Discovery of novel, potent and orally efficacious inhibitor of neutral amino acid transporter B0AT1 (SLC6A19)
Desai, Jigar, Patel, Bhaumin, Darji, Brijesh, Gite, Archana, Panchal, Nandini, Bhosale, Gokul, Shedage, Sandeep, Patel, Sandip, Kadam, Pravin, Patel, Gautam, Kumar Srivastava, Brijesh, Joharapurkar, Amit, Kshirsagar, Samadhan, Giri, Poonam, Bhayani, Hitesh, Patel, Ankit, Ghoshdastidar, Krishnarup, Bandyopadhyay, Debdutta, Kumar, Sanjay, Jain, Mukul, Sharma, Rajiv
Published in Bioorganic & medicinal chemistry letters (01.12.2021)
Published in Bioorganic & medicinal chemistry letters (01.12.2021)
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Journal Article
Diaryl Dihydropyrazole-3-carboxamides with Significant In Vivo Antiobesity Activity Related to CB1 Receptor Antagonism: Synthesis, Biological Evaluation, and Molecular Modeling in the Homology Model
Joharapurkar, Amit, Raval, Saurin, Patel, Jayendra Z, Soni, Rina, Raval, Preeti, Gite, Archana, Goswami, Amitgiri, Sadhwani, Nisha, Gandhi, Neha, Patel, Harilal, Mishra, Bhupendra, Solanki, Manish, Pandey, Bipin, Jain, Mukul R, Patel, Pankaj R
Published in Journal of medicinal chemistry (29.11.2007)
Published in Journal of medicinal chemistry (29.11.2007)
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Journal Article
Synthesis and antibacterial activity of 4,5,6,7-tetrahydro-thieno[3,2- c]pyridine quinolones
Srivastava, Brijesh Kumar, Solanki, Manish, Mishra, Bhupendra, Soni, Rina, Jayadev, Sanjaya, Valani, Darshan, Jain, Mukul, Patel, Pankaj R.
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
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Journal Article
Synthesis and in vitro antibacterial activities of novel oxazolidinones
Srivastava, Brijesh Kumar, Jain, Mukul R., Solanki, Manish, Soni, Rina, Valani, Darshan, Gupta, Sunil, Mishra, Bhupendra, Takale, Vijay, Kapadnis, Prashant, Patel, Harilal, Pandya, Purvi, Patel, Jayendra Z., Patel, Pankaj R.
Published in European journal of medicinal chemistry (01.04.2008)
Published in European journal of medicinal chemistry (01.04.2008)
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Journal Article
Novel 4-N-substituted aryl pent-2-ene-1,4-dione derivatives of piperazinyloxazolidinones as antibacterials
Lohray, Braj Bhushan, Lohray, Vidya Bhushan, Srivastava, Brijesh Kumar, Gupta, Sunil, Solanki, Manish, Pandya, Purvi, Kapadnis, Prashant
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
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Journal Article
Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide (SR141716) a potent CB1 receptor antagonist
Srivastava, Brijesh Kumar, Soni, Rina, Patel, Jayendra Z., Jha, Satadru, Shedage, Sandeep A., Gandhi, Neha, Sairam, Kalapatapu V. V. M., Pawar, Vishwanath, Sadhwani, Nisha, Mitra, Prasenjit, Jain, Mukul R., Patel, Pankaj R.
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
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Journal Article
Synthesis and in vitro antibacterial activity of novel methylamino piperidinyl oxazolidinones
Srivastava, Brijesh Kumar, Soni, Rina, Patel, Jayendra Z., Solanki, Manish, Valani, Darshan, Gupta, Sunil, Mishra, Bhupendra, Takale, Vijay, Pandya, Purvi, Jain, Mukul R., Patel, Pankaj R.
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
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Journal Article
Oxazolidinone: search for highly potent antibacterial
Lohray, Braj Bhushan, Lohray, Vidya Bhushan, Srivastava, Brijesh Kumar, Gupta, Sunil, Solanki, Manish, Kapadnis, Prashant, Takale, Vijay, Pandya, Purvi
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Journal Article
Novel Mannich ketones of oxazolidinones as antibacterial agents
Srivastava, Brijesh Kumar, Kapadnis, Prashant B., Pandya, Purvi, Lohray, Vidya Bhushan
Published in European journal of medicinal chemistry (01.11.2004)
Published in European journal of medicinal chemistry (01.11.2004)
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Journal Article
ZYDG2, a Potent, Selective, and Safe GPR40 Agonist for Treatment of Type 2 Diabetes
JAIN, MUKUL R., GIRI, SURESH R., TRIVEDI, CHITRANG J., BHOI, BIBHUTI B., RATH, AKSHYAYA CHANDAN, RATHOD, ROHAN MANUBHAI, SUNDAR, RAJESH, BANDYOPADHYAY, DEBDUTTA, RAMDHAVE, RASHMI, PATEL, GAUTAM D., SRIVASTAVA, BRIJESH KUMAR, DESAI, RANJIT C.
