Chemical synthesis of tripeptide thioesters for the biotechnological incorporation into the myxobacterial secondary metabolite argyrin via mutasynthesis
Siebert, David C B, Sommer, Roman, Pogorevc, Domen, Hoffmann, Michael, Wenzel, Silke C, Müller, Rolf, Titz, Alexander
Published in Beilstein journal of organic chemistry (05.12.2019)
Published in Beilstein journal of organic chemistry (05.12.2019)
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Journal Article
Molecular tools for GABAA receptors: High affinity ligands for β1-containing subtypes
Simeone, Xenia, Siebert, David C. B., Bampali, Konstantina, Varagic, Zdravko, Treven, Marco, Rehman, Sabah, Pyszkowski, Jakob, Holzinger, Raphael, Steudle, Friederike, Scholze, Petra, Mihovilovic, Marko D., Schnürch, Michael, Ernst, Margot
Published in Scientific reports (18.07.2017)
Published in Scientific reports (18.07.2017)
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Journal Article
SAR-Guided Scoring Function and Mutational Validation Reveal the Binding Mode of CGS-8216 at the α1+/γ2– Benzodiazepine Site
Siebert, David C. B, Wieder, Marcus, Schlener, Lydia, Scholze, Petra, Boresch, Stefan, Langer, Thierry, Schnürch, Michael, Mihovilovic, Marko D, Richter, Lars, Ernst, Margot, Ecker, Gerhard F
Published in Journal of chemical information and modeling (27.08.2018)
Published in Journal of chemical information and modeling (27.08.2018)
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Journal Article
Different Benzodiazepines Bind with Distinct Binding Modes to GABAA Receptors
Elgarf, Alshaimaa A, Siebert, David C. B, Steudle, Friederike, Draxler, Angelika, Li, Guanguan, Huang, Shengming, Cook, James M, Ernst, Margot, Scholze, Petra
Published in ACS chemical biology (17.08.2018)
Published in ACS chemical biology (17.08.2018)
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Journal Article
Different Benzodiazepines Bind with Distinct Binding Modes to GABA A Receptors
Elgarf, Alshaimaa A, Siebert, David C B, Steudle, Friederike, Draxler, Angelika, Li, Guanguan, Huang, Shengming, Cook, James M, Ernst, Margot, Scholze, Petra
Published in ACS chemical biology (17.08.2018)
Published in ACS chemical biology (17.08.2018)
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Journal Article
Towards functional selectivity for α6β3γ2 GABAA receptors: a series of novel pyrazoloquinolinones
Treven, Marco, Siebert, David C B, Holzinger, Raphael, Bampali, Konstantina, Fabjan, Jure, Varagic, Zdravko, Wimmer, Laurin, Steudle, Friederike, Scholze, Petra, Schnürch, Michael, Mihovilovic, Marko D, Ernst, Margot
Published in British journal of pharmacology (01.02.2018)
Published in British journal of pharmacology (01.02.2018)
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Journal Article
Engineered Flumazenil Recognition Site Provides Mechanistic Insight Governing Benzodiazepine Modulation in GABA A Receptors
Siebert, David C B, Bampali, Konstantina, Puthenkalam, Roshan, Varagic, Zdravko, Sarto-Jackson, Isabella, Scholze, Petra, Sieghart, Werner, Mihovilovic, Marko D, Schnürch, Michael, Ernst, Margot
Published in ACS chemical biology (17.08.2018)
Published in ACS chemical biology (17.08.2018)
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Journal Article
Engineered Flumazenil Recognition Site Provides Mechanistic Insight Governing Benzodiazepine Modulation in GABAA Receptors
Siebert, David C. B, Bampali, Konstantina, Puthenkalam, Roshan, Varagic, Zdravko, Sarto-Jackson, Isabella, Scholze, Petra, Sieghart, Werner, Mihovilovic, Marko D, Schnürch, Michael, Ernst, Margot
Published in ACS chemical biology (17.08.2018)
Published in ACS chemical biology (17.08.2018)
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Journal Article
SAR-Guided Scoring Function and Mutational Validation Reveal the Binding Mode of CGS-8216 at the a1+/?2– Benzodiazepine Site
Siebert, David C B, Wieder, Marcus, Schlener, Lydia, Scholze, Petra, Boresch, Stefan, Langer, Thierry, Schnürch, Michael, Mihovilovic, Marko D, Richter, Lars, Ernst, Margot, Ecker, Gerhard F
Published in Journal of chemical information and modeling (27.08.2018)
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Published in Journal of chemical information and modeling (27.08.2018)
Journal Article
Towards functional selectivity for α6β3γ2 GABA A receptors: a series of novel pyrazoloquinolinones
Treven, Marco, Siebert, David C B, Holzinger, Raphael, Bampali, Konstantina, Fabjan, Jure, Varagic, Zdravko, Wimmer, Laurin, Steudle, Friederike, Scholze, Petra, Schnürch, Michael, Mihovilovic, Marko D, Ernst, Margot
Published in British journal of pharmacology (01.02.2018)
Published in British journal of pharmacology (01.02.2018)
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Journal Article
Molecular tools for GABA A receptors: High affinity ligands for β1-containing subtypes
Simeone, Xenia, Siebert, David C B, Bampali, Konstantina, Varagic, Zdravko, Treven, Marco, Rehman, Sabah, Pyszkowski, Jakob, Holzinger, Raphael, Steudle, Friederike, Scholze, Petra, Mihovilovic, Marko D, Schnürch, Michael, Ernst, Margot
Published in Scientific reports (18.07.2017)
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Published in Scientific reports (18.07.2017)
Journal Article