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The Synthesis and Biological Evaluation of 2-(1H-Indol-3-yl)quinazolin-4(3H)-One Derivatives
Mendogralo, Elena Y., Nesterova, Larisa Y., Nasibullina, Ekaterina R., Shcherbakov, Roman O., Tkachenko, Alexander G., Sidorov, Roman Y., Sukonnikov, Maxim A., Skvortsov, Dmitry A., Uchuskin, Maxim G.
Published in Molecules (Basel, Switzerland) (11.07.2023)
Published in Molecules (Basel, Switzerland) (11.07.2023)
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Synthesis and Biological Evaluation of Novel Dispiro-Indolinones with Anticancer Activity
Ivanenkov, Yan A., Kukushkin, Maxim E., Beloglazkina, Anastasia A., Shafikov, Radik R., Barashkin, Alexander A., Ayginin, Andrey A., Serebryakova, Marina S., Majouga, Alexander G., Skvortsov, Dmitry A., Tafeenko, Viktor A., Beloglazkina, Elena K.
Published in Molecules (Basel, Switzerland) (30.01.2023)
Published in Molecules (Basel, Switzerland) (30.01.2023)
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[4+2]-Cycloaddition to 5-Methylidene-Hydantoins and 5-Methylidene-2-Thiohydantoins in the Synthesis of Spiro-2-Chalcogenimidazolones
Shybanov, Dmitry E., Kukushkin, Maxim E., Hrytseniuk, Yanislav S., Grishin, Yuri K., Roznyatovsky, Vitaly A., Tafeenko, Viktor A., Skvortsov, Dmitry A., Zyk, Nikolai V., Beloglazkina, Elena K.
Published in International journal of molecular sciences (01.03.2023)
Published in International journal of molecular sciences (01.03.2023)
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Amicoumacin A induces cancer cell death by targeting the eukaryotic ribosome
Prokhorova, Irina V., Akulich, Kseniya A., Makeeva, Desislava S., Osterman, Ilya A., Skvortsov, Dmitry A., Sergiev, Petr V., Dontsova, Olga A., Yusupova, Gulnara, Yusupov, Marat M., Dmitriev, Sergey E.
Published in Scientific reports (14.06.2016)
Published in Scientific reports (14.06.2016)
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Verubulin (Azixa) Analogues with Increased Saturation: Synthesis, SAR and Encapsulation in Biocompatible Nanocontainers Based on Ca2+ or Mg2+ Cross-Linked Alginate
Sedenkova, Kseniya N., Leschukov, Denis N., Grishin, Yuri K., Zefirov, Nikolay A., Gracheva, Yulia A., Skvortsov, Dmitry A., Hrytseniuk, Yanislav S., Vasilyeva, Lilja A., Spirkova, Elena A., Shevtsov, Pavel N., Shevtsova, Elena F., Lukmanova, Alina R., Spiridonov, Vasily V., Markova, Alina A., Nguyen, Minh T., Shtil, Alexander A., Zefirova, Olga N., Yaroslavov, Alexander A., Milaeva, Elena R., Averina, Elena B.
Published in Pharmaceuticals (Basel, Switzerland) (21.10.2023)
Published in Pharmaceuticals (Basel, Switzerland) (21.10.2023)
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Optimization of the dipeptide motifs in the PSMA ligands linker structure: synthesis and in vitro evaluation
Uspenskaya, Anastasiia A., Nimenko, Ekaterina A., Shafikov, Radik R., Zyk, Nikolay Y., Evteev, Sergei A., Dashkova, Natalia S., Ivanenkov, Yan A., Majouga, Alexander G., Skvortsov, Dmitry A., Garanina, Anastasiia S., Beloglazkina, Elena K., Machulkin, Aleksei E.
Published in Medicinal chemistry research (01.01.2023)
Published in Medicinal chemistry research (01.01.2023)
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Triphenilphosphonium Analogs of Chloramphenicol as Dual-Acting Antimicrobial and Antiproliferating Agents
Pavlova, Julia A., Khairullina, Zimfira Z., Tereshchenkov, Andrey G., Nazarov, Pavel A., Lukianov, Dmitrii A., Volynkina, Inna A., Skvortsov, Dmitry A., Makarov, Gennady I., Abad, Etna, Murayama, Somay Y., Kajiwara, Susumu, Paleskava, Alena, Konevega, Andrey L., Antonenko, Yuri N., Lyakhovich, Alex, Osterman, Ilya A., Bogdanov, Alexey A., Sumbatyan, Natalia V.
