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International Union of Basic and Clinical Pharmacology. CVIII. Calcium-Sensing Receptor Nomenclature, Pharmacology, and Function
Leach, Katie, Hannan, Fadil M., Josephs, Tracy M., Keller, Andrew N., Møller, Thor C., Ward, Donald T., Kallay, Enikö, Mason, Rebecca S., Thakker, Rajesh V., Riccardi, Daniela, Conigrave, Arthur D., Bräuner-Osborne, Hans
Published in Pharmacological reviews (01.07.2020)
Published in Pharmacological reviews (01.07.2020)
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Trending topics of SIRT1 in tumorigenicity
Garcia-Peterson, Liz M., Li, Xiaoling
Published in Biochimica et biophysica acta. General subjects (01.09.2021)
Published in Biochimica et biophysica acta. General subjects (01.09.2021)
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Novel Inhibitors of Cholesterol Degradation in Mycobacterium tuberculosis Reveal How the Bacterium’s Metabolism Is Constrained by the Intracellular Environment
VanderVen, Brian C., Fahey, Ruth J., Lee, Wonsik, Liu, Yancheng, Abramovitch, Robert B., Memmott, Christine, Crowe, Adam M., Eltis, Lindsay D., Perola, Emanuele, Deininger, David D., Wang, Tiansheng, Locher, Christopher P., Russell, David G.
Published in PLoS pathogens (01.02.2015)
Published in PLoS pathogens (01.02.2015)
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Identification of small molecule antagonists of sonic hedgehog/heparin binding with activity in hedgehog functional assays
Lamson, David R., Tarpley, Michael, Addo, Kezia, Ji, Xiaojia, Abu Rabe, Dina, Ehe, Ben, Hughes, Mark, Smith, Ginger R., Daye, Laura R., Musso, David L., Zheng, Weifan, Williams, Kevin P.
Published in Biochimica et biophysica acta. General subjects (01.11.2024)
Published in Biochimica et biophysica acta. General subjects (01.11.2024)
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Establishment of a suite of assays that support the discovery of proteasome stimulators
Trader, Darci J., Simanski, Scott, Dickson, Paige, Kodadek, Thomas
Published in Biochimica et biophysica acta (01.04.2017)
Published in Biochimica et biophysica acta (01.04.2017)
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A novel role for small molecule glycomimetics in the protection against lipid-induced endothelial dysfunction: Involvement of Akt/eNOS and Nrf2/ARE signaling
Mahmoud, Ayman M., Wilkinson, Fiona L., Jones, Alan M., Wilkinson, James A., Romero, Miguel, Duarte, Juan, Alexander, M. Yvonne
Published in Biochimica et biophysica acta. General subjects (01.01.2017)
Published in Biochimica et biophysica acta. General subjects (01.01.2017)
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PAI-1 augments mucosal damage in colitis
Kaiko, Gerard E, Chen, Feidi, Lai, Chin-Wen, Chiang, I-Ling, Perrigoue, Jacqueline, Stojmirović, Aleksandar, Li, Katherine, Muegge, Brian D, Jain, Umang, VanDussen, Kelli L, Goggins, Bridie J, Keely, Simon, Weaver, Jessica, Foster, Paul S, Lawrence, Daniel A, Liu, Ta-Chiang, Stappenbeck, Thaddeus S
Published in Science translational medicine (06.03.2019)
Published in Science translational medicine (06.03.2019)
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Characterization of novel small-molecule NRF2 activators: Structural and biochemical validation of stereospecific KEAP1 binding
Huerta, Carlos, Jiang, Xin, Trevino, Isaac, Bender, Christopher F., Ferguson, Deborah A., Probst, Brandon, Swinger, Kerren K., Stoll, Vincent S., Thomas, Philip J., Dulubova, Irina, Visnick, Melean, Wigley, W. Christian
Published in Biochimica et biophysica acta (01.11.2016)
Published in Biochimica et biophysica acta (01.11.2016)
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Targeted genetic and small molecule disruption of N-Ras CaaX cleavage alters its localization and oncogenic potential
Hildebrandt, Emily R., Hussain, Shaneela A., Sieburg, Michelle A., Ravishankar, Rajani, Asad, Nadeem, Gore, Sangram, Ito, Takahiro, Hougland, James L., Dore, Timothy M., Schmidt, Walter K.
