Bridging the translational innovation gap through good biomarker practice
van Gool, Alain J, Bietrix, Florence, Caldenhoven, Eric, Zatloukal, Kurt, Scherer, Andreas, Litton, Jan-Eric, Meijer, Gerrit, Blomberg, Niklas, Smith, Andy, Mons, Barend, Heringa, Jaap, Koot, Wim-Jan, Smit, Martin J, Hajduch, Marian, Rijnders, Ton, Ussi, Anton
Published in Nature reviews. Drug discovery (01.09.2017)
Published in Nature reviews. Drug discovery (01.09.2017)
Get full text
Journal Article
Org 214007-0: a novel non-steroidal selective glucocorticoid receptor modulator with full anti-inflammatory properties and improved therapeutic index
van Lierop, Marie-José C, Alkema, Wynand, Laskewitz, Anke J, Dijkema, Rein, van der Maaden, Hans M, Smit, Martin J, Plate, Ralf, Conti, Paolo G M, Jans, Christan G J M, Timmers, C Marco, van Boeckel, Constant A A, Lusher, Scott J, McGuire, Ross, van Schaik, Rene C, de Vlieg, Jacob, Smeets, Ruben L, Hofstra, Claudia L, Boots, Annemieke M H, van Duin, Marcel, Ingelse, Benno A, Schoonen, Willem G E J, Grefhorst, Aldo, van Dijk, Theo H, Kuipers, Folkert, Dokter, Wim H A
Published in PloS one (12.11.2012)
Published in PloS one (12.11.2012)
Get full text
Journal Article
Increased Hepatobiliary and Fecal Cholesterol Excretion upon Activation of the Liver X Receptor Is Independent of ABCA1
Plo¨sch, Torsten, Kok, Tineke, Bloks, Vincent W., Smit, Martin J., Havinga, Rick, Chimini, Giovanna, Groen, Albert K., Kuipers, Folkert
Published in The Journal of biological chemistry (13.09.2002)
Published in The Journal of biological chemistry (13.09.2002)
Get full text
Journal Article
Nonpeptidergic Allosteric Antagonists Differentially Bind to the CXCR2 Chemokine Receptor
de Kruijf, Petra, van Heteren, Jane, Lim, Herman D, Conti, Paolo G M, van der Lee, Miranda M C, Bosch, Leontien, Ho, Koc-Kan, Auld, Douglas, Ohlmeyer, Michael, Smit, Martin J, Wijkmans, Jac C H M, Zaman, Guido J R, Smit, Martine J, Leurs, Rob
Published in The Journal of pharmacology and experimental therapeutics (01.05.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2009)
Get full text
Journal Article
Liver receptor homolog‐1 is critical for adequate up‐regulation of Cyp7a1 gene transcription and bile salt synthesis during bile salt sequestration
Out, Carolien, Hageman, Jurre, Bloks, Vincent W., Gerrits, Han, Sollewijn Gelpke, Maarten D., Bos, Trijnie, Havinga, Rick, Smit, Martin J., Kuipers, Folkert, Groen, Albert K.
Published in Hepatology (Baltimore, Md.) (01.06.2011)
Published in Hepatology (Baltimore, Md.) (01.06.2011)
Get full text
Journal Article
Unique Overlap in the Prerequisites for Thrombin Inhibition and Oral Bioavailability Resulting in Potent Oral Antithrombotics
Adang, Anton E. P, de Man, Adrianus P. A, Vogel, Gerard M. T, Grootenhuis, Peter D. J, Smit, Martin J, Peters, Co A. M, Visser, Arie, Rewinkel, Jos B. M, van Dinther, Theo, Lucas, Hans, Kelder, Jan, van Aelst, Sjoerd, Meuleman, Dick G, van Boeckel, Constant A. A
Published in Journal of medicinal chemistry (26.09.2002)
Published in Journal of medicinal chemistry (26.09.2002)
Get full text
Journal Article
Tibolone Prevents Atherosclerotic Lesion Formation in Cholesterol-Fed, Ovariectomized Rabbits
Zandberg, Pieter, Peters, Jan L.M, Demacker, Pierre N.M, Smit, Martin J, de Reeder, Ernst G, Meuleman, Dirk G
Published in Arteriosclerosis, thrombosis, and vascular biology (01.12.1998)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.12.1998)
Get full text
Journal Article
Elimination of macrophages drives LXR-induced regression both in initial and advanced stages of atherosclerotic lesion development
van der Stoep, Marco, Li, Zhaosha, Calpe-Berdiel, Laura, van der Sluis, Ronald J., Saleh, Peshtiwan, McKinnon, Heather J., Smit, Martin J., Korporaal, Suzanne J.A., Van Berkel, Theo J.C., Van Eck, Miranda, Hoekstra, Menno
Published in Biochemical pharmacology (01.12.2013)
Published in Biochemical pharmacology (01.12.2013)
Get full text
Journal Article
A signaling-selective, nanomolar potent allosteric low molecular weight agonist for the human luteinizing hormone receptor
van Koppen, Chris J., Zaman, Guido J. R., Timmers, C. Marco, Kelder, Jan, Mosselman, Sietse, van de Lagemaat, Ruud, Smit, Martin J., Hanssen, Rob G. J. M.
