SIRT5 stabilizes mitochondrial glutaminase and supports breast cancer tumorigenesis
Greene, Kai Su, Lukey, Michael J., Wang, Xueying, Blank, Bryant, Druso, Joseph E., Lin, Miao-chong J., Stalnecker, Clint A., Zhang, Chengliang, Abril, Yashira Negrón, Erickson, Jon W., Wilson, Kristin F., Lin, Hening, Weiss, Robert S., Cerione, Richard A.
Published in Proceedings of the National Academy of Sciences - PNAS (26.12.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (26.12.2019)
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Journal Article
Combination Therapies with CDK4/6 Inhibitors to Treat KRAS-Mutant Pancreatic Cancer
Goodwin, Craig M, Waters, Andrew M, Klomp, Jennifer E, Javaid, Sehrish, Bryant, Kirsten L, Stalnecker, Clint A, Drizyte-Miller, Kristina, Papke, Bjoern, Yang, Runying, Amparo, Amber M, Ozkan-Dagliyan, Irem, Baldelli, Elisa, Calvert, Valerie, Pierobon, Mariaelena, Sorrentino, Jessica A, Beelen, Andrew P, Bublitz, Natalie, Lüthen, Mareen, Wood, Kris C, Petricoin, Emanuel F, Sers, Christine, McRee, Autumn J, Cox, Adrienne D, Der, Channing J
Published in Cancer research (Chicago, Ill.) (04.01.2023)
Published in Cancer research (Chicago, Ill.) (04.01.2023)
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Journal Article
Mechanism by which a recently discovered allosteric inhibitor blocks glutamine metabolism in transformed cells
Stalnecker, Clint A., Ulrich, Scott M., Li, Yunxing, Ramachandran, Sekar, McBrayer, Mary Kate, DeBerardinis, Ralph J., Cerione, Richard A., Erickson, Jon W.
Published in Proceedings of the National Academy of Sciences - PNAS (13.01.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (13.01.2015)
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Journal Article
Concurrent Inhibition of IGF1R and ERK Increases Pancreatic Cancer Sensitivity to Autophagy Inhibitors
Stalnecker, Clint A, Grover, Kajal R, Edwards, A Cole, Coleman, Michael F, Yang, Runying, DeLiberty, Jonathan M, Papke, Björn, Goodwin, Craig M, Pierobon, Mariaelena, Petricoin, Emanuel F, Gautam, Prson, Wennerberg, Krister, Cox, Adrienne D, Der, Channing J, Hursting, Stephen D, Bryant, Kirsten L
Published in Cancer research (Chicago, Ill.) (15.02.2022)
Published in Cancer research (Chicago, Ill.) (15.02.2022)
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Journal Article
TEAD Inhibition Overcomes YAP1/TAZ-Driven Primary and Acquired Resistance to KRASG12C Inhibitors
Edwards, A Cole, Stalnecker, Clint A, Jean Morales, Alexis, Taylor, Khalilah E, Klomp, Jennifer E, Klomp, Jeffrey A, Waters, Andrew M, Sudhakar, Niranjan, Hallin, Jill, Tang, Tracy T, Olson, Peter, Post, Leonard, Christensen, James G, Cox, Adrienne D, Der, Channing J
Published in Cancer research (Chicago, Ill.) (15.12.2023)
Published in Cancer research (Chicago, Ill.) (15.12.2023)
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Journal Article
Conformational changes in the activation loop of mitochondrial glutaminase C: A direct fluorescence readout that distinguishes the binding of allosteric inhibitors from activators
Stalnecker, Clint A., Erickson, Jon W., Cerione, Richard A.
Published in The Journal of biological chemistry (14.04.2017)
Published in The Journal of biological chemistry (14.04.2017)
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Journal Article
Determining the ERK-regulated phosphoproteome driving KRAS-mutant cancer
Klomp, Jennifer E, Diehl, J Nathaniel, Klomp, Jeffrey A, Edwards, A Cole, Yang, Runying, Morales, Alexis J, Taylor, Khalilah E, Drizyte-Miller, Kristina, Bryant, Kirsten L, Schaefer, Antje, Johnson, Jared L, Huntsman, Emily M, Yaron, Tomer M, Pierobon, Mariaelena, Baldelli, Elisa, Prevatte, Alex W, Barker, Natalie K, Herring, Laura E, Petricoin, 3rd, Emanuel F, Graves, Lee M, Cantley, Lewis C, Cox, Adrienne D, Der, Channing J, Stalnecker, Clint A
Published in Science (American Association for the Advancement of Science) (07.06.2024)
Published in Science (American Association for the Advancement of Science) (07.06.2024)
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Journal Article
Mechanistic Basis of Glutaminase Activation: A KEY ENZYME THAT PROMOTES GLUTAMINE METABOLISM IN CANCER CELLS
Li, Yunxing, Erickson, Jon W, Stalnecker, Clint A, Katt, William P, Huang, Qingqiu, Cerione, Richard A, Ramachandran, Sekar
Published in The Journal of biological chemistry (30.09.2016)
Published in The Journal of biological chemistry (30.09.2016)
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Journal Article
Defining the KRAS- and ERK-dependent transcriptome in KRAS-mutant cancers
