Discovery and characterization of a specific inhibitor of serine-threonine kinase cyclin-dependent kinase-like 5 (CDKL5) demonstrates role in hippocampal CA1 physiology
Castano, Anna, Silvestre, Margaux, Wells, Carrow I, Sanderson, Jennifer L, Ferrer, Carla A, Ong, Han Wee, Lang, Yi, Richardson, William, Silvaroli, Josie A, Bashore, Frances M, Smith, Jeffery L, Genereux, Isabelle M, Dempster, Kelvin, Drewry, David H, Pabla, Navlot S, Bullock, Alex N, Benke, Tim A, Ultanir, Sila K, Axtman, Alison D
Published in eLife (25.07.2023)
Published in eLife (25.07.2023)
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Cell type-specific expression, regulation and compensation of CDKL5 activity in mouse brain
Silvestre, Margaux, Dempster, Kelvin, Mihaylov, Simeon R, Claxton, Suzanne, Ultanir, Sila K
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Published in Molecular psychiatry (08.02.2024)
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Pandemic peak SARS-CoV-2 infection and seroconversion rates in London frontline health-care workers
Houlihan, Catherine F, Kelly, Gavin, Spyer, Moira J, Nastouli, Eleni, Allen, Zoe, Ambrose, Karen, Barns-Jenkins, Caitlin, Basu, Souradeep, Buck, Michael D, Cardoso, Ana, Carter, Nick, Carvalho, Luiz, Chen, Qu, Churchward, Laura, Cottrell, Sally, Davison, Dara, Debaisieux, Solene, Diaz-Romero, Monica, Diring, Jessica, Driscoll, Paul C, Edwards, Amelia, Evangelopoulos, Dimitrios, Ferron, Aaron, Fitz, Dan, Fleming, James, Gaiba, Alessandra, Goldstone, Robert, Halldorsson, Steinar, Hoskins, Beth, Houlihan, Catherine F, Hoyle, Jacqueline, Htun, Mint R, Hubank, Michael, Hughes, Deborah, Instrell, Rachael, Jamal-Hanjani, Mariam, Johnson, Mark, Kotzampaltiris, Paul, Kousis, Konstantinos, Kucharska, Ania, Lee, Stacey-Ann, Lu, Wei-Ting, MacRae, James I, McCoy, Laura E, Minutti, Carlos M, Molina-Arcas, Miriam, Moore, David, Moraiti, Anastasia, Nutan, Savita, Oedekoven, Caroline, O'Neill, Olga, Osborne, Neil, Papayannopoulos, Venizelos, Patel, Yogen, Paun, Oana, Perez Caballero, Ana, Perez-Lloret, Jimena, Pollitt, Marc, Shah Punatar, Rajvee, Ramaprasad, Abhinay, Richardson, Kayleigh, Ridewood, Sophie, Rossi, Alice, Rowan, Andrew, Sahai, Erik, Sawyer, Chelsea, Spyer, Moira J, Steel, Louisa, Strange, Amy, Swanton, Charles, Tautz-Davis, Zoe H, Taylor, Gunes, Toolan-Kerr, Patrick, Torelli, Francesca, Toteva, Tea, Ule, Jernej, Wenman, Catharina, Williams, Matthew J, Wright, Joshua, Xiang, Zheng, Matthews, Rebecca, Severn, Abigail, Michie, Susan, Shahmanesh, Maryam, Lukha, Hinal, Davies, Claudia, Williams, Bethany, Riddell, Andrew, Bartolovic, Kerol, Russell, Emma, Carr, Lotte, Crayton, Elise, Meyer, Carly, Vora, Nina, Stoltenberg, Andrea, Byrne, Tom, Gilson, Richard, Kelly, Gavin, Roberts, Fiona, Hatipoglu, Emine
Published in The Lancet (25.07.2020)
Published in The Lancet (25.07.2020)
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Chemical genetic identification of CDKL5 substrates reveals its role in neuronal microtubule dynamics
Baltussen, Lucas L, Negraes, Priscilla D, Silvestre, Margaux, Claxton, Suzanne, Moeskops, Max, Christodoulou, Evangelos, Flynn, Helen R, Snijders, Ambrosius P, Muotri, Alysson R, Ultanir, Sila K
Published in The EMBO journal (14.12.2018)
Published in The EMBO journal (14.12.2018)
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Chemical genetic identification of CDKL 5 substrates reveals its role in neuronal microtubule dynamics
Baltussen, Lucas L, Negraes, Priscilla D, Silvestre, Margaux, Claxton, Suzanne, Moeskops, Max, Christodoulou, Evangelos, Flynn, Helen R, Snijders, Ambrosius P, Muotri, Alysson R, Ultanir, Sila K
Published in The EMBO journal (14.12.2018)
Published in The EMBO journal (14.12.2018)
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Discovery of a Potent and Selective CDKL5/GSK3 Chemical Probe That Is Neuroprotective
Ong, Han Wee, Liang, Yi, Richardson, William, Lowry, Emily R., Wells, Carrow I., Chen, Xiangrong, Silvestre, Margaux, Dempster, Kelvin, Silvaroli, Josie A., Smith, Jeffery L., Wichterle, Hynek, Pabla, Navjot S., Ultanir, Sila K., Bullock, Alex N., Drewry, David H., Axtman, Alison D.
Published in ACS chemical neuroscience (03.05.2023)
Published in ACS chemical neuroscience (03.05.2023)
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A Potent and Selective CDKL5/GSK3 Chemical Probe is Neuroprotective
Ong, Han Wee, Liang, Yi, Richardson, William, Lowry, Emily R, Wells, Carrow I, Chen, Xiangrong, Silvestre, Margaux, Dempster, Kelvin, Silvaroli, Josie A, Smith, Jeffery L, Wichterle, Hynek, Pabla, Navjot S, Ultanir, Sila K, Bullock, Alex N, Drewry, David H, Axtman, Alison D
Published in bioRxiv : the preprint server for biology (10.02.2023)
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Published in bioRxiv : the preprint server for biology (10.02.2023)
Journal Article
A Potent and Selective CDKL5/GSK3 Chemical Probe is Neuroprotective
Han Wee Ong, Liang, Yi, Richardson, William, Lowry, Emily R, Wells, Carrow I, Chen, Xiangrong, Silvestre, Margaux, Dempster, Kelvin, Silvaroli, Josie A, Smith, Jeffery L, Wichterle, Hynek, Pabla, Navjot S, Ultanir, Sila K, Bullock, Alex N, Drewry, David, Alison Donnelly Axtman
Published in bioRxiv (10.02.2023)
Published in bioRxiv (10.02.2023)
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Journal Article
Discovery and characterization of a specific inhibitor of serine-threonine kinase cyclin dependent kinase-like 5 (CDKL5) demonstrates role in hippocampal CA1 physiology
Castano, Anna, Silvestre, Margaux, Wells, Carrow I, Sanderson, Jennifer L, Ferrer, Carla A, Ong, Han Wee, Lang, Yi, Richardson, William, Silvaroli, Josie A, Bashore, Frances M, Smith, Jeffery L, Genereux, Isabelle M, Dempster, Kelvin, Drewry, David H, Pabla, Navlot S, Bullock, Alex N, Benke, Tim A, Ultanir, Sila, Axtman, Alison D
Published in bioRxiv : the preprint server for biology (16.06.2023)
Published in bioRxiv : the preprint server for biology (16.06.2023)
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