Identification of Novel Fragments Binding to the PDZ1‐2 Domain of PSD‐95
Zang, Jie, Ye, Fei, Solbak, Sara M. Ø., Høj, Lars J., Zhang, Mingjie, Bach, Anders
Published in ChemMedChem (18.03.2021)
Published in ChemMedChem (18.03.2021)
Get full text
Journal Article
The dynamics of linear polyubiquitin
Jussupow, Alexander, Messias, Ana C, Stehle, Ralf, Geerlof, Arie, Solbak, Sara M Ø, Paissoni, Cristina, Bach, Anders, Sattler, Michael, Camilloni, Carlo
Published in Science advances (01.10.2020)
Published in Science advances (01.10.2020)
Get full text
Journal Article
Co-adjuvanting DDA/TDB liposomes with a TLR7 agonist allows for IgG2a/c class-switching in the absence of Th1 cells
Zimmermann, Julie, van Haren, Simon D., Diray-Arce, Joann, Adriawan, Ignatius Ryan, Wørzner, Katharina, Krog, Ricki T., Guleed, Safia, Hu, Tu, Mortensen, Rasmus, Dietrich, Jes, Solbak, Sara M. Ø., Levy, Ofer, Christensen, Dennis, Pedersen, Gabriel K.
Published in npj vaccines (22.12.2023)
Published in npj vaccines (22.12.2023)
Get full text
Journal Article
Author Correction: Co-adjuvanting DDA/TDB liposomes with a TLR7 agonist allows for IgG2a/c class-switching in the absence of Th1 cells
Zimmermann, Julie, van Haren, Simon D., Diray-Arce, Joann, Adriawan, Ignatius Ryan, Wørzner, Katharina, Krog, Ricki T., Guleed, Safia, Hu, Tu, Mortensen, Rasmus, Dietrich, Jes, Solbak, Sara M. Ø., Levy, Ofer, Christensen, Dennis, Pedersen, Gabriel K.
Published in npj vaccines (11.01.2024)
Published in npj vaccines (11.01.2024)
Get full text
Journal Article
Highly conserved serine residue 40 in HIV-1 p6 regulates capsid processing and virus core assembly
Votteler, Jörg, Neumann, Liane, Hahn, Sabine, Hahn, Friedrich, Rauch, Pia, Schmidt, Kerstin, Studtrucker, Nicole, Solbak, Sara M Ø, Fossen, Torgils, Henklein, Peter, Ott, David E, Holland, Gudrun, Bannert, Norbert, Schubert, Ulrich
Published in Retrovirology (16.02.2011)
Published in Retrovirology (16.02.2011)
Get full text
Journal Article
A Comparative Assessment Study of Known Small-Molecule Keap1−Nrf2 Protein–Protein Interaction Inhibitors: Chemical Synthesis, Binding Properties, and Cellular Activity
Tran, Kim T, Pallesen, Jakob S, Solbak, Sara M. Ø, Narayanan, Dilip, Baig, Amina, Zang, Jie, Aguayo-Orozco, Alejandro, Carmona, Rosa M. C, Garcia, Anthony D, Bach, Anders
Published in Journal of medicinal chemistry (12.09.2019)
Published in Journal of medicinal chemistry (12.09.2019)
Get full text
Journal Article
Deconstructing Noncovalent Kelch-like ECH-Associated Protein 1 (Keap1) Inhibitors into Fragments to Reconstruct New Potent Compounds
Pallesen, Jakob S, Narayanan, Dilip, Tran, Kim T, Solbak, Sara M. Ø, Marseglia, Giuseppe, Sørensen, Louis M. E, Høj, Lars J, Munafò, Federico, Carmona, Rosa M. C, Garcia, Anthony D, Desu, Haritha L, Brambilla, Roberta, Johansen, Tommy N, Popowicz, Grzegorz M, Sattler, Michael, Gajhede, Michael, Bach, Anders
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
Get full text
Journal Article
Ligand‐induced CaMKIIα hub Trp403 flip, hub domain stacking, and modulation of kinase activity
Narayanan, Dilip, Larsen, Anne Sofie G., Gauger, Stine Juul, Adafia, Ruth, Hammershøi, Rikke Bartschick, Hamborg, Louise, Bruus‐Jensen, Jesper, Griem‐Krey, Nane, Gee, Christine L., Frølund, Bente, Stratton, Margaret M., Kuriyan, John, Kastrup, Jette Sandholm, Langkilde, Annette E., Wellendorph, Petrine, Solbak, Sara M. Ø.
