Composition and Conformation of Hetero‐ versus Homo‐Fluorinated Triazolamers Influence their Activity on Islet Amyloid Polypeptide Aggregation
Laxio Arenas, José, Lesma, Jacopo, Ha‐Duong, Tap, Ranjan Sahoo, Bikash, Ramamoorthy, Ayyalusamy, Tonali, Nicolo, Soulier, Jean‐Louis, Halgand, Frédéric, Giraud, François, Crousse, Benoît, Kaffy, Julia, Ongeri, Sandrine
Published in Chemistry : a European journal (17.05.2024)
Published in Chemistry : a European journal (17.05.2024)
Get full text
Journal Article
β-Hairpin Peptide Mimics Decrease Human Islet Amyloid Polypeptide (hIAPP) Aggregation
Lesma, Jacopo, Bizet, Faustine, Berardet, Corentin, Tonali, Nicolo, Pellegrino, Sara, Taverna, Myriam, Khemtemourian, Lucie, Soulier, Jean-Louis, van Heijenoort, Carine, Halgand, Frédéric, Ha-Duong, Tâp, Kaffy, Julia, Ongeri, Sandrine
Published in Frontiers in cell and developmental biology (16.09.2021)
Published in Frontiers in cell and developmental biology (16.09.2021)
Get full text
Journal Article
The use of 4,4,4-trifluorothreonine to stabilize extended peptide structures and mimic β-strands
Xu, Yaochun, Correia, Isabelle, Ha-Duong, Tap, Kihal, Nadjib, Soulier, Jean-Louis, Kaffy, Julia, Crousse, Benoît, Lequin, Olivier, Ongeri, Sandrine
Published in Beilstein journal of organic chemistry (21.12.2017)
Published in Beilstein journal of organic chemistry (21.12.2017)
Get full text
Journal Article
Toward the First Nonpeptidic Molecular Tong Inhibitor of Wild-Type and Mutated HIV-1 Protease Dimerization
Vidu, Anamaria, Dufau, Laure, Bannwarth, Ludovic, Soulier, Jean-Louis, Sicsic, Sames, Piarulli, Umberto, Reboud-Ravaux, Michèle, Ongeri, Sandrine
Published in ChemMedChem (08.11.2010)
Published in ChemMedChem (08.11.2010)
Get full text
Journal Article
Towards a general synthesis of di-aza-amino acids containing peptides
Bizet, Faustine, Tonali, Nicolo, Soulier, Jean-Louis, Oliva, Agostino, Kaffy, Julia, Crousse, Benoit, Ongeri, Sandrine
Published in New journal of chemistry (08.10.2018)
Published in New journal of chemistry (08.10.2018)
Get full text
Journal Article
Structure-activity relationships of β-hairpin mimics as modulators of amyloid β-peptide aggregation
Tonali, Nicolo, Kaffy, Julia, Soulier, Jean-Louis, Gelmi, Maria Luisa, Erba, Emanuela, Taverna, Myriam, van Heijenoort, Carine, Ha-Duong, Tap, Ongeri, Sandrine
Published in European journal of medicinal chemistry (25.06.2018)
Published in European journal of medicinal chemistry (25.06.2018)
Get full text
Journal Article
Designed Glycopeptidomimetics Disrupt Protein–Protein Interactions Mediating Amyloid β‑Peptide Aggregation and Restore Neuroblastoma Cell Viability
Kaffy, Julia, Brinet, Dimitri, Soulier, Jean-Louis, Correia, Isabelle, Tonali, Nicolo, Fera, Katia Fabiana, Iacone, Yasmine, Hoffmann, Anaïs R. F, Khemtémourian, Lucie, Crousse, Benoit, Taylor, Mark, Allsop, David, Taverna, Myriam, Lequin, Olivier, Ongeri, Sandrine
Published in Journal of medicinal chemistry (10.03.2016)
Published in Journal of medicinal chemistry (10.03.2016)
Get full text
Journal Article
Structure–activity relationships of sugar-based peptidomimetics as modulators of amyloid β-peptide early oligomerization and fibrillization
Kaffy, Julia, Brinet, Dimitri, Soulier, Jean-Louis, Khemtémourian, Lucie, Lequin, Olivier, Taverna, Myriam, Crousse, Benoît, Ongeri, Sandrine
Published in European journal of medicinal chemistry (30.10.2014)
Published in European journal of medicinal chemistry (30.10.2014)
Get full text
Journal Article
α- and β-hydrazino acid-based pseudopeptides inhibit the chymotrypsin-like activity of the eukaryotic 20S proteasome
Bordessa, Andrea, Keita, Massaba, Maréchal, Xavier, Formicola, Lucia, Lagarde, Nathalie, Rodrigo, Jordi, Bernadat, Guillaume, Bauvais, Cyril, Soulier, Jean-Louis, Dufau, Laure, Milcent, Thierry, Crousse, Benoit, Reboud-Ravaux, Michèle, Ongeri, Sandrine
Published in European journal of medicinal chemistry (01.12.2013)
Published in European journal of medicinal chemistry (01.12.2013)