Published in Antibiotics (Basel) (23.04.2021)
Published in Antibiotics (Basel) (23.04.2021)
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Growth Hormone, Insulin-Like Growth Factor-1, Insulin Resistance, and Leukocyte Telomere Length as Determinants of Arterial Aging in Subjects Free of Cardiovascular Diseases
Strazhesko, Irina D., Tkacheva, Olga N., Akasheva, Dariga U., Dudinskaya, Ekaterina N., Plokhova, Ekaterina V., Pykhtina, Valentina S., Kruglikova, Anna S., Brailova, Natalia V., Sharashkina, Natalia V., Kashtanova, Daria A., Isaykina, Olesya Y., Pokrovskaya, Mariya S., Vygodin, Vladimir A., Ozerova, Irina N., Skvortsov, Dmitry A., Boytsov, Sergey A.
Published in Frontiers in genetics (15.12.2017)
Published in Frontiers in genetics (15.12.2017)
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Modern Collapse Therapy for Pulmonary Tuberculosis
Krasnov, Denis V, Skluev, Sergey V, Petrova, Yana K, Skvortsov, Dmitry A, Krasnov, Vladimir A, Felker, Irina G, Grischenko, Nikolay
Published in Thoracic surgery clinics (01.02.2019)
Published in Thoracic surgery clinics (01.02.2019)
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Nucleophilic Ring Opening of Donor–Acceptor Cyclopropanes with the Cyanate Ion: Access to Spiro[pyrrolidone-3,3′-oxindoles]
Zaytsev, Sergey V, Ivanov, Konstantin L, Skvortsov, Dmitry A, Bezzubov, Stanislav I, Melnikov, Mikhail Ya, Budynina, Ekaterina M
Published in Journal of organic chemistry (03.08.2018)
Published in Journal of organic chemistry (03.08.2018)
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Tetracenomycin X inhibits translation by binding within the ribosomal exit tunnel
Osterman, Ilya A., Wieland, Maximiliane, Maviza, Tinashe P., Lashkevich, Kseniya A., Lukianov, Dmitrii A., Komarova, Ekaterina S., Zakalyukina, Yuliya V., Buschauer, Robert, Shiriaev, Dmitrii I., Leyn, Semen A., Zlamal, Jaime E., Biryukov, Mikhail V., Skvortsov, Dmitry A., Tashlitsky, Vadim N., Polshakov, Vladimir I., Cheng, Jingdong, Polikanov, Yury S., Bogdanov, Alexey A., Osterman, Andrei L., Dmitriev, Sergey E., Beckmann, Roland, Dontsova, Olga A., Wilson, Daniel N., Sergiev, Petr V.
Published in Nature chemical biology (01.10.2020)
Published in Nature chemical biology (01.10.2020)
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A Route to (Het)arene-Annulated Pyrrolo[1,2‑d][1,4]diazepines via the Expanded Intramolecular Paal–Knorr Reaction: Nitro Group and Furan Ring as Equivalents of Amino Group and 1,4-Diketone
Zelina, Elena Y, Nevolina, Tatyana A, Skvortsov, Dmitry A, Trushkov, Igor V, Uchuskin, Maxim G
Published in Journal of organic chemistry (01.11.2019)
Published in Journal of organic chemistry (01.11.2019)
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Electrochemical Detection of a Novel Pt(IV) Prodrug with the Metronidazole Axial Ligand in the Hypoxic Area
Spector, Daniil V., Erofeev, Alexander S., Gorelkin, Petr V., Vaneev, Alexander N., Akasov, Roman A., Ul’yanovskiy, Nikolay V., Nikitina, Vita N., Semkina, Alevtina S., Vlasova, Kseniya Yu, Soldatov, Mikhail A., Trigub, Alexander L., Skvortsov, Dmitry A., Finko, Alexander V., Zyk, Nikolay V., Sakharov, Dmitry A., Majouga, Alexander G., Beloglazkina, Elena K., Krasnovskaya, Olga O.
