Amphetamines, new psychoactive drugs and the monoamine transporter cycle
Sitte, Harald H, Freissmuth, Michael
Published in Trends in pharmacological sciences (Regular ed.) (01.01.2015)
Published in Trends in pharmacological sciences (Regular ed.) (01.01.2015)
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Shock Wave Treatment Enhances Cell Proliferation and Improves Wound Healing by ATP Release-coupled Extracellular Signal-regulated Kinase (ERK) Activation
Weihs, Anna M., Fuchs, Christiane, Teuschl, Andreas H., Hartinger, Joachim, Slezak, Paul, Mittermayr, Rainer, Redl, Heinz, Junger, Wolfgang G., Sitte, Harald H., Rünzler, Dominik
Published in The Journal of biological chemistry (26.09.2014)
Published in The Journal of biological chemistry (26.09.2014)
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Structural basis of organic cation transporter-3 inhibition
Khanppnavar, Basavraj, Maier, Julian, Herborg, Freja, Gradisch, Ralph, Lazzarin, Erika, Luethi, Dino, Yang, Jae-Won, Qi, Chao, Holy, Marion, Jäntsch, Kathrin, Kudlacek, Oliver, Schicker, Klaus, Werge, Thomas, Gether, Ulrik, Stockner, Thomas, Korkhov, Volodymyr M, Sitte, Harald H
Published in Nature communications (07.11.2022)
Published in Nature communications (07.11.2022)
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Powerful Cocaine-Like Actions of 3,4-Methylenedioxypyrovalerone (MDPV), a Principal Constituent of Psychoactive 'Bath Salts' Products
BAUMANN, Michael H, PARTILLA, John S, BRANDT, Simon D, TELLA, Srihari R, COZZI, Nicholas V, SCHINDLER, Charles W, LEHNER, Kurt R, THORNDIKE, Eric B, HOFFMAN, Alexander F, HOLY, Marion, ROTHMAN, Richard B, GOLDBERG, Steven R, LUPICA, Carl R, SITTE, Harald H
Published in Neuropsychopharmacology (New York, N.Y.) (01.03.2013)
Published in Neuropsychopharmacology (New York, N.Y.) (01.03.2013)
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Ethanol inhibits dopamine uptake via organic cation transporter 3: Implications for ethanol and cocaine co-abuse
Clauss, N J, Mayer, F P, Owens, W A, Vitela, M, Clarke, K M, Bowman, M A, Horton, R E, Gründemann, D, Schmid, D, Holy, M, Gould, G G, Koek, W, Sitte, H H, Daws, L C
Published in Molecular psychiatry (01.07.2023)
Published in Molecular psychiatry (01.07.2023)
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An unsuspected role for organic cation transporter 3 in the actions of amphetamine
Mayer, Felix P, Schmid, Diethart, Owens, W Anthony, Gould, Georgianna G, Apuschkin, Mia, Kudlacek, Oliver, Salzer, Isabella, Boehm, Stefan, Chiba, Peter, Williams, Piper H, Wu, Hsiao-Huei, Gether, Ulrik, Koek, Wouter, Daws, Lynette C, Sitte, Harald H
Published in Neuropsychopharmacology (New York, N.Y.) (01.11.2018)
Published in Neuropsychopharmacology (New York, N.Y.) (01.11.2018)
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Cross-sectional survey and Bayesian network model analysis of traditional Chinese medicine in Austria: investigating public awareness, usage determinants and perception of scientific support
Eigenschink, Michael, Bellach, Luise, Leonard, Sebastian, Dablander, Tom Eric, Maier, Julian, Dablander, Fabian, Sitte, Harald H
Published in BMJ open (02.03.2023)
Published in BMJ open (02.03.2023)
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Globus pallidus dopamine and Parkinson motor subtypes: clinical and brain biochemical correlation
Rajput, A H, Sitte, H H, Rajput, A, Fenton, M E, Pifl, C, Hornykiewicz, O
Published in Neurology (15.04.2008)
Published in Neurology (15.04.2008)
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Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors
Gradisch, Ralph, Schlögl, Katharina, Lazzarin, Erika, Niello, Marco, Maier, Julian, Mayer, Felix P, Alves da Silva, Leticia, Skopec, Sophie M C, Blakely, Randy D, Sitte, Harald H, Mihovilovic, Marko D, Stockner, Thomas
Published in Nature communications (10.01.2024)
Published in Nature communications (10.01.2024)
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Phase I metabolites of mephedrone display biological activity as substrates at monoamine transporters