Get full text
Journal Article
Synthesis of Specific Bivalent Probes That Functionally Interact with 5-HT4 Receptor Dimers
Russo, Olivier, Berthouze, Magali, Giner, Mireille, Soulier, Jean-Louis, Rivail, Lucie, Sicsic, Sames, Lezoualc'h, Frank, Jockers, Ralf, Berque-Bestel, Isabelle
Published in Journal of medicinal chemistry (06.09.2007)
Published in Journal of medicinal chemistry (06.09.2007)
Get full text
Journal Article
New Esters of 4-Amino-5-chloro-2-methoxybenzoic Acid as Potent Agonists and Antagonists for 5-HT4 Receptors
Yang, Donglai, Soulier, Jean-Louis, Sicsic, Sames, Mathé-Allainmat, Monique, Brémont, Béatrice, Croci, Tiziano, Cardamone, Rosanna, Aureggi, Giulio, Langlois, Michel
Published in Journal of medicinal chemistry (14.02.1997)
Published in Journal of medicinal chemistry (14.02.1997)
Get full text
Journal Article
Carbonylhydrazide-Based Molecular Tongs Inhibit Wild-Type and Mutated HIV‑1 Protease Dimerization
Dufau, Laure, Marques Ressurreição, Ana Sofia, Fanelli, Roberto, Kihal, Nadjib, Vidu, Anamaria, Milcent, Thierry, Soulier, Jean-Louis, Rodrigo, Jordi, Desvergne, Audrey, Leblanc, Karine, Bernadat, Guillaume, Crousse, Benoit, Reboud-Ravaux, Michèle, Ongeri, Sandrine
Published in Journal of medicinal chemistry (09.08.2012)
Published in Journal of medicinal chemistry (09.08.2012)
Get full text
Journal Article
Design and Synthesis of Specific Probes for Human 5-HT4 Receptor Dimerization Studies
Soulier, Jean-Louis, Russo, Olivier, Giner, Mireille, Rivail, Lucie, Berthouze, Magali, Ongeri, Sandrine, Maigret, Bernard, Fischmeister, Rodolphe, Lezoualc'h, Frank, Sicsic, Sames, Berque-Bestel, Isabelle
Published in Journal of medicinal chemistry (06.10.2005)
Published in Journal of medicinal chemistry (06.10.2005)
Get full text
Journal Article
New insights into the human 5‐HT4 receptor binding site: exploration of a hydrophobic pocket
Rivail, Lucie, Giner, Mireille, Gastineau, Monique, Berthouze, Magali, Soulier, Jean‐Louis, Fischmeister, Rodolphe, Lezoualc'h, Frank, Maigret, Bernard, Sicsic, Sames, Berque‐Bestel, Isabelle
Published in British journal of pharmacology (01.10.2004)
Published in British journal of pharmacology (01.10.2004)
Get full text
Journal Article
Structure-activity relationships of beta-hairpin mimics as modulators of amyloid beta-peptide aggregation
Tonali, Nicolo, Kaffy, Julia, Soulier, Jean-Louis, Gelmi, Maria Luisa, Erba, Emanuela, Taverna, Myriam, van Heijenoort, Carine, Ha-Duong, Tap, Ongeri, Sandrine
Published in European journal of medicinal chemistry (25.06.2018)
Published in European journal of medicinal chemistry (25.06.2018)
Get full text
Journal Article
Towards a general synthesis of di-aza-amino acids containing peptidesElectronic supplementary information (ESI) available. See DOI: 10.1039/c8nj03635g
Bizet, Faustine, Tonali, Nicolo, Soulier, Jean-Louis, Oliva, Agostino, Kaffy, Julia, Crousse, Benoit, Ongeri, Sandrine
Year of Publication 08.10.2018
Year of Publication 08.10.2018
Get full text
Journal Article
Relation between conformation and activity on islet amyloid polypeptide aggregation of fluorinated foldamers based on N-difluoromethyl-1,4-triazole amino acids
Laxio Arenas, José, Lesma, Jacopo, Ha-Duong, Tap, Sahoo, Bikash Ranjan, Ramamoorthy, Ayyalusamy, Tonali, Nicolo, Soulier, Jean-Louis, Halgand, Frederic, Giraud, François, Crousse, Benoit, Kaffy, Julia, Ongeri, Sandrine
Published in Chemistry : a European journal (13.03.2024)
Get full text
Published in Chemistry : a European journal (13.03.2024)
Journal Article
Structure-activity relationships of β-hairpin mimics as modulators of amyloid β-peptide aggregation
Tonali, Nicolo, Kaffy, Julia, Soulier, Jean-Louis, Gelmi, Maria Luisa, Erba, Emanuela, Taverna, Myriam, van Heijenoort, Carine, Ha-Duong, Tap, Ongeri, Sandrine
Published in European journal of medicinal chemistry (01.06.2018)
Published in European journal of medicinal chemistry (01.06.2018)
Get full text
Journal Article