Published in Inorganic chemistry (19.09.2022)
Published in Inorganic chemistry (19.09.2022)
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Coculture‐Based Screening Revealed Selective Cytostatic Effects of Pyrazol–Azepinoindoles
Skvortsov, Dmitry A., Zhirkina, Irina V., Ipatova, Daria A., Vasilyeva, Lilya A., Ivanenkov, Yan A., Rubtsova, Maria P., Kartsev, Victor G., Sergiev, Petr V., Dontsova, Olga A.
Published in ChemMedChem (17.06.2025)
Published in ChemMedChem (17.06.2025)
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Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate
Machulkin, Aleksei E, Uspenskaya, Anastasia A, Zyk, Nikolay U, Nimenko, Ekaterina A, Ber, Anton P, Petrov, Stanislav A, Polshakov, Vladimir I, Shafikov, Radik R, Skvortsov, Dmitry A, Plotnikova, Ekaterina A, Pankratov, Andrei A, Smirnova, Galina B, Borisova, Yulia A, Pokrovsky, Vadim S, Kolmogorov, Vasilii S, Vaneev, Alexander N, Khudyakov, Alexander D, Chepikova, Olga E, Kovalev, Sergey, Zamyatnin Jr, Andrey A, Erofeev, Alexander, Gorelkin, Petr, Beloglazkina, Elena K, Zyk, Nikolay V, Khazanova, Elena S, Majouga, Alexander G
Published in Journal of medicinal chemistry (09.12.2021)
Published in Journal of medicinal chemistry (09.12.2021)
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A General Synthetic Route to Isomeric Pyrrolo[1,2‑x][1,4]diazepinones
Zelina, Elena Y, Nevolina, Tatyana A, Sorotskaja, Ludmila N, Skvortsov, Dmitry A, Trushkov, Igor V, Uchuskin, Maxim G
Published in Journal of organic chemistry (05.10.2018)
Published in Journal of organic chemistry (05.10.2018)
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Novel Copper-Containing Cytotoxic Agents Based on 2‑Thioxoimidazolones
Krasnovskaya, Olga O, Guk, Dmitry A, Naumov, Alexey E, Nikitina, Vita N, Semkina, Alevtina S, Vlasova, Kseniya Yu, Pokrovsky, Vadim, Ryabaya, Oksana O, Karshieva, Saida S, Skvortsov, Dmitry A, Zhirkina, Irina V, Shafikov, Radik R, Gorelkin, Petr V, Vaneev, Alexander N, Erofeev, Alexander S, Mazur, Dmitrii M, Tafeenko, Viktor A, Pergushov, Vladimir I, Melnikov, Mikhail Ya, Soldatov, Mikhail A, Shapovalov, Victor V, Soldatov, Alexander V, Akasov, Roman. A, Gerasimov, Vasily M, Sakharov, Dmitry A, Moiseeva, Anna A, Zyk, Nikolay V, Beloglazkina, Elena K, Majouga, Alexander G
Published in Journal of medicinal chemistry (12.11.2020)
Published in Journal of medicinal chemistry (12.11.2020)
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PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation
Machulkin, Aleksei E., Uspenskaya, Anastasia A., Zyk, Nikolay Y., Nimenko, Ekaterina A., Ber, Anton P., Petrov, Stanislav A., Shafikov, Radik R., Skvortsov, Dmitry A., Smirnova, Galina B., Borisova, Yulia A., Pokrovsky, Vadim S., Kolmogorov, Vasilii S., Vaneev, Alexander N., Ivanenkov, Yan A., Khudyakov, Alexander D., Kovalev, Sergei V., Erofeev, Alexander S., Gorelkin, Petr V., Beloglazkina, Elena K., Zyk, Nikolay V., Khazanova, Elena S., Majouga, Alexander G.
Published in European journal of medicinal chemistry (05.01.2022)
Published in European journal of medicinal chemistry (05.01.2022)
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Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom
Zyk, Nikolai Y., Ber, Anton P., Nimenko, Ekaterina A., Shafikov, Radik R., Evteev, Sergei A., Petrov, Stanislav A., Uspenskaya, Anastasia A., Dashkova, Natalia S., Ivanenkov, Yan A., Skvortsov, Dmitry A., Beloglazkina, Elena K., Majouga, Alexander G., Machulkin, Aleksei E.
Published in Bioorganic & medicinal chemistry letters (01.09.2022)
Published in Bioorganic & medicinal chemistry letters (01.09.2022)
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