A synthetic triptycene bisquinone, which blocks nucleoside transport and induces DNA fragmentation, retains its cytotoxic efficacy in daunorubicin-resistant HL-60 cell lines
Wang, B, Wu, M, Perchellet, E M, McIlvain, C J, Sperfslage, B J, Huang, X, Tamura, M, Stephany, H A, Hua, D H, Perchellet, J P
Published in International journal of oncology (01.12.2001)
Published in International journal of oncology (01.12.2001)
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Quinone isomers of the WS-5995 antibiotics: synthetic antitumor agents that inhibit macromolecule synthesis, block nucleoside transport, induce DNA fragmentation, and decrease the growth and viability of L1210 leukemic cells more effectively than ellagic acid and genistein in vitro
Perchellet, E M, Sperfslage, B J, Qabaja, G, Jones, G B, Perchellet, J P
Published in Anti-cancer drugs (01.06.2001)
Published in Anti-cancer drugs (01.06.2001)
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Synthetic 1,4-anthracenediones, which block nucleoside transport and induce DNA fragmentation, retain their cytotoxic efficacy in daunorubicin-resistant HL-60 cell lines
Wu, M, Wang, B, Perchellet, E M, Sperfslage, B J, Stephany, H A, Hua, D H, Perchellet, J P
Published in Anti-cancer drugs (01.11.2001)
Published in Anti-cancer drugs (01.11.2001)
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Antileukemic activity of synthetic daunomycinone derivatives bearing modifications in the glycosidic moiety
Perchellet, E M, Sperfslage, B J, McIlvain, C J, Aligiannis, N, Pouli, N, Marakos, P, Skaltsounis, A L, Perchellet, J P
Published in Anticancer research (01.11.2001)
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Published in Anticancer research (01.11.2001)
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Among substituted 9,10-dihydro-9,10-[1,2]benzenoanthracene-1,4,5,8-tetraones, the lead antitumor triptycene bisquinone TT24 blocks nucleoside transport, induces apoptotic DNA fragmentation and decreases the viability of L1210 leukemic cells in the nanomolar range of daunorubicin in vitro
Perchellet, Elisabeth M, Sperfslage, Bonnie J, Wang, Yang, Huang, Xiaodong, Tamura, Masafumi, Hua, Duy H, Perchellet, Jean-Pierre
Published in Anti-cancer drugs (01.07.2002)
Published in Anti-cancer drugs (01.07.2002)
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Syntheses and Bioactivities of Substituted 9,10-Dihydro-9,10-[1,2]benzenoanthracene-1,4,5,8-tetrones. Unusual Reactivities with Amines
Hua, Duy H, Tamura, Masafumi, Huang, Xiaodong, Stephany, Heidi A, Helfrich, Brian A, Perchellet, Elisabeth M, Sperfslage, Bonnie J, Perchellet, Jean-Pierre, Jiang, Suping, Kyle, Dennis E, Chiang, Peter K
Published in Journal of organic chemistry (03.05.2002)
Published in Journal of organic chemistry (03.05.2002)
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Synthetic 1,4-anthracenedione analogs induce cytochrome c release, caspase-9, -3, and -8 activities, poly(ADP-ribose) polymerase-1 cleavage and internucleosomal DNA fragmentation in HL-60 cells by a mechanism which involves caspase-2 activation but not Fas signaling
Perchellet, Elisabeth M, Wang, Yang, Weber, Rebeka L, Sperfslage, Bonnie J, Lou, Kaiyan, Crossland, Justin, Hua, Duy H, Perchellet, Jean-Pierre
Published in Biochemical pharmacology (01.02.2004)
Published in Biochemical pharmacology (01.02.2004)
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Preparation and Cytotoxic Activity of Some New Rhodomycin Derivatives Bearing Modifications in the Sugar Moiety
ALIGIANNIS, NECTARIOS, POULI, NICOLE, MARAKOS, PANAGIOTIS, SKALTSOUNIS, ALEXIOS-LEANDROS, FLORENT, JEAN-CLAUDE, PERCHELLET, ELISABETH M., SPERFSLAGE, BONNIE J., McILVAIN, CORBIN J., PERCHELLET, JEAN-PIERRE
Published in Journal of antibiotics (2002)
Published in Journal of antibiotics (2002)
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