Meal Pattern Analysis of Diet-Induced Obesity in Susceptible and Resistant Rats
Farley, Constance, Cook, John A., Spar, Brian D., Austin, Theodore M., Kowalski, Timothy J.
Published in Obesity (Silver Spring, Md.) (01.07.2003)
Published in Obesity (Silver Spring, Md.) (01.07.2003)
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Discovery of Orally Efficacious Melanin-Concentrating Hormone Receptor-1 Antagonists as Antiobesity Agents. Synthesis, SAR, and Biological Evaluation of Bicyclo[3.1.0]hexyl Ureas
McBriar, Mark D, Guzik, Henry, Shapiro, Sherry, Paruchova, Jaroslava, Xu, Ruo, Palani, Anandan, Clader, John W, Cox, Kathleen, Greenlee, William J, Hawes, Brian E, Kowalski, Timothy J, O'Neill, Kim, Spar, Brian D, Weig, Blair, Weston, Daniel J, Farley, Constance, Cook, John
Published in Journal of medicinal chemistry (06.04.2006)
Published in Journal of medicinal chemistry (06.04.2006)
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Effects of a selective melanin-concentrating hormone 1 receptor antagonist on food intake and energy homeostasis in diet-induced obese mice
Kowalski, Timothy J., Spar, Brian D., Weig, Blair, Farley, Constance, Cook, John, Ghibaudi, Lorraine, Fried, Steve, O'Neill, Kim, Del Vecchio, Robert A., McBriar, Mark, Guzik, Henry, Clader, John, Hawes, Brian E., Hwa, Joyce
Published in European journal of pharmacology (27.03.2006)
Published in European journal of pharmacology (27.03.2006)
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Diaryl piperidines as CB1 receptor antagonists
SCOTT, Jack D, LI, Sarah W, STAMFORD, Andrew W, CHACKALAMANNIL, Samuel, LACHOWICZ, Jean E, GREENLEE, William J, HONGWU WANG, YAN XIA, JAYNE, Charles L, MILLER, Michael W, DUFFY, Ruth A, BOYKOW, George C, KOWALSKI, Timothy J, SPAR, Brian D
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Novel aminobenzimidazoles as selective MCH-R1 antagonists for the treatment of metabolic diseases
Sasikumar, T.K., Qiang, Li, Burnett, Duane A., Greenlee, William J., Hawes, Brian E., Kowalski, Timothy J., O’Neill, Kim, Spar, Brian D., Weig, Blair
Published in Bioorganic & medicinal chemistry letters (15.10.2006)
Published in Bioorganic & medicinal chemistry letters (15.10.2006)
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Bicyclic[4.1.0]heptanes as phenyl replacements for melanin concentrating hormone receptor antagonists
Xu, Ruo, Li, Shengjian, Paruchova, Jaroslava, McBriar, Mark D., Guzik, Henry, Palani, Anandan, Clader, John W., Cox, Kathleen, Greenlee, William J., Hawes, Brian E., Kowalski, Timothy J., O’Neill, Kim, Spar, Brian D., Weig, Blair, Weston, Daniel J.