Published in Bioorganic chemistry (01.06.2024)
Published in Bioorganic chemistry (01.06.2024)
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Development of small molecules targeting the pseudokinase Her3
Lim, Sang Min, Xie, Ting, Westover, Kenneth D., Ficarro, Scott B., Tae, Hyun Seop, Gurbani, Deepak, Sim, Taebo, Marto, Jarrod A., Jänne, Pasi A., Crews, Craig M., Gray, Nathanael S.
Published in Bioorganic & medicinal chemistry letters (15.08.2015)
Published in Bioorganic & medicinal chemistry letters (15.08.2015)
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Synergy-Based Small-Molecule Screen Using a Human Lung Epithelial Cell Line Yields ΔF508-CFTR Correctors That Augment VX-809 Maximal Efficacy
Phuan, Puay-Wah, Veit, Guido, Tan, Joseph, Roldan, Ariel, Finkbeiner, Walter E., L. Lukacs, Gergely, Verkman, A.S.
Published in Molecular pharmacology (01.07.2014)
Published in Molecular pharmacology (01.07.2014)
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Negative feedback via RSK modulates Erk‐dependent progression from naïve pluripotency
Nett, Isabelle RE, Mulas, Carla, Gatto, Laurent, Lilley, Kathryn S, Smith, Austin
Published in EMBO reports (01.08.2018)
Published in EMBO reports (01.08.2018)
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Recent Synthetic Approaches towards Small Molecule Reactivators of p53
Silva, Jerson L., Lima, Carolina G. S., Rangel, Luciana P., Ferretti, Giulia D. S., Pauli, Fernanda P., Ribeiro, Ruan C. B., da Silva, Thais de B., da Silva, Fernando C., Ferreira, Vitor F.
Published in Biomolecules (Basel, Switzerland) (20.04.2020)
Published in Biomolecules (Basel, Switzerland) (20.04.2020)
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Chemical activation of a food deprivation signal extends lifespan
Lucanic, Mark, Garrett, Theo, Yu, Ivan, Calahorro, Fernando, Asadi Shahmirzadi, Azar, Miller, Aaron, Gill, Matthew S., Hughes, Robert E., Holden‐Dye, Lindy, Lithgow, Gordon J.
Published in Aging cell (01.10.2016)
Published in Aging cell (01.10.2016)
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Human Genetics in Rheumatoid Arthritis Guides a High-Throughput Drug Screen of the CD40 Signaling Pathway
Li, Gang, Diogo, Dorothée, Wu, Di, Spoonamore, Jim, Dancik, Vlado, Franke, Lude, Kurreeman, Fina, Rossin, Elizabeth J., Duclos, Grant, Hartland, Cathy, Zhou, Xuezhong, Li, Kejie, Liu, Jun, De Jager, Philip L., Siminovitch, Katherine A., Zhernakova, Alexandra, Raychaudhuri, Soumya, Bowes, John, Eyre, Steve, Padyukov, Leonid, Gregersen, Peter K., Worthington, Jane, Gupta, Namrata, Clemons, Paul A., Stahl, Eli, Tolliday, Nicola, Plenge, Robert M.
Published in PLoS genetics (01.05.2013)
Published in PLoS genetics (01.05.2013)
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Small molecule inhibitors of anthrax edema factor
Jiao, Guan-Sheng, Kim, Seongjin, Moayeri, Mahtab, Thai, April, Cregar-Hernandez, Lynne, McKasson, Linda, O'Malley, Sean, Leppla, Stephen H., Johnson, Alan T.
Published in Bioorganic & medicinal chemistry letters (15.01.2018)
Published in Bioorganic & medicinal chemistry letters (15.01.2018)
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