Leishmania donovani 90 kD Heat Shock Protein - Impact of Phosphosites on Parasite Fitness, Infectivity and Casein Kinase Affinity
Hombach-Barrigah, Antje, Bartsch, Katharina, Smirlis, Despina, Rosenqvist, Heidi, MacDonald, Andrea, Dingli, Florent, Loew, Damarys, Späth, Gerald F, Rachidi, Najma, Wiese, Martin, Clos, Joachim
Published in Scientific reports (25.03.2019)
Published in Scientific reports (25.03.2019)
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Journal Article
2-(4-Nitrophenyl)isothiazol-3(2H)-one: A Promising Selective Agent against Hepatocellular Carcinoma Cells
Marka, Sofia, Zografaki, Maria-Eleftheria, Tsolomiti, Georgia, Kalliampakou, Katerina I., Tsolomitis, Athanasios, Koumantou, Christina, Smirlis, Despina, Vassilaki, Niki, Kintzios, Spyros
Published in Pharmaceuticals (Basel, Switzerland) (24.05.2024)
Published in Pharmaceuticals (Basel, Switzerland) (24.05.2024)
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Journal Article
Targeting essential pathways in trypanosomatids gives insights into protozoan mechanisms of cell death
Smirlis, Despina, Duszenko, Michael, Ruiz, Antonio Jiménez, Scoulica, Effie, Bastien, Patrick, Fasel, Nicolas, Soteriadou, Ketty
Published in Parasites & vectors (17.11.2010)
Published in Parasites & vectors (17.11.2010)
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Journal Article
Towards discovery of new leishmanicidal scaffolds able to inhibit Leishmania GSK-3
Martínez de Iturrate, Paula, Sebastián-Pérez, Victor, Nácher-Vázquez, Montserrat, Tremper, Catherine S., Smirlis, Despina, Martín, Julio, Martínez, Ana, Campillo, Nuria E., Rivas, Luis, Gil, Carmen
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Journal Article
Identification of the Host Substratome of Leishmania -Secreted Casein Kinase 1 Using a SILAC-Based Quantitative Mass Spectrometry Assay
Smirlis, Despina, Dingli, Florent, Sabatet, Valentin, Roth, Aileen, Knippschild, Uwe, Loew, Damarys, Späth, Gerald F, Rachidi, Najma
Published in Frontiers in cell and developmental biology (03.01.2022)
Published in Frontiers in cell and developmental biology (03.01.2022)
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Journal Article
inhibitor-driven study for enhancing the selectivity of indirubin derivatives towards leishmanial Glycogen Synthase Kinase-3 over leishmanial cdc2-related protein kinase 3
Efstathiou, Antonia, Gaboriaud-Kolar, Nicolas, Smirlis, Despina, Myrianthopoulos, Vassilios, Vougogiannopoulou, Konstantina, Alexandratos, Alexandros, Kritsanida, Marina, Mikros, Emmanuel, Soteriadou, Ketty, Skaltsounis, Alexios-Leandros
Published in Parasites & vectors (20.05.2014)
Published in Parasites & vectors (20.05.2014)
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Journal Article
Indirubin derivatives are potent and selective anti-Trypanosoma cruzi agents
Efstathiou, Antonia, Meira, Cássio Santana, Gaboriaud-Kolar, Nicolas, Bastos, Tanira Matutino, Rocha, Vinícius Pinto Costa, Vougogiannopoulou, Konstantina, Skaltsounis, Alexios-Leandros, Smirlis, Despina, Soares, Milena Botelho Pereira
Published in Virulence (01.01.2018)
Published in Virulence (01.01.2018)
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Journal Article
Three new trixane glycosides obtained from the leaves of Jungia sellowii Less. using centrifugal partition chromatography
Azevedo, Luíse, Faqueti, Larissa, Kritsanida, Marina, Efstathiou, Antonia, Smirlis, Despina, Franchi, Jr, Gilberto C, Genta-Jouve, Grégory, Michel, Sylvie, Sandjo, Louis P, Grougnet, Raphaël, Biavatti, Maique Weber
Published in Beilstein journal of organic chemistry (12.04.2016)
Published in Beilstein journal of organic chemistry (12.04.2016)
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Journal Article
ER targeting and retention of the HCV NS4B protein relies on the concerted action of multiple structural features including its transmembrane domains