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.2008)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.2008)
Get full text
Journal Article
Uniform procedure of (1)H NMR analysis of rat urine and toxicometabonomics Part II: comparison of NMR profiles for classification of hepatotoxicity
Schoonen, Willem G E J, Kloks, Cathelijne P A M, Ploemen, Jan-Peter H T M, Smit, Martin J, Zandberg, Pieter, Horbach, G Jean, Mellema, Jan-Remt, Thijssen-Vanzuylen, Carol, Tas, Albert C, van Nesselrooij, Joop H J, Vogels, Jack T W E
Published in Toxicological sciences (01.07.2007)
Get full text
Published in Toxicological sciences (01.07.2007)
Journal Article
Differences in propionate-induced inhibition of cholesterol and triacylglycerol synthesis between human and rat hepatocytes in primary culture
Lin, Yuguang, Vonk, Roel J., Slooff, Maarten J. H., Kuipers, Folkert, Smit, Martin J.
Published in British journal of nutrition (01.08.1995)
Published in British journal of nutrition (01.08.1995)
Get full text
Journal Article
Uniform Procedure of super(1)H NMR Analysis of Rat Urine and Toxicometabonomics Part II: Comparison of NMR Profiles for Classification of Hepatotoxicity
Schoonen, Willem GEJ, Kloks, Cathelijne PAM, Ploemen, Jan-Peter HTM, Smit, Martin J, Zandberg, Pieter, Horbach, GJean, Mellema, Jan-Remt, Thijssen-vanZuylen, Carol, Tas, Albert C, van Nesselrooij, Joop HJ, Vogels, Jack TWE
Published in Toxicological sciences (01.07.2007)
Get full text
Published in Toxicological sciences (01.07.2007)
Journal Article
Sensitivity of super(1)H NMR Analysis of Rat Urine in Relation to Toxicometabonomics. Part I: Dose-Dependent Toxic Effects of Bromobenzene and Paracetamol
Schoonen, Willem GEJ, Kloks, Cathelijne PAM, Ploemen, Jan-Peter HTM, Horbach, GJean, Smit, Martin J, Zandberg, Pieter, Mellema, Jan-Remt, Zuylen, Carol Thijssen-van, Tas, Albert C, van Nesselrooij, Joop HJ, Vogels, Jack TWE
Published in Toxicological sciences (01.07.2007)
Get full text
Published in Toxicological sciences (01.07.2007)
Journal Article
Sensitivity of (1)H NMR analysis of rat urine in relation to toxicometabonomics. Part I: dose-dependent toxic effects of bromobenzene and paracetamol
Schoonen, Willem G E J, Kloks, Cathelijne P A M, Ploemen, Jan-Peter H T M, Horbach, G Jean, Smit, Martin J, Zandberg, Pieter, Mellema, Jan-Remt, Zuylen, Carol Thijssen-van, Tas, Albert C, van Nesselrooij, Joop H J, Vogels, Jack T W E
Published in Toxicological sciences (01.07.2007)
Get full text
Published in Toxicological sciences (01.07.2007)
Journal Article
Uniform Procedure of 1H NMR Analysis of Rat Urine and Toxicometabonomics Part II: Comparison of NMR Profiles for Classification of Hepatotoxicity
Schoonen, Willem G. E. J., Kloks, Cathelijne P. A. M., Ploemen, Jan-Peter H. T. M., Smit, Martin J., Zandberg, Pieter, Horbach, G. Jean, Mellema, Jan-Remt, Thijssen-vanZuylen, Carol, Tas, Albert C., van Nesselrooij, Joop H. J., Vogels, Jack T. W. E.
Published in Toxicological sciences (01.07.2007)
Published in Toxicological sciences (01.07.2007)
Get full text
Journal Article
Sensitivity of 1H NMR Analysis of Rat Urine in Relation to Toxicometabonomics. Part I: Dose-Dependent Toxic Effects of Bromobenzene and Paracetamol
Schoonen, Willem G. E. J., Kloks, Cathelijne P. A. M., Ploemen, Jan-Peter H. T. M., Horbach, G. Jean, Smit, Martin J., Zandberg, Pieter, Mellema, Jan-Remt, Zuylen, Carol Thijssen-van, Tas, Albert C., van Nesselrooij, Joop H. J., Vogels, Jack T. W. E.
Published in Toxicological sciences (01.07.2007)
Published in Toxicological sciences (01.07.2007)
Get full text
Journal Article
Comparison of the antiatherosclerotic effect of tibolone with that of estradiol and ethinyl estradiol in cholesterol-fed, ovariectomized rabbits
Zandberg, P, Peters JLM, Demacker, P N, de Reeder, E G, Smit, M J, Meuleman, D G
Published in Menopause (New York, N.Y.) (01.03.2001)
Published in Menopause (New York, N.Y.) (01.03.2001)
Get more information
Journal Article