: Fluorinated 3-[3-(Piperidin-1-yl)propyl]indoles
Castro, José L, Collins, Ian, Russell, Michael G. N, Watt, Alan P, Sohal, Bindi, Rathbone, Denise, Beer, Margaret S, Stanton, Josephine A
Published in Journal of medicinal chemistry (16.07.1998)
Published in Journal of medicinal chemistry (16.07.1998)
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Synthesis and Biological Activity of 3-[2-(Dimethylamino)ethyl]-5-[(1,1-dioxo-5-methyl-1,2,5-thiadiazolidin-2-yl)methyl]-1H-indole and Analogs: Agonists for the 5-HT1D Receptor
Castro, Jose L, Baker, Raymond, Guiblin, Alexander R, Hobbs, Sarah C, Jenkins, Matthew R, Russell, Michael G. N, Beer, Margaret S, Stanton, Josephine A, Scholey, Kate
Published in Journal of medicinal chemistry (01.09.1994)
Published in Journal of medicinal chemistry (01.09.1994)
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Journal Article
Selective, Orally Active 5-HT1D Receptor Agonists as Potential Antimigraine Agents
MacLeod, Angus M, Street, Leslie J, Reeve, Austin J, Jelley, Richard A, Sternfeld, Francine, Beer, Margaret S, Stanton, Josephine A, Watt, Alan P, Rathbone, Denise, Matassa, Victor G
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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Journal Article
3-[2-(Pyrrolidin-1-yl)ethyl]indoles and 3-[3-(Piperidin-1-yl)propyl]indoles: Agonists for the h5-HT1D Receptor with High Selectivity over the h5-HT1B Subtype
Castro, José L, Street, Leslie J, Guiblin, Alexander R, Jelley, Richard A, Russell, Michael G. N, Sternfeld, Francine, Beer, Margaret S, Stanton, Josephine A, Matassa, Victor G
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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Journal Article
Fluorination of 3-(3-(Piperidin-1-yl)propyl)indoles and 3-(3-(Piperazin-1-yl)propyl)indoles Gives Selective Human 5-HT1D Receptor Ligands with Improved Pharmacokinetic Profiles
van Niel, Monique B, Collins, Ian, Beer, Margaret S, Broughton, Howard B, Cheng, Susan K. F, Goodacre, Simon C, Heald, Anne, Locker, Karen L, MacLeod, Angus M, Morrison, Denise, Moyes, Christopher R, O'Connor, Desmond, Pike, Andrew, Rowley, Michael, Russell, Michael G. N, Sohal, Balbinder, Stanton, Josephine A, Thomas, Steven, Verrier, Hugh, Watt, Alan P, Castro, José L
Published in Journal of medicinal chemistry (17.06.1999)
Published in Journal of medicinal chemistry (17.06.1999)
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Edg2 Receptor Functionality: Giα1 Coexpression and Fusion Protein Studies
McAllister, George, Stanton, Josephine A., Salim, Kamran, Handford, Emma J., Beer, Margaret S.
Published in Molecular pharmacology (01.08.2000)
Published in Molecular pharmacology (01.08.2000)
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Journal Article
Edg2 Receptor Functionality: Giα1 Coexpression and Fusion Protein Studies
George McAllister, Josephine A. Stanton, Kamran Salim, Emma J. Handford, Margaret S. Beer
Published in Molecular pharmacology (01.08.2000)
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Published in Molecular pharmacology (01.08.2000)
Journal Article
3-[3-(Piperidin-1-yl)propyl]indoles as highly selective h5-HT(1D) receptor agonists
Russell, M G, Matassa, V G, Pengilley, R R, van Niel, M B, Sohal, B, Watt, A P, Hitzel, L, Beer, M S, Stanton, J A, Broughton, H B, Castro, J L
Published in Journal of medicinal chemistry (02.12.1999)
Published in Journal of medicinal chemistry (02.12.1999)
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Journal Article
2,7-diazabicyclo[3.3.0]octanes as novel h5-HT receptor agonists
Russell, M G, Beer, M S, Stanton, J A, Sohal, B, Mortishire-Smith, R J, Castro, J L
Published in Bioorganic & medicinal chemistry letters (06.09.1999)
Published in Bioorganic & medicinal chemistry letters (06.09.1999)
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Journal Article
Synthesis and Serotonergic Activity of N,N-Dimethyl-2-[5-(1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethylamine and Analogs: Potent Agonists for 5-HT1D Receptors
Street, Leslie J, Baker, Raymond, Davey, William B, Guiblin, Alexander R, Jelley, Richard A, Reeve, Austin J, Routledge, Helen, Sternfeld, Francine, Watt, Alan P
Published in Journal of medicinal chemistry (01.05.1995)
Published in Journal of medicinal chemistry (01.05.1995)
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