Mayer, F P, Wimmer, L, Dillon‐Carter, O, Partilla, J S, Burchardt, N V, Mihovilovic, M D, Baumann, M H, Sitte, H H
Published in British journal of pharmacology (01.09.2016)
Published in British journal of pharmacology (01.09.2016)
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A transporter’s doom or destiny: SLC6A1 in health and disease, novel molecular targets and emerging therapeutic prospects
Shah, Nikita, Kasture, Ameya S., Fischer, Florian P., Sitte, Harald H., Hummel, Thomas, Sucic, Sonja
Published in Frontiers in molecular neuroscience (29.08.2024)
Published in Frontiers in molecular neuroscience (29.08.2024)
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Interaction Profiles of Central Nervous System Active Drugs at Human Organic Cation Transporters 1-3 and Human Plasma Membrane Monoamine Transporter
Angenoorth, Thomas J F, Stankovic, Stevan, Niello, Marco, Holy, Marion, Brandt, Simon D, Sitte, Harald H, Maier, Julian
Published in International journal of molecular sciences (30.11.2021)
Published in International journal of molecular sciences (30.11.2021)
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Role of amino terminal substitutions in the pharmacological, rewarding and psychostimulant profiles of novel synthetic cathinones
Duart-Castells, L., Nadal-Gratacós, N., Muralter, M., Puster, B., Berzosa, X., Estrada-Tejedor, R., Niello, M., Bhat, S., Pubill, D., Camarasa, J., Sitte, H.H., Escubedo, E., López-Arnau, R.
Published in Neuropharmacology (15.03.2021)
Published in Neuropharmacology (15.03.2021)
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Dual Action of Zn2+ on the Transport Cycle of the Dopamine Transporter
Li, Yang, Hasenhuetl, Peter S., Schicker, Klaus, Sitte, Harald H., Freissmuth, Michael, Sandtner, Walter
Published in The Journal of biological chemistry (25.12.2015)
Published in The Journal of biological chemistry (25.12.2015)
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Interactions of calmodulin kinase II with the dopamine transporter facilitate cocaine-induced enhancement of evoked dopamine release
Keighron, Jacqueline D, Bonaventura, Jordi, Li, Yang, Yang, Jae-Won, DeMarco, Emily M, Hersey, Melinda, Cao, Jianjing, Sandtner, Walter, Michaelides, Michael, Sitte, Harald H, Newman, Amy Hauck, Tanda, Gianluigi
Published in Translational psychiatry (13.06.2023)
Published in Translational psychiatry (13.06.2023)
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Transition metal ion FRET uncovers K + regulation of a neurotransmitter/sodium symporter
Billesbølle, Christian B, Mortensen, Jonas S, Sohail, Azmat, Schmidt, Solveig G, Shi, Lei, Sitte, Harald H, Gether, Ulrik, Loland, Claus J
Published in Nature communications (28.09.2016)
Published in Nature communications (28.09.2016)
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The ugly side of amphetamines: short- and long-term toxicity of 3,4-methylenedioxymethamphetamine (MDMA, ‘Ecstasy’), methamphetamine and d-amphetamine
Steinkellner, Thomas, Freissmuth, Michael, Sitte, Harald H., Montgomery, Therese
Published in Biological chemistry (01.01.2011)
Published in Biological chemistry (01.01.2011)
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The Serotonin Transporter Is an Exclusive Client of the Coat Protein Complex II (COPII) Component SEC24C
Sucic, Sonja, El-Kasaby, Ali, Kudlacek, Oliver, Sarker, Subhodeep, Sitte, Harald H., Marin, Philippe, Freissmuth, Michael
Published in The Journal of biological chemistry (06.05.2011)
Published in The Journal of biological chemistry (06.05.2011)
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Dopamine Transporter Phosphorylation Site Threonine 53 Regulates Substrate Reuptake and Amphetamine-stimulated Efflux
Foster, James D., Yang, Jae-Won, Moritz, Amy E., ChallaSivaKanaka, Sathyavathi, Smith, Margaret A., Holy, Marion, Wilebski, Kyle, Sitte, Harald H., Vaughan, Roxanne A.
Published in The Journal of biological chemistry (24.08.2012)
Published in The Journal of biological chemistry (24.08.2012)
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