Klomp, Jeffrey A, Klomp, Jennifer E, Stalnecker, Clint A, Bryant, Kirsten L, Edwards, A Cole, Drizyte-Miller, Kristina, Hibshman, Priya S, Diehl, J Nathaniel, Lee, Ye S, Morales, Alexis J, Taylor, Khalilah E, Peng, Sen, Tran, Nhan L, Herring, Laura E, Prevatte, Alex W, Barker, Natalie K, Hover, Laura D, Hallin, Jill, Chowdhury, Saikat, Coker, Oluwadara, Lee, Hey Min, Goodwin, Craig M, Gautam, Prson, Olson, Peter, Christensen, James G, Shen, John P, Kopetz, Scott, Graves, Lee M, Lim, Kian-Huat, Wang-Gillam, Andrea, Wennerberg, Krister, Cox, Adrienne D, Der, Channing J
Published in Science (American Association for the Advancement of Science) (07.06.2024)
Published in Science (American Association for the Advancement of Science) (07.06.2024)
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Journal Article
CHK1 protects oncogenic KRAS-expressing cells from DNA damage and is a target for pancreatic cancer treatment
Klomp, Jennifer E, Lee, Ye S, Goodwin, Craig M, Papke, Björn, Klomp, Jeff A, Waters, Andrew M, Stalnecker, Clint A, DeLiberty, Jonathan M, Drizyte-Miller, Kristina, Yang, Runying, Diehl, J Nathaniel, Yin, Hongwei H, Pierobon, Mariaelena, Baldelli, Elisa, Ryan, Meagan B, Li, Siqi, Peterson, Jackson, Smith, Amber R, Neal, James T, McCormick, Aaron K, Kuo, Calvin J, Counter, Christopher M, Petricoin, 3rd, Emanuel F, Cox, Adrienne D, Bryant, Kirsten L, Der, Channing J
Published in Cell reports (Cambridge) (30.11.2021)
Published in Cell reports (Cambridge) (30.11.2021)
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Journal Article
Detection of phenotype‐specific therapeutic vulnerabilities in breast cells using a CRISPR loss‐of‐function screen
Barkovskaya, Anna, Goodwin, Craig M., Seip, Kotryna, Hilmarsdottir, Bylgja, Pettersen, Solveig, Stalnecker, Clint, Engebraaten, Olav, Briem, Eirikur, Der, Channing J., Moestue, Siver A., Gudjonsson, Thorarinn, Mælandsmo, Gunhild M., Prasmickaite, Lina
Published in Molecular oncology (01.08.2021)
Published in Molecular oncology (01.08.2021)
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Journal Article
Author Correction: Combination of ERK and autophagy inhibition as a treatment approach for pancreatic cancer
Bryant, Kirsten L, Stalnecker, Clint A, Zeitouni, Daniel, Klomp, Jennifer E, Peng, Sen, Tikunov, Andrey P, Gunda, Venugopal, Pierobon, Mariaelena, Waters, Andrew M, George, Samuel D, Tomar, Garima, Papke, Björn, Hobbs, G Aaron, Yan, Liang, Hayes, Tikvah K, Diehl, J Nathaniel, Goode, Gennifer D, Chaika, Nina V, Wang, Yingxue, Zhang, Guo-Fang, Witkiewicz, Agnieszka K, Knudsen, Erik S, Petricoin, 3rd, Emanuel F, Singh, Pankaj K, Macdonald, Jeffrey M, Tran, Nhan L, Lyssiotis, Costas A, Ying, Haoqiang, Kimmelman, Alec C, Cox, Adrienne D, Der, Channing J
Published in Nature medicine (01.06.2020)
Published in Nature medicine (01.06.2020)
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Journal Article
Balancing redox stress: anchorage-independent growth requires reductive carboxylation
Stalnecker, Clint A, Cluntun, Ahmad A, Cerione, Richard A
Published in Translational cancer research (01.09.2016)
Published in Translational cancer research (01.09.2016)
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Journal Article
Combination of ERK and autophagy inhibition as a treatment approach for pancreatic cancer
Bryant, Kirsten L, Stalnecker, Clint A, Zeitouni, Daniel, Klomp, Jennifer E, Peng, Sen, Tikunov, Andrey P, Gunda, Venugopal, Pierobon, Mariaelena, Waters, Andrew M, George, Samuel D, Tomar, Garima, Papke, Björn, Hobbs, G Aaron, Yan, Liang, Hayes, Tikvah K, Diehl, J Nathaniel, Goode, Gennifer D, Chaika, Nina V, Wang, Yingxue, Zhang, Guo-Fang, Witkiewicz, Agnieszka K, Knudsen, Erik S, Petricoin, 3rd, Emanuel F, Singh, Pankaj K, Macdonald, Jeffrey M, Tran, Nhan L, Lyssiotis, Costas A, Ying, Haoqiang, Kimmelman, Alec C, Cox, Adrienne D, Der, Channing J
Published in Nature medicine (01.04.2019)
Published in Nature medicine (01.04.2019)
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Journal Article
Characterization of the interactions of potent allosteric inhibitors with glutaminase C, a key enzyme in cancer cell glutamine metabolism
Huang, Qingqiu, Stalnecker, Clint, Zhang, Chengliang, McDermott, Lee A., Iyer, Prema, O’Neill, Jason, Reimer, Shawn, Cerione, Richard A., Katt, William P.
Published in The Journal of biological chemistry (09.03.2018)
Published in The Journal of biological chemistry (09.03.2018)
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