Cytochrome P450 reaction-phenotyping: an industrial perspective
Zhang, Hongjian, Davis, Carl D, Sinz, Michael W, Rodrigues, A David
Published in Expert opinion on drug metabolism & toxicology (01.10.2007)
Published in Expert opinion on drug metabolism & toxicology (01.10.2007)
Get more information
Journal Article
Comparative Effects of Thiazolidinediones on in Vitro P450 Enzyme Induction and Inhibition
SAHI, Jasminder, BLACK, Christopher B, HAMILTON, Geraldine A, XIANXIAN ZHENG, JOLLEY, Summer, ROSE, Kelly A, GILBERT, Darryl, LECLUYSE, Edward L, SINZ, Michael W
Published in Drug metabolism and disposition (01.04.2003)
Published in Drug metabolism and disposition (01.04.2003)
Get full text
Journal Article
Inactivation of Cytochrome P450 3A4 by Bergamottin, a Component of Grapefruit Juice
He, Kan, Iyer, Krishna R, Hayes, Roger N, Sinz, Michael W, Woolf, Thomas F, Hollenberg, Paul F
Published in Chemical research in toxicology (01.04.1998)
Published in Chemical research in toxicology (01.04.1998)
Get full text
Journal Article
Animal models of xenobiotic receptors in drug metabolism and diseases
Gong, Haibiao, Sinz, Michael W, Feng, Yan, Chen, Taosheng, Venkataramanan, Raman, Xie, Wen
Published in Methods in enzymology (2005)
Published in Methods in enzymology (2005)
Get more information
Journal Article
Fluorine Substitution Can Block CYP3A4 Metabolism-Dependent Inhibition: Identification of (S)-N-[1-(4-Fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an Orally Bioavailable KCNQ2 Opener Devoid of CYP3A4 Metabolism-Dependent Inhibition
Wu, Yong-Jin, Davis, Carl D, Dworetzky, Steven, Fitzpatrick, William C, Harden, David, He, Huan, Knox, Ronald J, Newton, Amy E, Philip, Thomas, Polson, Craig, Sivarao, Digavalli V, Sun, Li-Qiang, Tertyshnikova, Svetlana, Weaver, David, Yeola, Suresh, Zoeckler, Mary, Sinz, Michael W
Published in Journal of medicinal chemistry (28.08.2003)
Published in Journal of medicinal chemistry (28.08.2003)
Get full text
Journal Article
(S)-N-[1-(3-Morpholin-4-ylphenyl)ethyl]-3phenylacrylamide: An orally bioavailable KCNQ2 opener with significant activity in a cortical spreading depression model of migraine
Wu, YJ, Boissard, CG, Greco, C, Gribkoff, VK, Harden, DG, He, H, L'Heureux, A, Kang, SH, Kinney, GG, Knox, RJ, Natale, J, Newton, AE, Lehtinen-Oboma, S, Sinz, MW, Sivarao, DV, Starrett, JE, Sun, LQ, Tertyshnikova, S, Thompson, MW, Weaver, D, Wong, HS, Zhang, L, Dworetzky, SL
Published in Journal of medicinal chemistry (17.07.2003)
Published in Journal of medicinal chemistry (17.07.2003)
Get full text
Journal Article
Metabolism and transporter-mediated drug–drug interactions of the endothelin-A receptor antagonist CI-1034
Sahi, Jasminder, Sinz, Michael W., Campbell, Scott, Mireles, Rouchelle, Zheng, Xianxian, Rose, Kelly A., Raeissi, Shamsi, Hashim, Muhammed F., Ye, Yuyang, de Morais, Sonia M., Black, Christopher, Tugnait, Meera, Keller, Laurence H.
Published in Chemico-biological interactions (01.02.2006)
Published in Chemico-biological interactions (01.02.2006)
Get full text
Journal Article
The Effect of Troglitazone Biliary Excretion on Metabolite Distribution and Cholestasis in Transporter-Deficient Rats
KOSTRUBSKY, Vsevolod E, VORE, Mary, KINDT, Erick, BURLIEGH, James, ROGERS, Karen, PETER, Gregory, ALTROGGE, Douglas, SINZ, Michael W
Published in Drug metabolism and disposition (01.12.2001)
Get full text
Published in Drug metabolism and disposition (01.12.2001)
Journal Article
Distribution of tacrine and metabolites in rat brain and plasma after single- and multiple-dose regimens. Evidence for accumulation of tacrine in brain tissue
McNally, W P, Pool, W F, Sinz, M W, Dehart, P, Ortwine, D F, Huang, C C, Chang, T, Woolf, T F
Published in Drug metabolism and disposition (01.06.1996)
Get more information
Published in Drug metabolism and disposition (01.06.1996)
Journal Article
Multiple-model evaluation of absorption of a tachykinin receptor antagonist
Chan, O.Helen, Sinz, Michael W., Stewart, Barbra H.
Published in Advanced drug delivery reviews (15.01.1997)
Published in Advanced drug delivery reviews (15.01.1997)
Get full text
Journal Article