Synthesis, Potency, and in Vivo Evaluation of 2-Piperazin-1-ylquinoline Analogues as Dual Serotonin Reuptake Inhibitors and Serotonin 5-HT1A Receptor Antagonists
Zhou, Dahui, Stack, Gary P, Lo, Jennifer, Failli, Amedeo A, Evrard, Deborah A, Harrison, Boyd L, Hatzenbuhler, Nicole T, Tran, Megan, Croce, Susan, Yi, Soo, Golembieski, Jeannette, Hornby, Geoffrey A, Lai, Margaret, Lin, Qian, Schechter, Lee E, Smith, Deborah L, Shilling, Adam D, Huselton, Christine, Mitchell, Paul, Beyer, Chad E, Andree, Terrance H
Published in Journal of medicinal chemistry (13.08.2009)
Published in Journal of medicinal chemistry (13.08.2009)
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Journal Article
5-HT1A receptor antagonism reverses and prevents fluoxetine-induced sexual dysfunction in rats
Sukoff Rizzo, Stacey J., Pulicicchio, Claudine, Malberg, Jessica E., Andree, Terrance H., Stack, Gary P., Hughes, Zoë A., Schechter, Lee E., Rosenzweig-Lipson, Sharon
Published in The international journal of neuropsychopharmacology (01.09.2009)
Published in The international journal of neuropsychopharmacology (01.09.2009)
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Journal Article
Structure−Activity Relationships of the Cycloalkanol Ethylamine Scaffold: Discovery of Selective Norepinephrine Reuptake Inhibitors
Mahaney, Paige E, Gavrin, Lori K, Trybulski, Eugene J, Stack, Gary P, Vu, An T, Cohn, Stephen T, Ye, Fei, Belardi, Justin K, Santilli, Arthur A, Sabatucci, Joseph P, Leiter, Jennifer, Johnston, Grace H, Bray, Jenifer A, Burroughs, Kevin D, Cosmi, Scott A, Leventhal, Liza, Koury, Elizabeth J, Zhang, Yingru, Mugford, Cheryl A, Ho, Douglas M, Rosenzweig-Lipson, Sharon J, Platt, Brian, Smith, Valerie A, Deecher, Darlene C
Published in Journal of medicinal chemistry (10.07.2008)
Published in Journal of medicinal chemistry (10.07.2008)
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Journal Article
Novel pyridyl-fused 3-amino chroman derivatives with dual action at serotonin transporter and 5-HT1A receptor
DAHUI ZHOU, HATZENBUHLER, Nicole T, ANDREE, Terrance H, STACK, Gary P, GROSS, Jonathan L, HARRISON, Boyd L, EVRARD, Deborah A, CHLENOV, Michael, GOLEMBIESKI, Jeannette, HORNBY, Geoffrey, SCHECHTER, Lee E, SMITH, Deborah L
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
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Journal Article
Modulation of selective serotonin reuptake inhibitor and 5-HT1A antagonist activity in 8-aza-bicyclo[3.2.1]octane derivatives of 2,3-dihydro-1,4-benzodioxane
GILBERT, Adam M, STACK, Gary P, NILAKANTAN, Ramaswamy, KODAH, Jason, TRAN, Megan, SCERNI, Rosemary, XIAOJIE SHI, SMITH, Deborah L, ANDREE, Terrance H
Published in Bioorganic & medicinal chemistry letters (19.01.2004)
Published in Bioorganic & medicinal chemistry letters (19.01.2004)
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Journal Article
Synthesis, Potency, and in Vivo Evaluation of 2-Piperazin-1-ylquinoline Analogues as Dual Serotonin Reuptake Inhibitors and Serotonin 5-HT 1A Receptor Antagonists
Zhou, Dahui, Stack, Gary P., Lo, Jennifer, Failli, Amedeo A., Evrard, Deborah A., Harrison, Boyd L., Hatzenbuhler, Nicole T., Tran, Megan, Croce, Susan, Yi, Soo, Golembieski, Jeannette, Hornby, Geoffrey A., Lai, Margaret, Lin, Qian, Schechter, Lee E., Smith, Deborah L., Shilling, Adam D., Huselton, Christine, Mitchell, Paul, Beyer, Chad E., Andree, Terrance H.
Published in Journal of medicinal chemistry (13.08.2009)
Published in Journal of medicinal chemistry (13.08.2009)
Get full text
Journal Article
Novel pyridyl-fused 3-amino chroman derivatives with dual action at serotonin transporter and 5-HT sub(1A) receptor
Zhou, Dahui, Hatzenbuhler, Nicole T, Gross, Jonathan L, Harrison, Boyd L, Evrard, Deborah A, Chlenov, Michael, Golembieski, Jeannette, Hornby, Geoffrey, Schechter, Lee E, Smith, Deborah L, Andree, Terrance H, Stack, Gary P
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
Get full text
Journal Article
Novel pyridyl-fused 3-amino chroman derivatives with dual action at serotonin transporter and 5-HT 1A receptor
Zhou, Dahui, Hatzenbuhler, Nicole T., Gross, Jonathan L., Harrison, Boyd L., Evrard, Deborah A., Chlenov, Michael, Golembieski, Jeannette, Hornby, Geoffrey, Schechter, Lee E., Smith, Deborah L., Andree, Terrance H., Stack, Gary P.
Published in Bioorganic & medicinal chemistry letters (2007)
Published in Bioorganic & medicinal chemistry letters (2007)
Get full text
Journal Article
5-HT(1A) receptor antagonism reverses and prevents fluoxetine-induced sexual dysfunction in rats
Sukoff Rizzo, Stacey J, Pulicicchio, Claudine, Malberg, Jessica E, Andree, Terrance H, Stack, Gary P, Hughes, Zoë A, Schechter, Lee E, Rosenzweig-Lipson, Sharon
Published in The international journal of neuropsychopharmacology (01.09.2009)
Published in The international journal of neuropsychopharmacology (01.09.2009)
Get full text
Journal Article
Modulation of selective serotonin reuptake inhibitor and 5-HT 1A antagonist activity in 8-aza-bicyclo[3.2.1]octane derivatives of 2,3-dihydro-1,4-benzodioxane
Gilbert, Adam M., Stack, Gary P., Nilakantan, Ramaswamy, Kodah, Jason, Tran, Megan, Scerni, Rosemary, Shi, Xiaojie, Smith, Deborah L., Andree, Terrance H.
Published in Bioorganic & medicinal chemistry letters (2004)
Published in Bioorganic & medicinal chemistry letters (2004)
Get full text
Journal Article