Published in Protein science (01.10.2024)
Published in Protein science (01.10.2024)
Get full text
Journal Article
Nuclear import of isoforms of the cytomegalovirus kinase pUL97 is mediated by differential activity of NLS1 and NLS2 both acting through classical importin-α binding
WEBEL, Rike, SOLBAK, Sara M.Ø, MARSCHALL, Manfred, HELD, Christian, MILBRADT, Jens, GROSS, Andrea, EICHLER, Jutta, WITTENBERG, Thomas, JARDIN, Christophe, STICHT, Heinrich, FOSSEN, Torgils
Published in Journal of general virology (01.08.2012)
Published in Journal of general virology (01.08.2012)
Get full text
Journal Article
Exploring the NCS-382 Scaffold for CaMKIIα Modulation: Synthesis, Biochemical Pharmacology, and Biophysical Characterization of Ph-HTBA as a Novel High-Affinity Brain-Penetrant Stabilizer of the CaMKIIα Hub Domain
Tian, Yongsong, Shehata, Mohamed A., Gauger, Stine Juul, Veronesi, Carolina, Hamborg, Louise, Thiesen, Louise, Bruus-Jensen, Jesper, Royssen, Johanne Schlieper, Leurs, Ulrike, Larsen, Anne Sofie G., Krall, Jacob, Solbak, Sara M.Ø., Wellendorph, Petrine, Frølund, Bente
Published in Journal of medicinal chemistry (24.11.2022)
Published in Journal of medicinal chemistry (24.11.2022)
Get full text
Journal Article
Development of Noncovalent Small-Molecule Keap1-Nrf2 Inhibitors by Fragment-Based Drug Discovery
Narayanan, Dilip, Tran, Kim T., Pallesen, Jakob S., Solbak, Sara M. Ø., Qin, Yuting, Mukminova, Elina, Luchini, Martina, Vasilyeva, Kristina O., González Chichón, Dorleta, Goutsiou, Georgia, Poulsen, Cecilie, Haapanen, Nanna, Popowicz, Grzegorz M., Sattler, Michael, Olagnier, David, Gajhede, Michael, Bach, Anders
Published in Journal of medicinal chemistry (10.11.2022)
Published in Journal of medicinal chemistry (10.11.2022)
Get full text
Journal Article
The host-pathogen interaction of human cyclophilin A and HIV-1 Vpr requires specific N-terminal and novel C-terminal domains
Solbak, Sara M Ø, Wray, Victor, Horvli, Ole, Raae, Arnt J, Flydal, Marte I, Henklein, Petra, Henklein, Peter, Nimtz, Manfred, Schubert, Ulrich, Fossen, Torgils
Published in BMC structural biology (20.12.2011)
Published in BMC structural biology (20.12.2011)
Get full text
Journal Article
GHB analogs confer neuroprotection through specific interaction with the CaMKIIα hub domain
Leurs, Ulrike, Klein, Anders B., McSpadden, Ethan D., Griem-Krey, Nane, Solbak, Sara M. Ø., Houlton, Josh, Villumsen, Inge S., Vogensen, Stine B., Hamborg, Louise, Gauger, Stine J., Palmelund, Line B., Larsen, Anne Sofie G., Shehata, Mohamed A., Kelstrup, Christian D., Olsen, Jesper V., Bach, Anders, Burnie, Robert O., Kerr, D. Steven, Gowing, Emma K., Teurlings, Selina M. W., Chi, Chris C., Gee, Christine L., Frølund, Bente, Kornum, Birgitte R., van Woerden, Geeske M., Clausen, Rasmus P., Kuriyan, John, Clarkson, Andrew N., Wellendorph, Petrine
Published in Proceedings of the National Academy of Sciences - PNAS (03.08.2021)
Published in Proceedings of the National Academy of Sciences - PNAS (03.08.2021)
Get full text
Journal Article
Influenza A virus protein PB1-F2 from different strains shows distinct structural signatures
Solbak, Sara M.Ø., Sharma, Alok, Bruns, Karsten, Röder, René, Mitzner, David, Hahn, Friedrich, Niebert, Rebekka, Vedeler, Anni, Henklein, Petra, Henklein, Peter, Schubert, Ulrich, Wray, Victor, Fossen, Torgils
Published in Biochimica et biophysica acta (01.02.2013)
Published in Biochimica et biophysica acta (01.02.2013)
Get full text
Journal Article
HIV-1 p6—Another viral interaction partner to the host cellular protein cyclophilin A
Solbak, Sara M.Ø., Reksten, Tove R., Röder, Rene, Wray, Victor, Horvli, Ole, Raae, Arnt J., Henklein, Petra, Henklein, Peter, Fossen, Torgils
Published in Biochimica et biophysica acta (01.04.2012)
Published in Biochimica et biophysica acta (01.04.2012)
Get full text
Journal Article
GHB confers neuroprotection by stabilizing the CaMKIIα hub domain
Leurs, Ulrike, Klein, Anders B, Mcspadden, Ethan D, Griem-Krey, Nane, Sara M Ø Solbak, Houlton, Josh, Villumsen, Inge S, Vogensen, Stine B, Hamborg, Louise, Gauger, Stine J, Palmelund, Line B, Larsen, Anne Sofie G, Shehata, Mohamed A, Kelstrup, Christian D, Olsen, Jesper V, Bach, Anders, Burnie, Robert O, Kerr, D Steven, Gowing, Emma K, Teurlings, Selina M W, Chi, Chris C, Gee, Christine L, Frølund, Bente, Kornum, Birgitte R, Van Woerden, Geeske M, Clausen, Rasmus P, Kuriyan, John, Clarkson, Andrew N, Wellendorph, Petrine
Published in bioRxiv (28.09.2020)
Published in bioRxiv (28.09.2020)
Get full text
Paper