Boleti, Haralabia, Smirlis, Despina, Dalagiorgou, Georgia, Meurs, Eliane F., Christoforidis, Savvas, Mavromara, Penelope
Published in Molecular membrane biology (01.01.2010)
Published in Molecular membrane biology (01.01.2010)
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Journal Article
Orphan Receptor Promiscuity in the Induction of Cytochromes P450 by Xenobiotics
Smirlis, D, Muangmoonchai, R, Edwards, M, Phillips, I R, Shephard, E A
Published in The Journal of biological chemistry (20.04.2001)
Published in The Journal of biological chemistry (20.04.2001)
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Journal Article
Xenobiotic induction of cytochrome P450 2B1 (CYP2B1) is mediated by the orphan nuclear receptor constitutive androstane receptor (CAR) and requires steroid co-activator 1 (SRC-1) and the transcription factor Sp1
Muangmoonchai, R, Smirlis, D, Wong, S C, Edwards, M, Phillips, I R, Shephard, E A
Published in Biochemical journal (01.04.2001)
Published in Biochemical journal (01.04.2001)
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Journal Article
Induction of protective cellular immune responses against experimental visceral leishmaniasis mediated by dendritic cells pulsed with the N-terminal domain of Leishmania infantum elongation factor-2 and CpG oligodeoxynucleotides
Agallou, Maria, Pantazi, Eleni, Tsiftsaki, Elisavet, Toubanaki, Dimitra K., Gaitanaki, Catherine, Smirlis, Despina, Karagouni, Evdokia
Published in Molecular immunology (01.11.2018)
Published in Molecular immunology (01.11.2018)
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Journal Article
Vaccination with Leishmania histone H1-pulsed dendritic cells confers protection in murine visceral leishmaniasis
Agallou, Maria, Smirlis, Despina, Soteriadou, Ketty P, Karagouni, Evdokia
Published in Vaccine (20.07.2012)
Published in Vaccine (20.07.2012)
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Journal Article
Indirubin Analogues Inhibit Trypanosoma brucei Glycogen Synthase Kinase 3 Short and T. brucei Growth
Efstathiou, Antonia, Gaboriaud-Kolar, Nicolas, Myrianthopoulos, Vassilios, Vougogiannopoulou, Konstantina, Subota, Ines, Aicher, Stephanie, Mikros, Emmanuel, Bastin, Philippe, Skaltsounis, Alexios-Leandros, Soteriadou, Ketty, Smirlis, Despina
Published in Antimicrobial agents and chemotherapy (01.06.2019)
Published in Antimicrobial agents and chemotherapy (01.06.2019)
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Journal Article
Leishmania Genome Dynamics during Environmental Adaptation Reveal Strain-Specific Differences in Gene Copy Number Variation, Karyotype Instability, and Telomeric Amplification
Bussotti, Giovanni, Gouzelou, Evi, Côrtes Boité, Mariana, Kherachi, Ihcen, Harrat, Zoubir, Eddaikra, Naouel, Mottram, Jeremy C, Antoniou, Maria, Christodoulou, Vasiliki, Bali, Aymen, Guerfali, Fatma Z, Laouini, Dhafer, Mukhtar, Maowia, Dumetz, Franck, Dujardin, Jean-Claude, Smirlis, Despina, Lechat, Pierre, Pescher, Pascale, El Hamouchi, Adil, Lemrani, Meryem, Chicharro, Carmen, Llanes-Acevedo, Ivonne Pamela, Botana, Laura, Cruz, Israel, Moreno, Javier, Jeddi, Fakhri, Aoun, Karim, Bouratbine, Aïda, Cupolillo, Elisa, Späth, Gerald F
Published in mBio (06.11.2018)
Published in mBio (06.11.2018)
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Journal Article
SILAC-based quantitative proteomics reveals pleiotropic, phenotypic modulation in primary murine macrophages infected with the protozoan pathogen Leishmania donovani
Smirlis, Despina, Dingli, Florent, Pescher, Pascale, Prina, Eric, Loew, Damarys, Rachidi, Najma, Späth, Gerald F.
Published in Journal of proteomics (20.02.2020)
Published in Journal of proteomics (20.02.2020)
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Journal Article