Published in Diabetes (New York, N.Y.) (01.07.2018)
Published in Diabetes (New York, N.Y.) (01.07.2018)
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Journal Article
Identification and preclinical characterization of a novel and potent poly (ADP-ribose) polymerase (PARP) inhibitor ZYTP1
Jain, Mukul R., Mohapatra, Jogeswar, Bandhyopadhyay, Debdutta, Chatterjee, Abhijit, Ghoshdastidar, Krishnarup, Patel, Dinesh, Patel, Ankit, Bhayani, Hitesh, Srivastava, Brijesh Kumar, Shedage, Sandeep A., Kadam, Pravin, Sundar, Rajesh, Patel, Harilal, Giri, Poonam, Patel, Prakash, Gupta, Laxmikant, Srinivas, Nuggehally R., Patel, Pankaj R., Desai, Ranjit C.
Published in Cancer chemotherapy and pharmacology (01.10.2018)
Published in Cancer chemotherapy and pharmacology (01.10.2018)
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Journal Article
Cannabinoid receptor 1 antagonist treatment induces glucagon release and shows an additive therapeutic effect with GLP-1 agonist in diet-induced obese mice
Patel, Kartikkumar Navinchandra, Joharapurkar, Amit Arvind, Patel, Vishal, Kshirsagar, Samadhan Govind, Bahekar, Rajesh, Srivastava, Brijesh Kumar, Jain, Mukul R
Published in Canadian journal of physiology and pharmacology (01.12.2014)
Published in Canadian journal of physiology and pharmacology (01.12.2014)
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Journal Article
Diaryl dihydropyrazole-3-carboxamides with significant in vivo antiobesity activity related to CBI receptor antagonism: Synthesis, biological evaluation, and molecular modeling in the homology model
Srivastava, Brijesh Kumar, Joharapurkar, Amit, Raval, Saurin, Patel, Jayendra Z., Soni, Rina, Raval, Preeti, Gite, Archana, Goswami, Amitgiri, Sadhwani, Nisha, Gandhi, Neha, Patel, Harilal, Mishra, Bhupendra, Solanki, Manish, Pandey, Bipin, Jain, Mukul R., Patel, Pankaj R.
Published in Journal of medicinal chemistry (29.11.2007)
Published in Journal of medicinal chemistry (29.11.2007)
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Journal Article
Discovery of novel, potent and orally efficacious inhibitor of neutral amino acid transporter B 0 AT1 (SLC6A19)
Desai, Jigar, Patel, Bhaumin, Darji, Brijesh, Gite, Archana, Panchal, Nandini, Bhosale, Gokul, Shedage, Sandeep, Patel, Sandip, Kadam, Pravin, Patel, Gautam, Kumar Srivastava, Brijesh, Joharapurkar, Amit, Kshirsagar, Samadhan, Giri, Poonam, Bhayani, Hitesh, Patel, Ankit, Ghoshdastidar, Krishnarup, Bandyopadhyay, Debdutta, Kumar, Sanjay, Jain, Mukul, Sharma, Rajiv
Published in Bioorganic & medicinal chemistry letters (01.12.2021)
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Published in Bioorganic & medicinal chemistry letters (01.12.2021)
Journal Article
Hair growth stimulator property of thienyl substituted pyrazole carboxamide derivatives as a cb1 receptor antagonist with in vivo antiobesity effect
Srivastava, Brijesh Kumar, Soni, Rina, Patel, Jayendra Z., Joharapurkar, Amit, Sadhwani, Nisha, Kshirsagar, Samadhan, Mishra, Bhupendra, Takale, Vijay, Gupta, Sunil, Pandya, Purvi, Kapadnis, Prashant, Solanki, Manish, Patel, Harilal, Mitra, Prasenjit, Jain, Mukul R., Patel, Pankaj R.
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Journal Article
Hair growth stimulator property of thienyl substituted pyrazole carboxamide derivatives as a cbl receptor antagonist with in vivo antiobesity effect
BRIJESH KUMAR SRIVASTAVA, SONI, Rina, KAPADNIS, Prashant, SOLANKI, Manish, PATEL, Harilal, MITRA, Prasenjit, JAIN, Mukul R, PATEL, Pankaj R, PATEL, Jayendra Z, JOHARAPURKAR, Amit, SADHWANI, Nisha, KSHIRSAGAR, Samadhan, MISHRA, Bhupendra, TAKALE, Vijay, GUPTA, Sunil, PANDYA, Purvi
Published in Bioorganic & medicinal chemistry letters (2009)
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Published in Bioorganic & medicinal chemistry letters (2009)
Journal Article
Bioisosteric replacement of dihydropyrazole of 4S-(-)-3-(4-chlorophenyl)-N-methyl-N'-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a potent CB1 receptor antagonist by imidazole and oxazole
Srivastava, Brijesh Kumar, Soni, Rina, Joharapurkar, Amit, Sairam, Kalapatapu V V M, Patel, Jayendra Z, Goswami, Amitgiri, Shedage, Sandeep A, Kar, Sidhartha S, Salunke, Rahul P, Gugale, Shivaji B, Dhawas, Amol, Kadam, Pravin, Mishra, Bhupendra, Sadhwani, Nisha, Unadkat, Vishal B, Mitra, Prasenjit, Jain, Mukul R, Patel, Pankaj R
Published in Bioorganic & medicinal chemistry letters (01.02.2008)
Published in Bioorganic & medicinal chemistry letters (01.02.2008)
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Journal Article