Published in Bioorganic & medicinal chemistry (15.05.2006)
Published in Bioorganic & medicinal chemistry (15.05.2006)
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Discovery of Bicycloalkyl Urea Melanin Concentrating Hormone Receptor Antagonists: Orally Efficacious Antiobesity Therapeutics
McBriar, Mark D, Guzik, Henry, Xu, Ruo, Paruchova, Jaroslava, Li, Shengjian, Palani, Anandan, Clader, John W, Greenlee, William J, Hawes, Brian E, Kowalski, Timothy J, O'Neill, Kim, Spar, Brian, Weig, Blair
Published in Journal of medicinal chemistry (07.04.2005)
Published in Journal of medicinal chemistry (07.04.2005)
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Biaryl Ureas as Potent and Orally Efficacious Melanin Concentrating Hormone Receptor 1 Antagonists for the Treatment of Obesity
Palani, Anandan, Shapiro, Sherry, McBriar, Mark D, Clader, John W, Greenlee, William J, Spar, Brian, Kowalski, Timothy J, Farley, Constance, Cook, John, van Heek, Margaret, Weig, Blair, O'Neill, Kim, Graziano, Michael, Hawes, Brian
Published in Journal of medicinal chemistry (28.07.2005)
Published in Journal of medicinal chemistry (28.07.2005)
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Hypocalcemia and Inhibition of Parathyroid Hormone Secretion after Administration of WR-2721 (a Radioprotective and Chemoprotective Agent)
Glover, Donna, Riley, Louis, Carmichael, Kim, Spar, Brian, Glick, John, Kligerman, Morton M, Agus, Zalman S, Slatopolsky, Eduardo, Attie, Maurice, Goldfarb, Stanley
Published in The New England journal of medicine (10.11.1983)
Published in The New England journal of medicine (10.11.1983)
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Diaryl piperidines as CB sub(1) receptor antagonists
Scott, Jack D, Li, Sarah W, Wang, Hongwu, Xia, Yan, Jayne, Charles L, Miller, Michael W, Duffy, Ruth A, Boykow, George C, Kowalski, Timothy J, Spar, Brian D, Stamford, Andrew W, Chackalamannil, Samuel, Lachowicz, Jean E, Greenlee, William J
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Diaryl piperidines as CB 1 receptor antagonists
Scott, Jack D., Li, Sarah W., Wang, Hongwu, Xia, Yan, Jayne, Charles L., Miller, Michael W., Duffy, Ruth A., Boykow, George C., Kowalski, Timothy J., Spar, Brian D., Stamford, Andrew W., Chackalamannil, Samuel, Lachowicz, Jean E., Greenlee, William J.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Design and synthesis of orally efficacious benzimidazoles as melanin-concentrating hormone receptor 1 antagonists
Wu, Wen-Lian, Burnett, Duane A., Caplen, Mary Ann, Domalski, Martin S., Bennett, Chad, Greenlee, William J., Hawes, Brian E., O’Neill, Kim, Weig, Blair, Weston, Daniel, Spar, Brian, Kowalski, Timothy
Published in Bioorganic & medicinal chemistry letters (15.07.2006)
Published in Bioorganic & medicinal chemistry letters (15.07.2006)
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SAR study of bicyclo[4.1.0]heptanes as melanin-concentrating hormone receptor R1 antagonists: Taming hERG
Su, Jing, McKittrick, Brian A., Tang, Haiqun, Burnett, Duane A., Clader, John W., Greenlee, William J., Hawes, Brian E., O’Neill, Kim, Spar, Brian, Weig, Blair, Kowalski, Timothy, Sorota, Steve, Li, Cheng, Liu, Tongtong
Published in Bioorganic & medicinal chemistry (15.08.2007)
Published in Bioorganic & medicinal chemistry (15.08.2007)
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Synthesis of novel bicyclo[4.1.0]heptane and bicyclo[3.1.0]hexane derivatives as melanin-concentrating hormone receptor R1 antagonists
Su, Jing, Tang, Haiqun, McKittrick, Brian A., Gu, Huizhong, Guo, Tao, Qian, Gang, Burnett, Duane A., Clader, John W., Greenlee, William J., Hawes, Brian E., O’Neill, Kim, Spar, Brian, Weig, Blair, Kowalski, Timothy, Sorota, Steve
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Journal Article
Sar study of bicyclo [4.1.0]heptanes as melanin-concentrating hormone receptor R1 antagoniARs : Taming hERG
JING SU, MCKITTRICK, Brian A, KOWALSKI, Timothy, SOROTA, Steve, CHENG LI, TONGTONG LIU, HAIQUN TANG, BURNETT, Duane A, CLADER, John W, GREENLEE, William J, HAWES, Brian E, O'NEILL, Kim, SPAR, Brian, WEIG, Blair
Published in Bioorganic & medicinal chemistry (2007)
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Published in Bioorganic & medicinal chemistry (2007)
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