Synthesis and Structure-Activity Relationships of Phenylenebis(methylene)-Linked Bis-Tetraazamacrocycles That Inhibit HIV Replication. Effects of Macrocyclic Ring Size and Substituents on the Aromatic Linker
Bridger, Gary J, Skerlj, Renato T, Thornton, David, Padmanabhan, Sreenivasan, Martellucci, Stephen A, Henson, Geoffrey W, Abrams, Michael J, Yamamoto, Naohiko, Vreese, Karen De
Published in Journal of medicinal chemistry (01.01.1995)
Published in Journal of medicinal chemistry (01.01.1995)
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Molecular mechanism of AMD3100 antagonism in the CXCR4 receptor: transfer of binding site to the CXCR3 receptor
Rosenkilde, Mette M, Gerlach, Lars-Ole, Jakobsen, Janus S, Skerlj, Renato T, Bridger, Gary J, Schwartz, Thue W
Published in The Journal of biological chemistry (23.01.2004)
Published in The Journal of biological chemistry (23.01.2004)
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Molecular Interactions of Cyclam and Bicyclam Non-peptide Antagonists with the CXCR4 Chemokine Receptor
Gerlach, L O, Skerlj, R T, Bridger, G J, Schwartz, T W
Published in The Journal of biological chemistry (27.04.2001)
Published in The Journal of biological chemistry (27.04.2001)
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Synthesis and Structure−Activity Relationships of Phenylenebis(methylene)- Linked Bis-azamacrocycles That Inhibit HIV-1 and HIV-2 Replication by Antagonism of the Chemokine Receptor CXCR4
Bridger, Gary J, Skerlj, Renato T, Padmanabhan, Sreenivasan, Martellucci, Stephen A, Henson, Geoffrey W, Struyf, Sofie, Witvrouw, Myriam, Schols, Dominique, De Clercq, Erik
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Activity of Different Bicyclam Derivatives against Human Immunodeficiency Virus Depends on Their Interaction with the CXCR4 Chemokine Receptor
Esté, J A, Cabrera, C, De Clercq, E, Struyf, S, Van Damme, J, Bridger, G, Skerlj, R T, Abrams, M J, Henson, G, Gutierrez, A, Clotet, B, Schols, D
Published in Molecular pharmacology (01.01.1999)
Published in Molecular pharmacology (01.01.1999)
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The antiviral activity of the CXCR4 antagonist AMD3100 is independent of the cytokine-induced CXCR4/HIV coreceptor expression level
Princen, Katrien, Hatse, Sigrid, Vermeire, Kurt, Bridger, Gary J, Skerlj, Renato T, De Clercq, Erik, Schols, Dominique
Published in AIDS research and human retroviruses (01.12.2003)
Published in AIDS research and human retroviruses (01.12.2003)
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Convenient Synthesis of 5,6,7,8-Tetrahydroquinolin-8-ylamine and 6,7-Dihydro-5H-quinolin-8-one
McEachern, E. J., Yang, W., Chen, G., Skerlj, R. T., Bridger, G. J.
Published in Synthetic communications (01.01.2003)
Published in Synthetic communications (01.01.2003)
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Synthesis and Structure−Activity Relationships of Phenylenebis(methylene)- Linked Bis-tetraazamacrocycles That Inhibit Human Immunodeficiency Virus Replication. 2. Effect of Heteroaromatic Linkers on the Activity of Bicyclams
Bridger, Gary J, Skerlj, Renato T, Padmanabhan, Sreenivasan, Martellucci, Stephen A, Henson, Geoffrey W, Abrams, Michael J, Joao, Heidi C, Witvrouw, Myriam, De Vreese, Karen, Pauwels, Rudi, De Clercq, Erik
Published in Journal of medicinal chemistry (05.01.1996)
Published in Journal of medicinal chemistry (05.01.1996)
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AMD3465, a monomacrocyclic CXCR4 antagonist and potent HIV entry inhibitor
Hatse, Sigrid, Princen, Katrien, Clercq, Erik De, Rosenkilde, Mette M., Schwartz, Thue W., Hernandez-Abad, Pedro E., Skerlj, Renato T., Bridger, Gary J., Schols, Dominique
Published in Biochemical pharmacology (01.09.2005)
Published in Biochemical pharmacology (01.09.2005)
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Synthesis and structure-activity relationships of phenylenebis(methylene)-linked bis-azamacrocycles that inhibit HIV-1 and HIV-8 replication by antagonism of the chemokine receptor CXCR4
Bridger, GJ, Skerlj, RT, Padmanabhan, S, Martellucci, SA, Henson, GW, Struyf, S, Witvrouw, M, Schols, D, De Clercq, E
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Journal Article
Convenient Synthesis of 5,6,7,8-Tetrahydroquinolin-8-ylamine and 6,7-Dihydro-5 H -quinolin-8-one
McEachern, E. J., Yang, W., Chen, G., Skerlj, R. T., Bridger, G. J.
Published in Synthetic communications (01.10.2003)
Published in Synthetic communications (01.10.2003)
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REGIOSELECTIVE GERMYL-STANNYLATION OF ALPHA,BETA-ACETYLENIC ESTERS
PIERS, E, SKERLJ, RT
Published in Journal of the Chemical Society. Chemical communications (01.07.1987)
Published in Journal of the Chemical Society. Chemical communications (01.07.1987)
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