From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effects
Pont, Caterina, Ginex, Tiziana, Griñán-Ferré, Christian, Scheiner, Matthias, Mattellone, Alexia, Martínez, Noemí, Arce, Elsa M., Soriano-Fernández, Yolanda, Naldi, Marina, De Simone, Angela, Barenys, Marta, Gómez-Catalán, Jesús, Pérez, Belén, Sabate, Raimon, Andrisano, Vincenza, Loza, María Isabel, Brea, José, Bartolini, Manuela, Bolognesi, Maria Laura, Decker, Michael, Pallàs, Mercè, Luque, F. Javier, Muñoz-Torrero, Diego
Published in European journal of medicinal chemistry (05.12.2021)
Published in European journal of medicinal chemistry (05.12.2021)
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